(Q28359706)

English

Binding and functional properties of antimuscarinics of the hexocyclium/sila-hexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes

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scholarly article

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Binding and functional properties of antimuscarinics of the hexocyclium/sila-hexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes (English)

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author name string

M Waelbroeck

1

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M Tastenoy

2

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J Camus

3

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J Christophe

4

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C Strohmann

5

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H Linoh

6

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H Zilch

7

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R Tacke

8

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E Mutschler

9

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G Lambrecht

10

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language of work or name

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publication date

September 1989

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British Journal of Pharmacology

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98

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1

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197-205

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

20 March 2017

Some quantitative uses of drug antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

7 April 2017

Antimuscarinic action of methoctramine, a new cardioselective M-2 muscarinic receptor antagonist, alone and in combination with atropine and gallamine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

29 September 2017

A comparison of affinity constants for muscarine-sensitive acetylcholine receptors in guinea-pig atrial pacemaker cells at 29 degrees C and in ileum at 29 degrees C and 37 degrees C

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

29 September 2017

pA2 and receptor differentiation: a statistical analysis of competitive antagonism

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

29 September 2017

Antagonist discrimination between ganglionic and ileal muscarinic receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

Pirenzepine distinguishes between different subclasses of muscarinic receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

Structure-activity relationships of unsaturated esters of arecaidine and dihydroarecaidine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

The relative potencies of some agonists at M2 muscarinic receptors in guinea-pig ileum, atria and bronchi

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

Cardioselective profile of AF-DX 116, a muscarine M2 receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

Binding profile of a novel cardioselective muscarine receptor antagonist, AF-DX 116, to membranes of peripheral tissues and brain in the rat.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

o-Methoxy-sila-hexocyclium: a new quaternary M1-selective muscarinic antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

80% of muscarinic receptors expressed by the NB-OK 1 human neuroblastoma cell line show high affinity for pirenzepine and are comparable to rat hippocampus M1 receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

p-fluoro-hexahydro-sila-difenidol: the first M2 beta-selective muscarinic antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

Methoctramine, a polymethylene tetraamine, differentiates three subtypes of muscarinic receptor in direct binding studies

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1854665

2 June 2018

The origin of acetylcholine released from guinea-pig intestine and longitudinal muscle strips.

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1989.TB16882.X

21 January 2018

Selectivity of muscarinic antagonists in radioligand and in vivo experiments for the putative M1, M2 and M3 receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2804545

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Muscarinic receptor heterogeneity in rat central nervous system. I. Binding of four selective antagonists to three muscarinic receptor subclasses: a comparison with M2 cardiac muscarinic receptors of the C type

1 reference

https://pubmed.ncbi.nlm.nih.gov/2804545

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cumulative dose-response curves. II. Technique for the making of dose-response curves in isolated organs and the evaluation of drug parameters

1 reference

https://pubmed.ncbi.nlm.nih.gov/2804545

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Different antagonist binding properties of rat pancreatic and cardiac muscarinic receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/2804545

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Muscarinic receptor subtypes: M1 and M2 biochemical and functional characterization

1 reference

https://pubmed.ncbi.nlm.nih.gov/2804545

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Sila-substitution--a useful strategy for drug design?

1 reference

https://pubmed.ncbi.nlm.nih.gov/2804545

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.1989.TB16882.X

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