(Q28297986)

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Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: structure-activity relationships of novel substituted indole analogues and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)-carbonyl]-4-[3- [(1-methylethyl)amino]-pyridinyl]piperazine monomethanesulfonate (U-90152S), a second-generation clinical candidate (English)
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D L Romero
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R A Morge
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M J Genin
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C Biles
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M Busso
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L Resnick
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I W Althaus
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F Reusser
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R C Thomas
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W G Tarpley
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14 May 1993
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36
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10
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1505-8
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