(Q39035003)

8 September 2017

Identification and synthesis of a unique thiocarbazate cathepsin L inhibitor (English)

1 reference

8 September 2017

Donna M Huryn

4

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author name string

Michael C Myers

1

1 reference

8 September 2017

Parag P Shah

2

1 reference

8 September 2017

Scott L Diamond

3

1 reference

8 September 2017

Amos B Smith

5

1 reference

8 September 2017

language of work or name

English

0 references

publication date

1 November 2007

1 reference

8 September 2017

5

1 reference

Bioorganic & Medicinal Chemistry Letters

inferred from page(s)

published in

1 reference

8 September 2017

18

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8 September 2017

210-214

1 reference

8 September 2017

1

1 reference

Identification and characterization of 3-substituted pyrazolyl esters as alternate substrates for cathepsin B: the confounding effects of DTT and cysteine in biological assays

8 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Emerging roles of cysteine cathepsins in disease and their potential as drug targets.

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Inhibitors of cathepsin L prevent severe acute respiratory syndrome coronavirus entry

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Non-peptidic inhibitors of cysteine proteases.

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Synthesis and NMR structure of p41icf, a potent inhibitor of human cathepsin L

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Irreversible inhibitors of serine, cysteine, and threonine proteases

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Recent advances in the synthesis, design and selection of cysteine protease inhibitors

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Pyrrolidine-3-carboxylic acids as endothelin antagonists. 4. Side chain conformational restriction leads to ET(B) selectivity

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

The lysosomal cysteine proteases

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Design of potent and selective human cathepsin K inhibitors that span the active site

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

The crystal structure of human cathepsin L complexed with E-64

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Azapeptides as inhibitors and active site titrants for cysteine proteinases.

9 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Cysteine protease inhibition by azapeptide esters

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

Azepanone-based inhibitors of human cathepsin L.

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

3-Acylamino-azetidin-2-one as a novel class of cysteine proteases inhibitors

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

CA-074, but not its methyl ester CA-074Me, is a selective inhibitor of cathepsin B within living cells

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

General solid-phase method to prepare novel cyclic ketone inhibitors of the cysteine protease cruzain

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2423727

From good substrates to good inhibitors: design of inhibitors for serine and thiol proteases

21 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18060772

12 December 2020

inferred from PubMed ID database lookup

Cysteine proteinase inhibitors decrease articular cartilage and bone destruction in chronic inflammatory arthritis

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18060772

12 December 2020

inferred from PubMed ID database lookup

Cysteine Proteases and Their Inhibitors

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18060772

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1016/J.BMCL.2007.10.107

1 reference

8 September 2017

1 reference

8 September 2017

1 reference