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Past strategies and future directions for identifying AMP-activated protein kinase (AMPK) modulators
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title
Past strategies and future directions for identifying AMP-activated protein kinase (AMPK) modulators
(English)
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PubMed
author name string
Sarah E. Sinnett
series ordinal
1
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Crossref
Jay E. Brenman
series ordinal
2
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stated in
Crossref
language of work or name
English
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stated in
PubMed
publication date
July 2014
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PubMed
published in
Pharmacology & Therapeutics
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PubMed
volume
143
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PubMed
issue
1
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PubMed
page(s)
111-8
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PubMed
cites work
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Structure of the bone morphogenetic protein receptor ALK2 and implications for fibrodysplasia ossificans progressiva
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Structure of mammalian AMPK and its regulation by ADP
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AMPK and PPARdelta agonists are exercise mimetics
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21 March 2017
Structural basis for AMP binding to mammalian AMP-activated protein kinase
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21 March 2017
Fatal congenital heart glycogenosis caused by a recurrent activating R531Q mutation in the gamma 2-subunit of AMP-activated protein kinase (PRKAG2), not by phosphorylase kinase deficiency
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21 March 2017
Role of AMP-activated protein kinase in mechanism of metformin action
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21 March 2017
Mammalian AMP-activated protein kinase subfamily
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AMPK: a target for drugs and natural products with effects on both diabetes and cancer
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21 March 2017
Structural basis of AMPK regulation by small molecule activators
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21 March 2017
X-ray structure of p38α bound to TAK-715: comparison with three classic inhibitors
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21 March 2017
AMP-activated protein kinase undergoes nucleotide-dependent conformational changes
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21 March 2017
Crystallographic studies of the complexes of antiviral protein griffithsin with glucose and N-acetylglucosamine
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AMP-activated protein kinase, a metabolic master switch: possible roles in type 2 diabetes
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21 March 2017
Suppressor of MEK null (SMEK)/protein phosphatase 4 catalytic subunit (PP4C) is a key regulator of hepatic gluconeogenesis
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Dorsomorphin inhibits BMP signals required for embryogenesis and iron metabolism
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7 April 2017
5-aminoimidazole-4-carboxamide ribonucleoside. A specific method for activating AMP-activated protein kinase in intact cells?
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Development of Novel Alkene Oxindole Derivatives As Orally Efficacious AMP-Activated Protein Kinase Activators
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A High Throughput Assay for Discovery of Small Molecules that Bind AMP-activated Protein Kinase (AMPK).
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28 September 2017
AMP is a true physiological regulator of AMP-activated protein kinase by both allosteric activation and enhancing net phosphorylation
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28 September 2017
AMP-Activated Protein Kinase α 2 Isoform Suppression in Primary Breast Cancer Alters AMPK Growth Control and Apoptotic Signaling
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28 September 2017
Exercise, GLUT4, and skeletal muscle glucose uptake
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28 September 2017
Investigational anticoagulants for hematological conditions: a new generation of therapies.
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28 September 2017
AICAR-dependent AMPK activation improves scar formation in the aged heart in a murine model of reperfused myocardial infarction
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28 September 2017
AMP-activated protein kinase: a target for old drugs against diabetes and cancer
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28 September 2017
Identification of a novel de novo mutation associated with PRKAG2 cardiac syndrome and early onset of heart failure
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28 September 2017
AMPKβ subunits: more than just a scaffold in the formation of AMPK complex
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28 September 2017
The dark face of AMPK as an essential tumor promoter
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28 September 2017
LKB1 and AMPK and the cancer-metabolism link - ten years after
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28 September 2017
Function of the master energy regulator adenosine monophosphate-activated protein kinase in stroke
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28 September 2017
AMPK activation by oncogenesis is required to maintain cancer cell proliferation in astrocytic tumors
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28 September 2017
Novel strategies for managing dyslipidemia: treatment beyond statins
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28 September 2017
Iron deficiency causes a shift in AMP-activated protein kinase (AMPK) subunit composition in rat skeletal muscle.
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28 September 2017
Over-expressions of AMPK subunits in ovarian carcinomas with significant clinical implications
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28 September 2017
AMP-activated protein kinase: new regulation, new roles?
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28 September 2017
Redox implications of AMPK-mediated signal transduction beyond energetic clues
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28 September 2017
Regulation of hepatic glucose uptake and storage in vivo
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28 September 2017
Sestrin2 modulates AMPK subunit expression and its response to ionizing radiation in breast cancer cells
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28 September 2017
AMPK isoform expression in the normal and failing hearts
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28 September 2017
AMPK functions as an adenylate charge-regulated protein kinase.
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28 September 2017
Preconditioning induces sustained neuroprotection by downregulation of adenosine 5'-monophosphate-activated protein kinase
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28 September 2017
Introduction to fragment-based drug discovery
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28 September 2017
Improvement of cardiac functions by chronic metformin treatment is associated with enhanced cardiac autophagy in diabetic OVE26 mice
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28 September 2017
Targeting AMPK for cardiac protection: opportunities and challenges
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28 September 2017
Metabolic functions of AMPK: aspects of structure and of natural mutations in the regulatory gamma subunits
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28 September 2017
β-Subunit myristoylation is the gatekeeper for initiating metabolic stress sensing by AMP-activated protein kinase (AMPK)
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28 September 2017
The rational design of a novel potent analogue of the 5′-AMP-activated protein kinase inhibitor compound C with improved selectivity and cellular activity
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28 September 2017
Whole body deletion of AMP-activated protein kinase {beta}2 reduces muscle AMPK activity and exercise capacity.
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28 September 2017
AMPK-dependent repression of hepatic gluconeogenesis via disruption of CREB.CRTC2 complex by orphan nuclear receptor small heterodimer partner.
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28 September 2017
Adenosine monophosphate activated protein kinase inhibition is protective in both sexes after experimental stroke
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28 September 2017
Sunitinib-induced cardiotoxicity is mediated by off-target inhibition of AMP-activated protein kinase
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28 September 2017
Homo-oligomerization and activation of AMP-activated protein kinase are mediated by the kinase domain alphaG-helix.
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28 September 2017
The 5' adenosine monophosphate-activated protein kinase: regulating the ebb and flow of cellular energetics
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28 September 2017
AMPK in Health and Disease
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28 September 2017
Small molecule antagonizes autoinhibition and activates AMP-activated protein kinase in cells
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28 September 2017
Cardiotoxicity associated with tyrosine kinase inhibitor sunitinib
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28 September 2017
Neuroprotective effects of adenosine monophosphate-activated protein kinase inhibition and gene deletion in stroke
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28 September 2017
Mechanism of action of A-769662, a valuable tool for activation of AMP-activated protein kinase.
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28 September 2017
The complement of protein kinases of the microsporidium Encephalitozoon cuniculi in relation to those of Saccharomyces cerevisiae and Schizosaccharomyces pombe
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28 September 2017
Defining the mechanism of activation of AMP-activated protein kinase by the small molecule A-769662, a member of the thienopyridone family.
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28 September 2017
Prodrugs of nucleoside analogues for improved oral absorption and tissue targeting
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28 September 2017
Leptin stimulates fatty acid oxidation and peroxisome proliferator-activated receptor alpha gene expression in mouse C2C12 myoblasts by changing the subcellular localization of the alpha2 form of AMP-activated protein kinase
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28 September 2017
AICAR inhibits adipocyte differentiation in 3T3L1 and restores metabolic alterations in diet-induced obesity mice model
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28 September 2017
Identification and characterization of a small molecule AMPK activator that treats key components of type 2 diabetes and the metabolic syndrome
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28 September 2017
Microarrayed compound screening (microARCS) to identify activators and inhibitors of AMP-activated protein kinase
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28 September 2017
Acute and chronic treatment of ob/ob and db/db mice with AICAR decreases blood glucose concentrations.
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28 September 2017
AMP-activated protein kinase: greater AMP dependence, and preferential nuclear localization, of complexes containing the alpha2 isoform.
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28 September 2017
SU11248 (sunitinib) directly inhibits the activity of mammalian 5'-AMP-activated protein kinase (AMPK).
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31 May 2018
Investigating the mechanism for AMP activation of the AMP-activated protein kinase cascade
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31 May 2018
The 5'-AMP-activated protein kinase gamma3 isoform has a key role in carbohydrate and lipid metabolism in glycolytic skeletal muscle
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31 May 2018
Interaction of mant-adenosine nucleotides and magnesium with kinesin
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31 May 2018
5'-AMP inhibits dephosphorylation, as well as promoting phosphorylation, of the AMP-activated protein kinase. Studies using bacterially expressed human protein phosphatase-2C alpha and native bovine protein phosphatase-2AC.
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31 May 2018
Novel small-molecule AMPK activator orally exerts beneficial effects on diabetic db/db mice.
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28 November 2018
Different expression of the catalytic alpha subunits of the AMP activated protein kinase--an immunohistochemical study in human tissue
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28 November 2018
Thienopyridone drugs are selective activators of AMP-activated protein kinase beta1-containing complexes.
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28 November 2018
Dissecting the role of 5'-AMP for allosteric stimulation, activation, and deactivation of AMP-activated protein kinase.
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retrieved
28 November 2018
Mammalian AMP-activated protein kinase: functional, heterotrimeric complexes by co-expression of subunits in Escherichia coli
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3991011
retrieved
28 November 2018
Predominant alpha2/beta2/gamma3 AMPK activation during exercise in human skeletal muscle
1 reference
stated in
PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/24583089
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Localization of AMP kinase is regulated by stress, cell density, and signaling through the MEK-->ERK1/2 pathway
1 reference
stated in
PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/24583089
retrieved
12 December 2020
based on heuristic
inferred from PubMed ID database lookup
Identifiers
DOI
10.1016/J.PHARMTHERA.2014.02.008
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
4949118
OpenCitations bibliographic resource ID
4949118
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
4949118
PMC publication ID
3991011
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
4949118
PubMed publication ID
24583089
1 reference
stated in
Consolidated OpenCitations Corpus – April 2017
OpenCitations bibliographic resource ID
4949118
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