(Q33213253)

24 July 2017

title

GPCR antitarget modeling: pharmacophore models for biogenic amine binding GPCRs to avoid GPCR-mediated side effects (English)

1 reference

G protein-coupled receptor

24 July 2017

main subject

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author name string

Thomas Klabunde

series ordinal

1

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24 July 2017

Andreas Evers

series ordinal

2

1 reference

24 July 2017

publication date

1 May 2005

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24 July 2017

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24 July 2017

volume

6

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24 July 2017

issue

5

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24 July 2017

page(s)

876-889

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Drug design strategies for targeting G-protein-coupled receptors

24 July 2017

cites work

1 reference

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21 January 2018

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Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes

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Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist

21 January 2018

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Characterization of an α1D‐adrenoceptor mediating the contractile response of rat aorta to noradrenaline

21 January 2018

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Influence of chain length and N-alkylation on the selective serotonin receptor ligand 9-(aminomethyl)-9,10-dihydroanthracene

21 January 2018

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Binding of 5H-dibenzo[b,e][1,4]diazepine and chiral 5H-dibenzo[a,d]cycloheptene analogues of clozapine to dopamine and serotonin receptors

21 January 2018

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21 January 2018

Identifiers

DOI

10.1002/CBIC.200400369

1 reference

24 July 2017

1 reference