(Q28356112)

1

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S Barone

2

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U Kammula

3

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G L Stiles

Journal of Medicinal Chemistry

4

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language of work or name

English

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publication date

May 1989

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published in

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volume

32

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issue

5

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page(s)

1043-51

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cites work

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

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cDNA for the human beta 2-adrenergic receptor: a protein with multiple membrane-spanning domains and encoded by a gene whose chromosomal location is shared with that of the receptor for platelet-derived growth factor

20 March 2017

1 reference

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Functionalized congeners of adenosine: preparation of analogues with high affinity for A1-adenosine receptors

20 March 2017

1 reference

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Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes

20 March 2017

1 reference

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Species differences in structure-activity relationships of adenosine agonists and xanthine antagonists at brain A1 adenosine receptors

29 September 2017

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A new high affinity, iodinated adenosine receptor antagonist as a radioligand/photoaffinity crosslinking probe

29 September 2017

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Antagonism of phencyclidine action by metaphit in rat cerebellar Purkinje neurons: an electrophysiological study

29 September 2017

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XAC, a functionalized congener of 1,3-dialkylxanthine, antagonizes A1 adenosine receptor-mediated inhibition of renin secretion in vitro

29 September 2017

1 reference

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8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.

29 September 2017

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Molecular probes for extracellular adenosine receptors

29 September 2017

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[3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors

29 September 2017

1 reference

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Functionalized congeners of 1,3-dialkylxanthines: preparation of analogues with high affinity for adenosine receptors

29 September 2017

1 reference

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Affinity labels for opioid receptors

29 September 2017

1 reference

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A specific acylating agent for the [3H]phencyclidine receptors in rat brain

29 September 2017

1 reference

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The physiological role of adenosine in the central nervous system

29 September 2017

1 reference

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Role of adenine compounds in autonomic neurotransmission

29 September 2017

1 reference

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Evidence that a novel 8-phenyl-substituted xanthine derivative is a cardioselective adenosine receptor antagonist in vivo

29 September 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Metaphit, a receptor acylator, inactivates cocaine binding sites in striatum and antagonizes cocaine-induced locomotor stimulation in rodents.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Metaphit prevents locomotor activation induced by various psychostimulants and interferes with the dopaminergic system in mice

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Metaphit, an acylating ligand for phencyclidine receptors: characterization of in vivo actions in the rat.

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Characterization of the A2 adenosine receptor labeled by [3H]NECA in rat striatal membranes

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Effects of metaphit, a proposed phencyclidine receptor acylator, on catalepsy in pigeons

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

The A1 adenosine receptor. Identification of the binding subunit by photoaffinity cross-linking.

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

The A1 adenosine receptor. Solubilization and characterization of a guanine nucleotide-sensitive form of the receptor

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Phencyclidine (PCP)-like discriminative stimulus effects of metaphit and of 2-amino-5-phosphonovalerate in pigeons: generality across different training doses of PCP.

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Affinity labels for beta-adrenoceptors: preparation and properties of alkylating beta-blockers derived from indole

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Novel irreversible ligands specific for "peripheral" type benzodiazepine receptors: (+/-)-, (+)-, and (-)-1-(2-chlorophenyl)-N-(1-methylpropyl)-N- (2-isothiocyanatoethyl)-3-isoquinolinecarboxamide and 1-(2-isothiocyanatoethyl)-7-chloro-1,3-dihydro-5

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Identification of a Mr 58 000 glycoprotein subunit of the opiate receptor

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for .mu. or .delta. opiate receptors

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Irreversible Ligands with High Selectivity Toward δ and μ Opiate Receptors

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3442263

Kinetics of cholesterol and phospholipid exchange from membranes containing cross-linked proteins or cross-linked phosphatidylethanolamines

27 November 2018

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12 December 2020

A specific alkylating ligand for phencyclidine (PCP) receptors antagonizes PCP behavioral effects

1 reference

12 December 2020

THE AGGREGATION OF BLOOD PLATELETS

1 reference

12 December 2020

Cross-linking of myosin subfragment 1. Nucleotide-enhanced modification by a variety of bifunctional reagents

1 reference

12 December 2020

Visual methods for the nanomolar detection of electrophilic reagents

1 reference

12 December 2020

Solid-phase Edman degradation. The use of p-phenyl diisothiocyanate to attach lysine- and arginine-containing peptides to insoluble resins

1 reference

12 December 2020