(Q28343259)

English

Distinction between surmountable and insurmountable selective AT1 receptor antagonists by use of CHO-K1 cells expressing human angiotensin II AT1 receptors

scientific article (publication date: February 1999)

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scholarly article

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Distinction between surmountable and insurmountable selective AT1 receptor antagonists by use of CHO-K1 cells expressing human angiotensin II AT1 receptors (English)

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author name string

P M Vanderheyden

1

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F L Fierens

2

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J P De Backer

3

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N Fraeyman

4

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G Vauquelin

5

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language of work or name

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publication date

February 1999

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British Journal of Pharmacology

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126

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4

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1057-65

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Pharmacology of LR-B/081, a new highly potent, selective and orally active, nonpeptide angiotensin II AT1 receptor antagonist

1 reference

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20 March 2017

A new generation of Ca2+ indicators with greatly improved fluorescence properties

1 reference

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20 March 2017

Molecular cloning and sequencing of the gene encoding human angiotensin II type 1 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

20 March 2017

Some quantitative uses of drug antagonists

1 reference

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7 April 2017

Quantitative studies of antagonists for 5-hydroxytryptamine

1 reference

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29 September 2017

The conformational change responsible for AT1 receptor activation is dependent upon two juxtaposed asparagine residues on transmembrane helices III and VII.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

29 September 2017

Agonist-antagonist interactions at angiotensin receptors: application of a two-state receptor model

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

29 September 2017

Inositol phosphates turnover, cytosolic Ca++ and pH: putative signals for the control of cell growth

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

29 September 2017

Deregulation of hamster fibroblast proliferation by mutated ras oncogenes is not mediated by constitutive activation of phosphoinositide-specific phospholipase C.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

29 September 2017

Nonpeptide angiotensin II receptor antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

29 September 2017

Angiotensin II Receptors and Functional Correlates

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

29 September 2017

Intracellular trafficking of angiotensin II and its AT1 and AT2 receptors: evidence for selective sorting of receptor and ligand

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

Elucidation of the insurmountable nature of an angiotensin receptor antagonist, SC-54629.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

Non-peptide angiotensin agonist. Functional and molecular interaction with the AT1 receptor.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

BMS-180560, an insurmountable inhibitor of angiotensin II-stimulated responses: comparison with losartan and EXP3174.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

Different types of receptor interaction of peptide and nonpeptide angiotensin II antagonists revealed by receptor binding and functional studies

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

Pharmacological profile of GR117289 in vitro: a novel, potent and specific non-peptide angiotensin AT1 receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

Evidence that the apparent complexity of receptor antagonism by angiotensin II analogues is due to a reversible and syntopic action

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

2 June 2018

Angiotensin II receptor subtypes

1 reference

https://api.crossref.org/works/10.1038%2FSJ.BJP.0702398

21 January 2018

Pharmacological properties of KT3-671, a novel nonpeptide angiotensin II receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

27 November 2018

Effects of an angiotensin II receptor antagonist, CV-11974, on angiotensin II-induced increases in cytosolic free calcium concentration, hyperplasia, and hypertrophy of cultured vascular smooth muscle cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571230

27 November 2018

In vivo receptor occupancy of the angiotensin II receptor by nonpeptide antagonists: relationship to in vitro affinities and in vivo pharmacologic potency

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Functional studies but not receptor binding can distinguish surmountable from insurmountable AT1 antagonism

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacology of LR-B/057, a novel orally active AT1 receptor antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Candesartan (CV-11974) dissociates slowly from the angiotensin AT1 receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Desensitization, two-state receptors and pharmacological parameters

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Processing of angiotensin II (A-II) and (Sar1,Ala8)A-II by cultured bovine adrenocortical cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Nonpeptide angiotensin II receptor antagonists. XI. Pharmacology of EXP3174: an active metabolite of DuP 753, an orally active antihypertensive agent

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The cytosensor microphysiometer: biological applications of silicon technology

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological characterization of SR 47436, a new nonpeptide AT1 subtype angiotensin II receptor antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological profile of a highly potent and long-acting angiotensin II receptor antagonist, 2-ethoxy-1-[[2'-(1H-tetrazol-5-yl)biphenyl-4- yl]methyl]-1H-benzimidazole-7-carboxylic acid (CV-11974), and its prodrug, (+/-)-1-(cyclohexyloxycarbonyloxy

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Inhibition of rabbit aortic angiotensin II (AII) receptor by CV-11974, a new nonpeptide AII antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Different types of angiotensin II receptor antagonism induced by BIBS 222 in the rat portal vein and rabbit aorta; the influence of receptor reserve

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Internalization of the rat AT1a and AT1b receptors: pharmacological and functional requirements

1 reference

https://pubmed.ncbi.nlm.nih.gov/10193788

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1038/SJ.BJP.0702398

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