(Q24681849)

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Centrally acting hypotensive agents with affinity for 5-HT1A binding sites inhibit forskolin-stimulated adenylate cyclase activity in calf hippocampus

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scholarly article

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Centrally acting hypotensive agents with affinity for 5-HT1A binding sites inhibit forskolin-stimulated adenylate cyclase activity in calf hippocampus (English)

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author name string

P Schoeffter

1

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D Hoyer

2

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language of work or name

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publication date

November 1988

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British Journal of Pharmacology

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95

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975-85

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3

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Characterization of the 5-hydroxytryptamine1a receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in guinea pig and rat hippocampal membranes

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Cardiovascular response to 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT) in the rat: site of action and pharmacological analysis.

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Binding characteristics of a radiolabeled agonist and antagonist at central nervous system alpha noradrenergic receptors

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Hypotensive properties of benzodioxane derivatives structurally related to R 28935. Comparison of activity with some receptor affinities

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30 May 2018

Two 5-HT receptors linked to adenylate cyclase in guinea pig hippocampus are discriminated by 5-carboxamidotryptamine and spiperone.

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5-HT-1a and 5-HT-1b selectivity of two phenylpiperazine derivatives: evidence for 5-HT-1b heterogeneity.

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30 May 2018

Serotonin receptors in the human brain. I. Characterization and autoradiographic localization of 5-HT1A recognition sites. Apparent absence of 5-HT1B recognition sites.

1 reference

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Electrophysiological responses of serotoninergic dorsal raphe neurons to 5-HT1A and 5-HT1B agonists

1 reference

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30 May 2018

5-HT1D receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in calf substantia nigra.

1 reference

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30 May 2018

5-HT1B receptors are negatively coupled with adenylate cyclase in rat substantia nigra

1 reference

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[3H]spiroxatrine labels a serotonin1A-like site in the rat hippocampus

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Evidence that the putative 5-HT1A receptor agonists, 8-OH-DPAT and ipsapirone, have a central hypotensive action that differs from that of clonidine in anaesthetised cats.

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Serotonin receptors in the human brain--III. Autoradiographic mapping of serotonin-1 receptors

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Pharmacological characterization of two 5-hydroxytryptamine receptors coupled to adenylate cyclase in guinea pig hippocampal membranes.

1 reference

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5-HT1A-receptors mediate stimulation of adenylate cyclase in rat hippocampus.

1 reference

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Canine basilar artery contractions mediated by 5-hydroxytryptamine1A receptors.

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Species variations in RU 24969 interactions with non-5-HT1A binding sites

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Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites.

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Inhibition of forskolin-stimulated adenylate cyclase activity by 5-HT receptor agonists

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Spiperone differentiates multiple 5-hydroxytryptamine responses in rat hippocampal slices in vitro.

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Piperazine derivatives including the putative anxiolytic drugs, buspirone and ipsapirone, are agonists at 5-HT1A receptors negatively coupled with adenylate cyclase in hippocampal neurons

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Studies on the influence of the antihypertensive drug urapidil on blood circulation and its regulation in animal experiments (author's transl)

1 reference

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30 May 2018

Molecular pharmacology of 5-HT1D recognition sites: radioligand binding studies in human, pig and calf brain membranes.

1 reference

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1 reference

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1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11728.X

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Hypotensive action of 8-hydroxy-2-(di-N-propylamino)tetralin (8-OH-DPAT) in spontaneously hypertensive rats.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854240

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The 5-hydroxytryptamine 5-HT1D receptor subtype is negatively coupled to adenylate cyclase in calf substantia nigra

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11728.X

21 January 2018

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1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11728.X

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1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Disposition and pharmacological effects of m-Chlorophenylpiperazine in rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

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based on heuristic

inferred from PubMed ID database lookup

Evidence for a central depressor action of postsynaptic α1-adrenergic receptor antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

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based on heuristic

inferred from PubMed ID database lookup

Tryptophan analogues. 1. Synthesis and antihypertensive activity of positional isomers

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

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based on heuristic

inferred from PubMed ID database lookup

8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

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based on heuristic

inferred from PubMed ID database lookup

Hypotensive activity of serotonin receptor agonists in rats is related to their affinity for 5-HT1 receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

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based on heuristic

inferred from PubMed ID database lookup

LY165163 and 8-OH-DPAT have agonist effects on a serotonin responsive muscle of Aplysia

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Acute administration of 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT), a selective 5-HT-receptor agonist, causes a biphasic blood pressure response and a bradycardia in the normotensive Sprague-Dawley rat and in the spontaneously hypertensive r

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

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based on heuristic

inferred from PubMed ID database lookup

Cardiovascular effects and interaction with adrenoceptors of urapidil

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Spiroxatrine: a selective serotonin1A receptor antagonist.

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Neurochemical and behavioural evidence for an agonist action of 1-[2-(4-aminophenyl)ethyl]-4-(3-trifluoromethylphenyl)piperazine (LY 165163) at central 5-HT receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/3207999

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

(-)-Propranolol and (+/-)-cyanopindolol are mixed agonists-antagonists at serotonin autoreceptors in the hippocampus of the rat brain

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11728.X

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1111/J.1476-5381.1988.TB11728.X

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