(Q31561831)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

title

Constitutive activity at serotonin 5-HT(1D) receptors: detection by homologous GTPgammaS versus [(35)S]-GTPgammaS binding isotherms (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

author

Adrian Newman-Tancredi

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

author name string

V Audinot

series ordinal

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

M J Millan

series ordinal

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

publication date

1 January 2001

1 reference

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2 November 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

volume

40

1 reference

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2 November 2019

issue

1

1 reference

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2 November 2019

page(s)

57-64

1 reference

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Binding profile of the novel 5-HT1B/1D receptor antagonist, [3H]GR 125,743, in guinea-pig brain: a comparison with [3H]5-carboxamidotryptamine

2 November 2019

cites work

1 reference

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Physiological effects of inverse agonists in transgenic mice with myocardial overexpression of the beta 2-adrenoceptor

7 January 2021

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Cannabinoid receptor agonist efficacy for stimulating [35S]GTPgammaS binding to rat cerebellar membranes correlates with agonist-induced decreases in GDP affinity.

7 January 2021

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Characterization of human serotonin 1D and 1B receptors using [3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist

7 January 2021

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Pharmacological analysis of dopamine stimulation of [35S]-GTP gamma S binding via human D2short and D2long dopamine receptors expressed in recombinant cells

7 January 2021

1 reference

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The selective 5-HT1B receptor inverse agonist 1'-methyl-5-[[2'-methyl-4'-(5-methyl-1,2, 4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) potently blocks terminal 5-HT autoreceptor func

7 January 2021

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G protein-coupled receptors. II. Mechanism of agonist activation

7 January 2021

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Antipsychotics with inverse agonist activity at the dopamine D3 receptor

7 January 2021

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Diversity and selectivity of receptor-G protein interaction

7 January 2021

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Muscarinic acetylcholine receptor-stimulated binding of guanosine 5'-O-(3-thiotriphosphate) to guanine-nucleotide-binding proteins in cardiac membranes

7 January 2021

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Dissociation of guanosine 5'-[gamma-thio]triphosphate from guanine-nucleotide-binding regulatory proteins in native cardiac membranes. Regulation by nucleotides and muscarinic acetylcholine receptors

7 January 2021

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Estimation of antagonist Kb from inhibition curves in functional experiments: alternatives to the Cheng-Prusoff equation.

7 January 2021

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Pharmacological characterization of guanine nucleotide exchange reactions in membranes from CHO cells stably transfected with human muscarinic receptors m1-m4

7 January 2021

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Mechanisms of agonism and inverse agonism at serotonin 5-HT1A receptors

7 January 2021

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The induction of pain: an integrative review

7 January 2021

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Inhibition of the constitutive activity of human 5-HT1A receptors by the inverse agonist, spiperone but not the neutral antagonist, WAY 100,635

7 January 2021

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Agonist and inverse agonist efficacy at human recombinant serotonin 5-HT1A receptors as a function of receptor:G-protein stoichiometry

7 January 2021

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Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study

7 January 2021

1 reference

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Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists

7 January 2021

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Inverse agonism at dopamine D2 receptors. Haloperidol-induced prolactin release from GH4C1 cells transfected with the human D2 receptor is antagonized by R(-)-n-propylnorapomorphine, raclopride, and phenoxybenzamine

7 January 2021

1 reference

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Stimulated [35S]GTP gamma S binding by 5-HT1A receptor agonists in recombinant cell lines. Modulation of apparent efficacy by G-protein activation state

7 January 2021

1 reference

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How efficacious are 5-HT1B/D receptor ligands: an answer from GTP gamma S binding studies with stably transfected C6-glial cell lines

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2800%2900104-0

Pharmacological analysis of G-protein activation mediated by guinea-pig recombinant 5-HT1B receptors in C6-glial cells: similarities with the human 5-HT1B receptor

7 January 2021

1 reference

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SB-224289--a novel selective (human) 5-HT1B receptor antagonist with negative intrinsic activity

7 January 2021

1 reference

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Pharmacological characterisation of [35S]-GTPgammaS binding to Chinese hamster ovary cell membranes stably expressing cloned human 5-HT1D receptor subtypes

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2800%2900104-0

10.1016/S0028-3908(00)00104-0

7 January 2021

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11077071%20AND%20SRC:MED&resulttype=core&format=json

2 November 2019

1 reference