(Q31440471)

English

Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives: a novel series of mixed dopamine D2/D4 receptor antagonists

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scholarly article

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Europe PubMed Central

PubMed publication ID

2 July 2017

Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives: a novel series of mixed dopamine D2/D4 receptor antagonists (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

author name string

Zhao H

1

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

Thurkauf A

2

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

Braun J

3

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

Brodbeck R

4

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

Kieltyka A

5

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

language of work or name

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publication date

1 September 2000

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Europe PubMed Central

PubMed publication ID

2 July 2017

Bioorganic & Medicinal Chemistry Letters

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Europe PubMed Central

PubMed publication ID

2 July 2017

10

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

18

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

2119-2122

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

Dopamine receptor pharmacology

1 reference

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Molecular cloning and expression of the gene for a human D1 dopamine receptor

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Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1

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Cloning and expression of a rat D2 dopamine receptor cDNA

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Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics

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Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine

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D4 receptors and their antagonists

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Isoindolinone enantiomers having affinity for the dopamine D4 receptor

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SAR of novel biarylmethylamine dopamine D4 receptor ligands

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4-N-linked-heterocyclic piperidine derivatives with high affinity and selectivity for human dopamine D4 receptors

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2,2-dicyanovinyl as a nonaromatic aryl bioisostere: synthesis, binding experiments and SAR studies of highly selective dopamine D4 receptor ligands

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Piperidinylpyrroles: Design, synthesis and binding properties of novel and selective dopamine D4 receptor ligands

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1-(3-Cyanobenzylpiperidin-4-yl)-5-methyl-4-phenyl-1, 3-dihydroimidazol-2-one: a selective high-affinity antagonist for the human dopamine D(4) receptor with excellent selectivity over ion channels

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Design, synthesis, and evaluation of chromen-2-ones as potent and selective human dopamine D4 antagonists

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A series of 6- and 7-piperazinyl- and -piperidinylmethylbenzoxazinones with dopamine D4 antagonist activity: discovery of a potential atypical antipsychotic agent

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A structure-affinity relationship study on derivatives of N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a high-affinity and selective D(4) receptor ligand.

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2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors

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(S)-(-)-4-[4-[2-(isochroman-1-yl)ethyl]-piperazin-1-yl] benzenesulfonamide, a selective dopamine D4 antagonist

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Synthesis, SAR and pharmacology of CP-293,019: a potent, selective dopamine D4 receptor antagonist

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Centrally acting dopamine D2 receptor ligands: agonists

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New generation dopaminergic agents. 6. Structure-activity relationship studies of a series of 4-(aminoethoxy)indole and 4-(aminoethoxy)indolone derivatives based on the newly discovered 3-hydroxyphenoxyethylamine D2 template.

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Identifiers

10.1016/S0960-894X(00)00421-2

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

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