(Q30320568)

English

Lipophilicities of baclofen ester prodrugs correlate with affinities to the ATP-dependent efflux pump P-glycoprotein: relevance for their permeation across the blood-brain barrier?

scientific article published on May 1, 2003

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Lipophilicities of baclofen ester prodrugs correlate with affinities to the ATP-dependent efflux pump P-glycoprotein: relevance for their permeation across the blood-brain barrier? (English)

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

blood–brain barrier

1 reference

based on heuristic

inferred from title

organic chemistry

1 reference

10.1023/A:1023437603555

https://api.crossref.org/works/10.1023/A:1023437603555

3 January 2024

pharmaceutical science

1 reference

10.1023/A:1023437603555

https://api.crossref.org/works/10.1023/A:1023437603555

3 January 2024

1 reference

10.1023/A:1023437603555

https://api.crossref.org/works/10.1023/A:1023437603555

3 January 2024

molecular medicine

1 reference

10.1023/A:1023437603555

https://api.crossref.org/works/10.1023/A:1023437603555

3 January 2024

1 reference

10.1023/A:1023437603555

https://api.crossref.org/works/10.1023/A:1023437603555

3 January 2024

author name string

Christiane Leisen

1

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Peter Langguth

2

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Bernd Herbert

3

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Cornelia Dressler

4

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Annette Koggel

5

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Hilde Spahn-Langguth

6

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

language of work or name

1 reference

National Center for Biotechnology Information

PubMed publication ID

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=12751633

3 January 2024

publication date

1 May 2003

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Pharmaceutical Research

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

20

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

5

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

772-778

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

Study on brain interstitial fluid distribution and blood-brain barrier transport of baclofen in rats by microdialysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Drug transfer across the blood-brain barrier and improvement of brain delivery

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Bisphosphonate prodrugs: synthesis and in vitro evaluation of alkyl and acyloxymethyl esters of etidronic acid as bioreversible prodrugs of etidronate

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Interaction of taurine on baclofen intestinal absorption: a nonlinear mathematical treatment using differential equations to describe kinetic inhibition models.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Molecular and functional identification of large neutral amino acid transporters LAT1 and LAT2 and their pharmacological relevance at the blood-brain barrier

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Transport of valganciclovir, a ganciclovir prodrug, via peptide transporters PEPT1 and PEPT2.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Transporter-mediated permeation of drugs across the blood-brain barrier

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The use of esters as prodrugs for oral delivery of beta-lactam antibiotics

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Expression of a system L neutral amino acid transporter at the blood-brain barrier

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Blood-brain barrier glucose transporter: effects of hypo- and hyperglycemia revisited.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of P-glycoprotein-mediated secretion in absorptive drug permeability: An approach using passive membrane permeability and affinity to P-glycoprotein

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Improved long-term stability of blood cocaine in evacuated collection tubes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The human brain GLUT1 glucose transporter: ultrastructural localization to the blood-brain barrier endothelia.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Selective expression of the large neutral amino acid transporter at the blood-brain barrier

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Improved brain delivery of a nonsteroidal anti-inflammatory drug with a synthetic glyceride ester: a preliminary attempt at a CNS drug delivery system for the therapy of Alzheimer's disease.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Stereoselective transport of baclofen across the blood-brain barrier in rats as determined by the unit impulse response methodology

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

P-glycoprotein: a defense mechanism limiting oral bioavailability and CNS accumulation of drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The blood-brain barrier and oncology: new insights into function and modulation

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Brain microvascular P-glycoprotein and a revised model of multidrug resistance in brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/12751633

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1023/A:1023437603555

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

17 June 2017

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