(Q27639887)

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X-ray Crystal Structure of a Bisubstrate Inhibitor Bound to the Enzyme Catechol-O-methyltransferase: A Dramatic Effect of Inhibitor Preorganization on Binding Affinity

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X-ray Crystal Structure of a Bisubstrate Inhibitor Bound to the Enzyme Catechol-O-methyltransferase: A Dramatic Effect of Inhibitor Preorganization on Binding Affinity (English)
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Christian Lerner
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Armin Ruf
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Volker Gramlich
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Birgit Masjost
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Gerhard Zürcher
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Roland Jakob-Roetne
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Edilio Borroni
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5 November 2001
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40
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21
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4040-4042
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