(Q28115233)

English

Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognition

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PubMed publication ID

3 January 2017

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognition (English)

2 references

PubMed publication ID

3 January 2017

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

transmembrane protein

0 references

author name string

Q Jiang

1

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

A M Van Rhee

2

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

J Kim

3

1 reference

Europe PubMed Central

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19 October 2019

S Yehle

4

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

J Wess

5

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

K A Jacobson

6

1 reference

Europe PubMed Central

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19 October 2019

language of work or name

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publication date

1 September 1996

2 references

PubMed publication ID

3 January 2017

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

Molecular Pharmacology

2 references

PubMed publication ID

3 January 2017

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

50

2 references

PubMed publication ID

3 January 2017

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

3

2 references

PubMed publication ID

3 January 2017

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

512-521

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8794889%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

DNA sequencing with chain-terminating inhibitors

1 reference

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Site-directed mutagenesis identifies residues involved in ligand recognition in the human A2a adenosine receptor

1 reference

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Structure-activity relationships of N6-benzyladenosine-5'-uronamides as A3-selective adenosine agonists

1 reference

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1 reference

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Allele-specific activation of genetically engineered receptors

1 reference

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1 reference

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A cDNA cloning vector that permits expression of cDNA inserts in mammalian cells

1 reference

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Use of eukaryotic expression technology in the functional analysis of cloned genes

1 reference

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2-[2-[4-[2-[2-[ 1,3-Dihydro- 1,1-bis (4-hydroxyphenyl)-3-oxo-5-isobenzofuranthioureidyl]ethylaminocarbonyl]ethyl]phenyl] ethylamino]-5'-N-ethylcarboxamidoadenosine (FITC-APEC): A Fluorescent Ligand For A2a-Adenosine Receptors.

1 reference

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29 September 2017

Identification of an adenosine receptor domain specifically involved in binding of 5'-substituted adenosine agonists

1 reference

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A1 adenosine receptors. Two amino acids are responsible for species differences in ligand recognition

1 reference

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The in vitro pharmacology of ZM 241385, a potent, non‐xanthine, A2a selective adenosine receptor antagonist

1 reference

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29 September 2017

Identification of the A2 adenosine receptor binding subunit by photoaffinity crosslinking

1 reference

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29 September 2017

Agonist derived molecular probes for A2 adenosine receptors

1 reference

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Muscarinic acetylcholine receptors. Peptide sequencing identifies residues involved in antagonist binding and disulfide bond formation

1 reference

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Cardiovascular purinoceptors

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Molecular recognition. Conformational analysis of limited proteolytic sites and serine proteinase protein inhibitors

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Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential

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Chemical modification and irreversible inhibition of striatal A2a adenosine receptors

1 reference

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29 September 2017

Cloning, expression, and characterization of the unique bovine A1 adenosine receptor. Studies on the ligand binding site by site-directed mutagenesis

1 reference

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29 September 2017

Adenosine A1 and A2 receptors: structure--function relationships

1 reference

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29 September 2017

Constitutive activation of the alpha 1B-adrenergic receptor by all amino acid substitutions at a single site. Evidence for a region which constrains receptor activation

1 reference

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Constitutively active mutants of the alpha 2-adrenergic receptor

1 reference

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Site-directed mutagenesis of the serotonin 5-hydroxytrypamine2 receptor: identification of amino acids necessary for ligand binding and receptor activation

1 reference

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A threonine residue in the seventh transmembrane domain of the human A1 adenosine receptor mediates specific agonist binding

1 reference

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2 June 2018

Role of adenosine A2a receptors in the nucleus accumbens

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KF17837: a novel selective adenosine A2A receptor antagonist with anticataleptic activity

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[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain

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The role of conserved aspartate and serine residues in ligand binding and in function of the 5-HT1A receptor: a site-directed mutation study

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Site-directed mutagenesis of the human dopamine D2 receptor

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Adenosine agonists reduce conditioned avoidance responding in the rat.

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Movement of the retinylidene Schiff base counterion in rhodopsin by one helix turn reverses the pH dependence of the metarhodopsin I to metarhodopsin II transition

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