(Q42026894)

English

Tritium-labeled N(1)-[3-(1H-imidazol-4-yl)propyl]-N(2)-propionylguanidine ([(3)H]UR-PI294), a high-affinity histamine H(3) and H(4) receptor radioligand

scientific article published on February 2009

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

Tritium-labeled N(1)-[3-(1H-imidazol-4-yl)propyl]-N(2)-propionylguanidine ([(3)H]UR-PI294), a high-affinity histamine H(3) and H(4) receptor radioligand (English)

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

author name string

Patrick Igel

1

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

David Schnell

2

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

Günther Bernhardt

3

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

Roland Seifert

4

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

Armin Buschauer

5

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

publication date

1 February 2009

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

4

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

2

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

225-231

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

The histamine H4 receptor and potential therapeutic uses for H4 ligands

1 reference

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21 January 2018

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

1 reference

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7 January 2021

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Cloning and functional expression of the human histamine H3 receptor

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7 January 2021

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The histamine H3 receptor: from gene cloning to H3 receptor drugs

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The role of histamine H1 and H4 receptors in allergic inflammation: the search for new antihistamines

1 reference

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7 January 2021

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Histamine H4 receptor antagonists are superior to traditional antihistamines in the attenuation of experimental pruritus

1 reference

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7 January 2021

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Effects of guanine, inosine, and xanthine nucleotides on beta(2)-adrenergic receptor/G(s) interactions: evidence for multiple receptor conformations

1 reference

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Reconstitution of beta2-adrenoceptor-GTP-binding-protein interaction in Sf9 cells--high coupling efficiency in a beta2-adrenoceptor-G(s alpha) fusion protein

1 reference

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Highly potent and selective ligands for histamine H3-receptors

1 reference

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Characterization and tissue distribution of H3 histamine receptors in guinea pigs by N alpha-methylhistamine

1 reference

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7 January 2021

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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives

1 reference

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7 January 2021

based on heuristic

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A selective human H(4)-receptor agonist: (-)-2-cyano-1-methyl-3-[(2R,5R)-5- [1H-imidazol-4(5)-yl]tetrahydrofuran-2-y] methylguanidine

1 reference

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7 January 2021

based on heuristic

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Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

1 reference

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7 January 2021

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A potent and selective histamine H4 receptor antagonist with anti-inflammatory properties

1 reference

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7 January 2021

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Preparation and biological evaluation of indole, benzimidazole, and thienopyrrole piperazine carboxamides: potent human histamine h(4) antagonists

1 reference

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7 January 2021

based on heuristic

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Oligomerization of recombinant and endogenously expressed human histamine H(4) receptors

1 reference

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7 January 2021

based on heuristic

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Detection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligand

1 reference

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7 January 2021

based on heuristic

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Characterization of the binding of [3H]-clobenpropit to histamine H3-receptors in guinea-pig cerebral cortex membranes

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Molecular modeling and pharmacological analysis of species-related histamine H(3) receptor heterogeneity

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

Cloning, expression, and pharmacological characterization of a novel human histamine receptor.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

The first potent and selective non-imidazole human histamine H4 receptor antagonists

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and structure-activity relationships of indole and benzimidazole piperazines as histamine H(4) receptor antagonists.

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

Human skin mast cells express H2 and H4, but not H3 receptors

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

Histamine H4 receptor mediates eosinophil chemotaxis with cell shape change and adhesion molecule upregulation

1 reference

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7 January 2021

based on heuristic

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

Quantification of receptor interactions using binding methods

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

Multiple differences in agonist and antagonist pharmacology between human and guinea pig histamine H1-receptor

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

Distinct interaction of human and guinea pig histamine H2-receptor with guanidine-type agonists.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200800349

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1002/CMDC.200800349

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

15 October 2017

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