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What systems can and can't do
scientific article
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instance of
scholarly article
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title
What systems can and can't do
(English)
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author name string
T Kenakin
series ordinal
1
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language of work or name
English
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publication date
March 2008
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published in
British Journal of Pharmacology
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volume
153
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issue
5
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page(s)
841-3
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cites work
The receptor concept: pharmacology's big idea
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PubMed Central
reference URL
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7 April 2017
Some quantitative uses of drug antagonists
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PubMed Central
reference URL
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retrieved
7 April 2017
A study of antagonist affinities for the human histamine H2 receptor
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PubMed Central
reference URL
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28 September 2017
Allosteric GPCR modulators: taking advantage of permissive receptor pharmacology.
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28 September 2017
Versatility of GPCR recognition by drugs: from biological implications to therapeutic relevance
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28 September 2017
Multiple GPCR conformations and signalling pathways: implications for antagonist affinity estimates.
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28 September 2017
A novel, conformation-specific allosteric inhibitor of the tachykinin NK2 receptor (NK2R) with functionally selective properties
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28 September 2017
Determining the potency and molecular mechanism of action of insurmountable antagonists
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28 September 2017
New concepts in drug discovery: collateral efficacy and permissive antagonism
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28 September 2017
GPCR drug discovery through the exploitation of allosteric drug binding sites
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28 September 2017
Identification of allosteric peptide agonists of CXCR4.
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28 September 2017
G protein-coupled receptor allosterism and complexing
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28 September 2017
The putative beta4-adrenergic receptor is a novel state of the beta1-adrenergic receptor
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28 September 2017
On the application of "a plausible model" of allosteric proteins to the receptor for acetylcholine
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28 September 2017
Evidence for a secondary state of the human beta3-adrenoceptor.
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30 May 2018
A three-state receptor model of agonist action
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30 May 2018
On the analysis of pharmacological experiments in terms of an allosteric receptor model
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PubMed Central
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30 May 2018
Estimation of the affinities of allosteric ligands using radioligand binding and pharmacological null methods.
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PubMed Central
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30 May 2018
Allosteric Modulation of G Protein–Coupled Receptors
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2267279
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28 November 2018
Analysis of allosterism in functional assays
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2267279
retrieved
28 November 2018
Identification of indole derivatives exclusively interfering with a G protein-independent signaling pathway of the prostaglandin D2 receptor CRTH2.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2267279
retrieved
28 November 2018
Site of action of beta-ligands at the human beta1-adrenoceptor
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2267279
retrieved
28 November 2018
Agonist actions of "beta-blockers" provide evidence for two agonist activation sites or conformations of the human beta1-adrenoceptor
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2267279
retrieved
28 November 2018
Modeling the functional effects of allosteric modulators at pharmacological receptors: an extension of the two-state model of receptor activation.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2267279
retrieved
28 November 2018
Identifiers
DOI
10.1038/SJ.BJP.0707677
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PMC publication ID
2267279
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PubMed publication ID
18204481
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ResearchGate publication ID
5648090
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