(Q27683848)

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A novel class of oral direct renin inhibitors: highly potent 3,5-disubstituted piperidines bearing a tricyclic p3-p1 pharmacophore

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A novel class of oral direct renin inhibitors: highly potent 3,5-disubstituted piperidines bearing a tricyclic p3-p1 pharmacophore (English)
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Nils Ostermann
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Simon Ruedisser
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Claus Ehrhardt
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Werner Breitenstein
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Andreas Marzinzik
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Edgar Jacoby
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Johannes Ottl
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Martin Klumpp
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J Constanze D Hartwieg
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Frederic Cumin
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Ulrich Hassiepen
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Jörg Trappe
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Richard Sedrani
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Sabine Geisse
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Bernd Gerhartz
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Paul Richert
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Eric Francotte
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Trixie Wagner
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Markus Krömer
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Takatoshi Kosaka
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Randy L Webb
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Dean F Rigel
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Jürgen Maibaum
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Daniel K Baeschlin
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28 March 2013
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56
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6
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2196-206
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