(Q27728279)

5

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Claudiu T Supuran

11

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Vincenzo Alterio

1

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Simona Maria Monti

6

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Jean-Yves Winum

13

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Daniela Vullo

4

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author name string

Roberta Cadoni

2

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Davide Esposito

3

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Andrea Caporale

7

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Menotti Ruvo

8

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Mario Sechi

9

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Pascal Dumy

Multiple binding modes of inhibitors to carbonic anhydrases: how to design specific drugs targeting 15 different isoforms?

10

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language of work or name

English

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publication date

29 September 2016

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published in

Chemical Communications

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volume

52

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issue

80

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page(s)

11983-11986

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cites work

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Targeting tumor hypoxia: suppression of breast tumor growth and metastasis by novel carbonic anhydrase IX inhibitors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isoforms I and II and transmembrane, tumor-associated isoforms IX and XII with boronic acids

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

3D-QSAR-aided design, synthesis, in vitro and in vivo evaluation of dipeptidyl boronic acid proteasome inhibitors and mechanism studies.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Development of the proteasome inhibitor Velcade (Bortezomib).

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

An assessment of the genetic toxicology of novel boron-containing therapeutic agents.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Discovery of a new boron-containing antifungal agent, 5-fluoro-1,3-dihydro-1-hydroxy-2,1- benzoxaborole (AN2690), for the potential treatment of onychomycosis

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

An antifungal agent inhibits an aminoacyl-tRNA synthetase by trapping tRNA in the editing site

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Linking phenotype to kinase: identification of a novel benzoxaborole hinge-binding motif for kinase inhibition and development of high-potency rho kinase inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Interfering with pH regulation in tumours as a therapeutic strategy

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Hydroxylamine-O-sulfonamide is a versatile lead compound for the development of carbonic anhydrase inhibitors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

REFMAC5 for the refinement of macromolecular crystal structures

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Overview of the CCP4 suite and current developments

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Refined structure of human carbonic anhydrase II at 2.0 A resolution

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Benzoxaboroles: a new class of potential drugs for human African trypanosomiasis

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Nitrogen-15 NMR spectroscopy of the catalytic-triad histidine of a serine protease in peptide boronic acid inhibitor complexes

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Ring Structure and Aromatic Substituent Effects on the pK a of the Benzoxaborole Pharmacophore

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C

Carbonic anhydrase inhibitors. Inhibition of the fungal β-carbonic anhydrases from Candida albicans and Cryptococcus neoformans with boronic acids

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC6CC06399C