(Q44389982)

English

Cooperative interactions at M2 muscarinic acetylcholine receptors: structure/activity relationships in stepwise shortened bispyridinium- and bis(ammonio)alkane-type allosteric modulators

scientific article published in April 2003

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scholarly article

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Europe PubMed Central

PubMed publication ID

2 December 2017

Cooperative interactions at M2 muscarinic acetylcholine receptors: structure/activity relationships in stepwise shortened bispyridinium- and bis(ammonio)alkane-type allosteric modulators (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

1

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2 December 2017

Ulrike Holzgrabe

6

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2 December 2017

author name string

Maren Grossmüller

2

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Europe PubMed Central

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2 December 2017

Vildan Alptüzün

3

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Ercin Erciyas

4

1 reference

Europe PubMed Central

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2 December 2017

Christian Tränkle

5

1 reference

Europe PubMed Central

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2 December 2017

Klaus Mohr

7

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

publication date

1 April 2003

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Europe PubMed Central

PubMed publication ID

2 December 2017

Neurochemical Research

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Europe PubMed Central

PubMed publication ID

2 December 2017

28

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2 December 2017

3-4

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2 December 2017

667-673

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

Allosteric site on muscarinic acetylcholine receptors: a single amino acid in transmembrane region 7 is critical to the subtype selectivities of caracurine V derivatives and alkane-bisammonium ligands

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Site-directed mutagenesis reveals two epitopes involved in the subtype selectivity of the allosteric interactions of gallamine at muscarinic acetylcholine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The effects of brucine and alcuronium on the inhibition of [3H]acetylcholine release from rat striatum by muscarinic receptor agonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Positive cooperativity of acetylcholine and other agonists with allosteric ligands on muscarinic acetylcholine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

M2 receptor binding of the selective antagonist AF-DX 384: possible involvement of the common allosteric site.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Positive allosteric interactions on cardiac muscarinic receptors: effects of chemical modifications of disulphide and carboxyl groups

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Allosteric interactions of staurosporine and other indolocarbazoles with N-[methyl-(3)H]scopolamine and acetylcholine at muscarinic receptor subtypes: identification of a second allosteric site

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification of a [3H]Ligand for the common allosteric site of muscarinic acetylcholine M2 receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Subtype-selective positive cooperative interactions between brucine analogs and acetylcholine at muscarinic receptors: functional studies

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Allosteric modulation of muscarinic receptor signaling: alcuronium-induced conversion of pilocarpine from an agonist into an antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Quantitation of mRNAs for M(1) to M(5) subtypes of muscarinic receptors in rat heart and brain cortex

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence for a multiple binding mode of bispyridinium-type allosteric modulators of muscarinic receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Allosteric modulation of muscarinic acetylcholine receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Search for the Pharmacophore of Bispyridinium-Type Allosteric Modulators of Muscarinic Receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Interactions between allosteric modulators and 4-DAMP and other antagonists at muscarinic receptors: potential significance of the distance between the N and carboxyl C atoms in the molecules of antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Use of chimeric muscarinic receptors to investigate epitopes involved in allosteric interactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Modes of allosteric interactions with free and [3H]N-methylscopolamine-occupied muscarinic M2 receptors as deduced from buffer-dependent potency shifts

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Elevation of ligand binding to muscarinic M(2) acetylcholine receptors by bis(ammonio)alkane-type allosteric modulators

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Divergent modes of action among cationic allosteric modulators of muscarinic M2 receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Two allosteric modulators interact at a common site on cardiac muscarinic receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Activation of muscarinic acetylcholine receptors via their allosteric binding sites.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Assessing the distribution of parameters in models of ligand-receptor interaction: to log or not to log.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Allosteric binding sites on cell-surface receptors: novel targets for drug discovery

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Estimation of the affinities of allosteric ligands using radioligand binding and pharmacological null methods.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Protein measurement with the Folin phenol reagent

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of acidic amino acids in the allosteric modulation by gallamine of antagonist binding at the m2 muscarinic acetylcholine receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

G protein-coupled receptor allosterism and complexing

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Changes of cooperativity between N-methylscopolamine and allosteric modulators alcuronium and gallamine induced by mutations of external loops of muscarinic M(3) receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Search for lead structures to develop new allosteric modulators of muscarinic receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Detection, quantitation, and verification of allosteric interactions of agents with labeled and unlabeled ligands at G protein-coupled receptors: interactions of strychnine and acetylcholine at muscarinic receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of an agonist, allosteric modulator, and antagonist on guanosine-gamma-[35S]thiotriphosphate binding to liposomes with varying muscarinic receptor/Go protein stoichiometry

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Interactions of alcuronium, TMB-8, and other allosteric ligands with muscarinic acetylcholine receptors: studies with chimeric receptors.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Modification of the binding properties of muscarinic receptors by gallamine

1 reference

https://pubmed.ncbi.nlm.nih.gov/12675159

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1023/A:1022858414900

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

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PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 December 2017

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