(Q28259053)

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Piperazine-based CCR5 antagonists as HIV-1 inhibitors. IV. Discovery of 1-[(4,6-dimethyl-5-pyrimidinyl)carbonyl]- 4-[4-[2-methoxy-1(R)-4-(trifluoromethyl)phenyl]ethyl-3(S)-methyl-1-piperazinyl]- 4-methylpiperidine (Sch-417690/Sch-D), a potent, highly selective, and orally bioavailable CCR5 antagonist (English)
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Jayaram R Tagat
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Stuart W McCombie
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Dennis Nazareno
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Marc A Labroli
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Yushi Xiao
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Ruo W Steensma
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Julie M Strizki
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Bahige M Baroudy
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Kathleen Cox
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Jean Lachowicz
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Geoffrey Varty
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Robert Watkins
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6 May 2004
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47
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10
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2405-8
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