(Q27650937)

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Kinesin spindle protein (KSP) inhibitors. 9. Discovery of (2S)-4-(2,5-difluorophenyl)-n-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide (MK-0731) for the treatment of taxane-refractory cancer (English)
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Christopher D Cox
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Paul J Coleman
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Michael J Breslin
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David B Whitman
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Robert M Garbaccio
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Mark E Fraley
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Carolyn A Buser
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Eileen S Walsh
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Kelly Hamilton
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Michael D Schaber
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Robert B Lobell
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Weikang Tao
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Joseph P Davide
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Ronald E Diehl
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Marc T Abrams
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Vicki J South
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Hans E Huber
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Maricel Torrent
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Thomayant Prueksaritanont
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Chunze Li
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Donald E Slaughter
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Elizabeth Mahan
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Carmen Fernandez-Metzler
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Youwei Yan
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Lawrence C Kuo
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Nancy E Kohl
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George D Hartman
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24 July 2008
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51
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14
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4239-52
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