(Q28343952)

English

Bradyzide, a potent non-peptide B(2) bradykinin receptor antagonist with long-lasting oral activity in animal models of inflammatory hyperalgesia

scientific article

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scholarly article

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Bradyzide, a potent non-peptide B(2) bradykinin receptor antagonist with long-lasting oral activity in animal models of inflammatory hyperalgesia (English)

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author name string

G M Burgess

1

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M N Perkins

2

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H P Rang

3

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E A Campbell

4

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M C Brown

5

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P McIntyre

6

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L Urban

7

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E K Dziadulewicz

8

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T J Ritchie

9

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A Hallett

10

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C R Snell

11

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R Wrigglesworth

12

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W Lee

13

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C Davis

14

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S B Phagoo

15

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A J Davis

16

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E Phillips

17

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G S Drake

18

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G A Hughes

19

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A Dunstan

20

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G C Bloomfield

21

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language of work or name

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publication date

January 2000

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British Journal of Pharmacology

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129

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77-86

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1

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Molecular characterisation of cloned bradykinin B1 receptors from rat and human

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

The nonpeptide B2 receptor antagonist FR173657: inhibition of effects of bradykinin related to its role in nociception

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

Cloned murine bradykinin receptor exhibits a mixed B1 and B2 pharmacological selectivity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

The nonpeptide WIN 64338 is a bradykinin B2 receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

Bradykinin-induced activation of nociceptors: receptor and mechanistic studies on the neonatal rat spinal cord-tail preparation in vitro

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

Cloning and pharmacological characterization of a human bradykinin (BK-2) receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

Bioregulation of kinins: kallikreins, kininogens, and kininases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

20 March 2017

Hoe 140 a new potent and long acting bradykinin-antagonist: in vivo studies

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

6 April 2017

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

7 April 2017

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

7 April 2017

The identification of an orally active, nonpeptide bradykinin B2 receptor antagonist, FR173657

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Selective labelling of bradykinin receptor subtypes in WI38 human lung fibroblasts

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Induction of bradykinin B1 receptors in vivo in a model of ultra-violet irradiation-induced thermal hyperalgesia in the rat.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Bradykinin and inflammatory pain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Pharmacology of bradykinin and related kinins.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Bradykinin as a pain mediator: receptors are localized to sensory neurons, and antagonists have analgesic actions

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Suppression of carrageenan-induced hyperalgesia, hyperthermia and edema by a bradykinin antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Bradykinin antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

New, long-acting, potent bradykinin antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Hoe 140 a new potent and long acting bradykinin-antagonist: in vitro studies

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

A critical review of the afferent pathways and the potential chemical mediators involved in cardiac pain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Bradykinin receptors: pharmacological properties and biological roles

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Biochemical and Molecular Pharmacology of Kinin Receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

29 September 2017

Design of potent non-peptide competitive antagonists of the human bradykinin B2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

2 June 2018

ATP-induced calcium mobilization and inositol 1,4,5-triphosphate formation in H-35 hepatoma cells.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

2 June 2018

Chemosensitivity of fine afferents from rat skin in vitro

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

2 June 2018

Characterization of bradykinin receptors solubilized from rat uterus and NG108-15 cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

2 June 2018

The nociceptor sensitization by bradykinin does not depend on sympathetic neurons.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

2 June 2018

Capsazepine reversal of the antinociceptive action of capsaicin in vivo

1 reference

https://api.crossref.org/works/10.1038%2FSJ.BJP.0703012

21 January 2018

A novel class of orally active non-peptide bradykinin B2 receptor antagonists. 4. Discovery of novel frameworks mimicking the active conformation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1621130

27 November 2018

Interleukin-1 beta induced-desArg9bradykinin-mediated thermal hyperalgesia in the rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Signal transduction pathways for B1 and B2 bradykinin receptors in bovine pulmonary artery endothelial cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Responsiveness of slowly conducting articular afferents to bradykinin: effects of an experimental arthritis

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Sensitization of articular afferents to mechanical stimuli by bradykinin

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Sensitization of peripheral afferent fibres in the in vitro neonatal rat spinal cord-tail by bradykinin and prostaglandins

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antinociceptive activity of the bradykinin B1 and B2 receptor antagonists, des-Arg9, [Leu8]-BK and HOE 140, in two models of persistent hyperalgesia in the rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Induction of B1 receptors in vivo in a model of persistent inflammatory mechanical hyperalgesia in the rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/10694205

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1038/SJ.BJP.0703012

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