(Q27660322)

English

Optimization of phenyl-substituted benzimidazole carboxamide poly(ADP-ribose) polymerase inhibitors: identification of (S)-2-(2-fluoro-4-(pyrrolidin-2-yl)phenyl)-1H-benzimidazole-4-carboxamide (A-966492), a highly potent and efficacious inhibitor

scientific article

Statements

Optimization of phenyl-substituted benzimidazole carboxamide poly(ADP-ribose) polymerase inhibitors: identification of (S)-2-(2-fluoro-4-(pyrrolidin-2-yl)phenyl)-1H-benzimidazole-4-carboxamide (A-966492), a highly potent and efficacious inhibitor (English)
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Thomas D Penning
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Gui-Dong Zhu
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Jianchun Gong
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Sheela Thomas
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Viraj B Gandhi
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Xuesong Liu
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Yan Shi
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Vered Klinghofer
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Eric F Johnson
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Chang H Park
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Elizabeth H Fry
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Cherrie K Donawho
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David J Frost
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Fritz G Buchanan
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Gail T Bukofzer
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Luis E Rodriguez
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Velitchka Bontcheva-Diaz
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Jennifer J Bouska
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Donald J Osterling
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Amanda M Olson
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Kennan C Marsh
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Yan Luo
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Vincent L Giranda
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22 April 2010
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53
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3142-53
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8
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