(Q24646822)

English

Evidence that the plant cannabinoid cannabigerol is a highly potent alpha2-adrenoceptor agonist and moderately potent 5HT1A receptor antagonist

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scholarly article

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Evidence that the plant cannabinoid cannabigerol is a highly potent alpha2-adrenoceptor agonist and moderately potent 5HT1A receptor antagonist (English)

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cannabinoid receptor

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author name string

M G Cascio

1

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L A Gauson

2

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L A Stevenson

3

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R A Ross

4

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R G Pertwee

5

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language of work or name

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publication date

January 2010

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British Journal of Pharmacology

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159

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1

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129-41

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The diverse CB1 and CB2 receptor pharmacology of three plant cannabinoids: delta9-tetrahydrocannabinol, cannabidiol and delta9-tetrahydrocannabivarin

1 reference

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7 April 2017

Evidence that the plant cannabinoid Delta9-tetrahydrocannabivarin is a cannabinoid CB1 and CB2 receptor antagonist

1 reference

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7 April 2017

Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656, and AM630

1 reference

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7 April 2017

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

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7 April 2017

Structure-activity relationship for the endogenous cannabinoid, anandamide, and certain of its analogues at vanilloid receptors in transfected cells and vas deferens

1 reference

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7 April 2017

Isolation and structure of a brain constituent that binds to the cannabinoid receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2823359

7 April 2017

Alpha2-agonists as analgesic agents.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2823359

27 September 2017

Plant-derived cannabinoids modulate the activity of transient receptor potential channels of ankyrin type-1 and melastatin type-8.

1 reference

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27 September 2017

Cannabidiol displays unexpectedly high potency as an antagonist of CB1 and CB2 receptor agonists in vitro

1 reference

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Cannabinoids inhibit human keratinocyte proliferation through a non-CB1/CB2 mechanism and have a potential therapeutic value in the treatment of psoriasis

1 reference

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2 references

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27 September 2017

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Chemical constituents of marijuana: the complex mixture of natural cannabinoids

1 reference

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Modulation of transmitter release via presynaptic cannabinoid receptors

1 reference

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Structural determinants of the partial agonist-inverse agonist properties of 6'-azidohex-2'-yne-delta8-tetrahydrocannabinol at cannabinoid receptors

1 reference

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27 September 2017

Pharmacology of cannabinoid CB1 and CB2 receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2823359

27 September 2017

Agonist-antagonist characterization of 6'-cyanohex-2'-yne-delta 8-tetrahydrocannabinol in two isolated tissue preparations.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2823359

27 September 2017

Noradrenaline-ATP co-transmission in the sympathetic nervous system

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2823359

27 September 2017

pA2 and receptor differentiation: a statistical analysis of competitive antagonism

1 reference

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27 September 2017

[Gamma-35S]GTP autoradiography allows region-specific detection of muscarinic receptor-dependent G-protein activation in the chick optic tectum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2823359

30 May 2018

Maprotiline: an antidepressant with an unusual pharmacological profile.

1 reference

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30 May 2018

Guide to Receptors and Channels (GRAC), 3rd edition

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

Plant cannabinoids: a neglected pharmacological treasure trove

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

(-)-Cannabidiol antagonizes cannabinoid receptor agonists and noradrenaline in the mouse vas deferens

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

Evidence that (-)-7-hydroxy-4'-dimethylheptyl-cannabidiol activates a non-CB(1), non-CB(2), non-TRPV1 target in the mouse vas deferens

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

Stimulation frequency-noradrenaline release relationships examined in alpha2A-, alpha2B- and alpha2C-adrenoceptor-deficient mice

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

Presynaptic autoreceptors in the third decade: focus on alpha2-adrenoceptors

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

6"-Azidohex-2"-yne-cannabidiol: a potential neutral, competitive cannabinoid CB1 receptor antagonist

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00515.X

21 January 2018

Modulation of (3)H-noradrenaline release by presynaptic opioid, cannabinoid and bradykinin receptors and beta-adrenoceptors in mouse tissues

1 reference

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21 January 2018

Evidence for a new G protein-coupled cannabinoid receptor in mouse brain.

1 reference

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28 November 2018

Psychopharmacological activity of the active constituents of hashish and some related cannabinoids

1 reference

https://pubmed.ncbi.nlm.nih.gov/20002104

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Actions of alpha2 adrenoceptor ligands at alpha2A and 5-HT1A receptors: the antagonist, atipamezole, and the agonist, dexmedetomidine, are highly selective for alpha2A adrenoceptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/20002104

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A pharmacological profile of the selective silent 5-HT1A receptor antagonist, WAY-100635

1 reference

https://pubmed.ncbi.nlm.nih.gov/20002104

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological characterization of three novel cannabinoid receptor agonists in the mouse isolated vas deferens

1 reference

https://pubmed.ncbi.nlm.nih.gov/20002104

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Chemical basis of hashish activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/20002104

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.2009.00515.X

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

OpenCitations bibliographic resource ID

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Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

PMC publication ID

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Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

PubMed publication ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

ResearchGate publication ID

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