(Q28536518)

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Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts

scientific article (publication date: 2013)

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scholarly article

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Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts (English)

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David Wifling

2

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author name string

Uwe Nordemann

1

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David Schnell

3

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Günther Bernhardt

4

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Holger Stark

5

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Roland Seifert

6

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Armin Buschauer

7

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publication date

2013

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8

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e73961

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Creative Commons Attribution 4.0 International

2 September 2013

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April 2022 Public Data File from Crossref

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Structural Basis for Inhibition of Mammalian Adenylyl Cyclase by Calcium †

1 reference

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19 March 2017

A potent and selective histamine H4 receptor antagonist with anti-inflammatory properties

1 reference

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19 March 2017

Comparison of human, mouse, rat, and guinea pig histamine H4 receptors reveals substantial pharmacological species variation

1 reference

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19 March 2017

Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

1 reference

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1 reference

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Some quantitative uses of drug antagonists

1 reference

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7 April 2017

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1 reference

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Paradoxical stimulatory effects of the "standard" histamine H4-receptor antagonist JNJ7777120: the H4 receptor joins the club of 7 transmembrane domain receptors exhibiting functional selectivity.

1 reference

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Agonist-biased signaling at the histamine H4 receptor: JNJ7777120 recruits β-arrestin without activating G proteins.

1 reference

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1 reference

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Molecular determinants of ligand binding to H4R species variants

1 reference

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Adenylyl cyclases as innovative therapeutic goals.

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In vitro and in vivo characterization of A-940894: a potent histamine H4 receptor antagonist with anti-inflammatory properties

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Molecular and biochemical pharmacology of the histamine H4 receptor

1 reference

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N(G)-acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.

1 reference

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High constitutive activity and a G-protein-independent high-affinity state of the human histamine H(4)-receptor.

1 reference

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Histamine H4 receptor mediates chemotaxis and calcium mobilization of mast cells

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Cloning and characterization of a novel human histamine receptor

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Cloning, expression, and pharmacological characterization of a novel human histamine receptor.

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Discovery of a novel member of the histamine receptor family

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Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow

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The histamine H4 receptor mediates allergic airway inflammation by regulating the activation of CD4+ T cells.

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Histamine 4 receptor activation induces recruitment of FoxP3+ T cells and inhibits allergic asthma in a murine model.

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The histamine H4 receptor antagonist JNJ7777120 induces increases in the histamine content of the rat conjunctiva

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10.1371/JOURNAL.PONE.0073961

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2013PLoSO...873961N

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