(Q36047851)

English

Novel bis-tetrahydrofuranylurethane-containing nonpeptidic protease inhibitor (PI) UIC-94017 (TMC114) with potent activity against multi-PI-resistant human immunodeficiency virus in vitro.

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14506019%20AND%20SRC:MED&resulttype=core&format=json

19 December 2019

Novel bis-tetrahydrofuranylurethane-containing nonpeptidic protease inhibitor (PI) UIC-94017 (TMC114) with potent activity against multi-PI-resistant human immunodeficiency virus in vitro (English)

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14506019%20AND%20SRC:MED&resulttype=core&format=json

19 December 2019

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3

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19 December 2019

14

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Irene T Weber

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19 December 2019

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Yasuhiro Koh

1

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19 December 2019

Hirotomo Nakata

2

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19 December 2019

Hiromi Ogata

4

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19 December 2019

Geoffrey Bilcer

5

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19 December 2019

Thippeswamy Devasamudram

6

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19 December 2019

John F Kincaid

7

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19 December 2019

Peter Boross

8

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19 December 2019

Yuan-Fang Wang

9

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19 December 2019

Yunfeng Tie

10

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19 December 2019

Patra Volarath

11

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19 December 2019

Laquasha Gaddis

12

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19 December 2019

Robert W Harrison

13

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19 December 2019

Arun K Ghosh

15

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19 December 2019

Hiroaki Mitsuya

16

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19 December 2019

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publication date

1 October 2003

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19 December 2019

number of pages

7

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Antimicrobial Agents and Chemotherapy

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19 December 2019

47

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19 December 2019

10

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19 December 2019

3123-3129

1 reference

Europe PubMed Central

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19 December 2019

SHELXL: high-resolution refinement

1 reference

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2 October 2017

Activities of atazanavir (BMS-232632) against a large panel of human immunodeficiency virus type 1 clinical isolates resistant to one or more approved protease inhibitors

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2 October 2017

Strategies in the design of antiviral drugs

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2 October 2017

Antiretroviral treatment for adult HIV infection in 2002: updated recommendations of the International AIDS Society-USA Panel.

1 reference

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2 October 2017

A potent human immunodeficiency virus type 1 protease inhibitor, UIC-94003 (TMC-126), and selection of a novel (A28S) mutation in the protease active site

1 reference

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2 October 2017

Novel low molecular weight spirodiketopiperazine derivatives potently inhibit R5 HIV-1 infection through their antagonistic effects on CCR5.

1 reference

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2 October 2017

Highly active antiretroviral therapy decreases mortality and morbidity in patients with advanced HIV disease

1 reference

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2 October 2017

AIDS — The First 20 Years

1 reference

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2 October 2017

Structural implications of drug-resistant mutants of HIV-1 protease: high-resolution crystal structures of the mutant protease/substrate analogue complexes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=201142

2 October 2017

HIV chemotherapy

1 reference

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2 October 2017

New antiretroviral drugs in development.

1 reference

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2 October 2017

In vitro resistance profile of the human immunodeficiency virus type 1 protease inhibitor BMS-232632

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=201142

2 October 2017

JE-2147: a dipeptide protease inhibitor (PI) that potently inhibits multi-PI-resistant HIV-1.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=201142

2 October 2017

Genotypic and phenotypic characterization of human immunodeficiency virus type 1 variants isolated from patients treated with the protease inhibitor nelfinavir.

1 reference

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2 October 2017

In vitro selection and characterization of human immunodeficiency virus type 1 variants with increased resistance to ABT-378, a novel protease inhibitor

1 reference

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2 October 2017

Antiviral and resistance studies of AG1343, an orally bioavailable inhibitor of human immunodeficiency virus protease

1 reference

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2 October 2017

Structural mechanisms of HIV drug resistance

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2 October 2017

Emergence of human immunodeficiency virus type 1 variants with resistance to multiple dideoxynucleosides in patients receiving therapy with dideoxynucleosides.

1 reference

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2 October 2017

Improved methods for building protein models in electron density maps and the location of errors in these models

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2 October 2017

Genotype and phenotype at baseline and at failure in human immunodeficiency virus-infected antiretroviral-naive patients in a randomized trial comparing zidovudine and lamivudine plus nelfinavir or nevirapine

1 reference

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23 September 2018

Antiretroviral-drug resistance among patients recently infected with HIV.

1 reference

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23 September 2018

Sequencing of protease inhibitor therapy: insights from an analysis of HIV phenotypic resistance in patients failing protease inhibitors

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23 September 2018

Phenotypic and genotypic analysis of clinical HIV-1 isolates reveals extensive protease inhibitor cross-resistance: a survey of over 6000 samples.

1 reference

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23 September 2018

Factors associated with clinical and virological failure in patients receiving a triple therapy including a protease inhibitor.

1 reference

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23 September 2018

Prevalence of HIV-1 resistant to antiretroviral drugs in 81 individuals newly infected by sexual contact or injecting drug use. Investigators of the Quebec Primary Infection Study.

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23 September 2018

Efavirenz plus zidovudine and lamivudine, efavirenz plus indinavir, and indinavir plus zidovudine and lamivudine in the treatment of HIV-1 infection in adults. Study 006 Team

1 reference

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23 September 2018

Energy calculations and analysis of HIV-1 protease-inhibitor crystal structures

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Transmission of antiretroviral-drug-resistant HIV-1 variants

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Processing of X-ray diffraction data collected in oscillation mode

1 reference

https://pubmed.ncbi.nlm.nih.gov/14506019

12 December 2020

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inferred from PubMed ID database lookup

Public Health Implications of Antiretroviral Therapy and HIV Drug Resistance

1 reference

https://pubmed.ncbi.nlm.nih.gov/14506019

12 December 2020

based on heuristic

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Identifiers

10.1128/AAC.47.10.3123-3129.2003

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Europe PubMed Central

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19 December 2019

PMC publication ID

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Europe PubMed Central

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19 December 2019

PubMed publication ID

1 reference

Europe PubMed Central

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19 December 2019

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