(Q28238260)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

title

New substrate analogues of human serotonin N-acetyltransferase produce in situ specific and potent inhibitors (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

0 references

14

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Jean A Boutin

16

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

author name string

Gilles Ferry

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Caroline Ubeaud

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Julien Mozo

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Christophe Péan

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Philippe Hennig

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Marianne Rodriguez

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Catherine Scoul

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Anne Bonnaud

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Olivier Nosjean

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Jean-Pierre Galizzi

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Philippe Delagrange

11

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Pierre Renard

12

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Jean-Paul Volland

13

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

Daniel Lesieur

15

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

language of work or name

English

0 references

publication date

1 January 2004

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

volume

271

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

17 November 2019

issue

2

1 reference

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17 November 2019

page(s)

418-428

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:14717709%20AND%20SRC:MED&resulttype=core&format=json

The human serotonin N-acetyltransferase (EC 2.3.1.87) gene (AANAT): structure, chromosomal localization, and tissue expression

17 November 2019

cites work

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

Substrate specificity and inhibition studies of human serotonin N-acetyltransferase

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

Structure-activity relationships for substrates and inhibitors of pineal 5-hydroxytryptamine-N-acetyltransferase: preliminary studies

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

Mechanism-based inhibition of the melatonin rhythm enzyme: pharmacologic exploitation of active site functional plasticity

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

X-ray crystallographic studies of serotonin N-acetyltransferase catalysis and inhibition

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

A Potent Inhibitor of the Melatonin Rhythm Enzyme

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

Role of a pineal cAMP-operated arylalkylamine N-acetyltransferase/14-3-3-binding switch in melatonin synthesis

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

Kinetic analysis of the catalytic mechanism of serotonin N-acetyltransferase (EC 2.3.1.87)

21 April 2017

1 reference

https://api.crossref.org/works/10.1046/J.1432-1033.2003.03942.X

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

21 April 2017

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Involvement of the mt1 melatonin receptor in human breast cancer

21 April 2017

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Effect of melatonin on bone metabolism in ovariectomized rats

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Characterization and regulation of a CHO cell line stably expressing human serotonin N-acetyltransferase (EC 2.3.1.87).

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Bisubstrate ketone analogues as serotonin N-acetyltransferase inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Synthesis of 2-amido-2,3-dihydro-1H-phenalene derivatives as new conformationally restricted ligands for melatonin receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Synthesis of phenalene and acenaphthene derivatives as new conformationally restricted ligands for melatonin receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Melatonergic properties of the (+)- and (-)-enantiomers of N-(4-methoxy-2,3-dihydro-1H-phenalen-2-yl)amide derivatives

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Synthesis of a small library of phenylalkylamide derivatives as melatoninergic ligands for human mt1 and MT2 receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Synthesis and structure-affinity-activity relationships of novel benzofuran derivatives as MT(2) melatonin receptor selective ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Control of melatonin synthesis in the mammalian pineal gland: the critical role of serotonin acetylation

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Therapeutic perspectives for melatonin agonists and antagonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Serotonin N-acetyltransferase: mechanism and inhibition

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Pharmacological treatment of obesity: therapeutic strategies

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Synthesis and structure-activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Tetrahydronaphthalenic derivatives as new agonist and antagonist ligands for melatonin receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X

Substituted oxygenated heterocycles and thio-analogues: synthesis and biological evaluation as melatonin ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.1432-1033.2003.03942.X