(Q33793201)

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Drugs acting on imidazoline receptors: a review of their pharmacology, their use in blood pressure control and their potential interest in cardioprotection

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scholarly article

1 reference

Europe PubMed Central

29 July 2017

1 reference

Europe PubMed Central

Drugs acting on imidazoline receptors: a review of their pharmacology, their use in blood pressure control and their potential interest in cardioprotection (English)

1 reference

Europe PubMed Central

29 July 2017

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author name string

P Bousquet

1

1 reference

Europe PubMed Central

29 July 2017

J Feldman

2

1 reference

Europe PubMed Central

29 July 2017

publication date

1 November 1999

1 reference

Europe PubMed Central

29 July 2017

1 reference

Europe PubMed Central

29 July 2017

58

1 reference

Europe PubMed Central

29 July 2017

5

1 reference

Europe PubMed Central

29 July 2017

799-812

1 reference

Europe PubMed Central

29 July 2017

https://scigraph.springernature.com/pub.10.2165/00003495-199958050-00003

0 references

Effects of clonidine and other imidazole-receptor binding agents on second messenger systems and calcium influx in bovine adrenal chromaffin cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antihypertensive efficacy and acceptability of rilmenidine in elderly hypertensive patients

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence for the involvement of imidazoline receptors in the central hypotensive effect of rilmenidine in the rabbit

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of Swim Training Alone and in Combination with Clonidine and Rilmenidine on Blood Pressure, Plasma Electrolytes, Vasopressin, and Renin Activity in Spontaneously Hypertensive Rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Suppressing sympathetic activation with clonidine on ventricular arrhythmias in congestive heart failure

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Efficacy and safety of rilmenidine for arterial hypertension.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence that locus coeruleus is the site where clonidine and drugs acting at alpha 1- and alpha 2-adrenoceptors affect sleep and arousal mechanisms

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Treatment of systemic hypertension in insulin-treated diabetes mellitus with rilmenidine.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Differences in the ability of yohimbine to antagonize the hypotensive effect of clonidine in normotensive and spontaneously hypertensive anesthetized rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The nucleus reticularis lateralis: a region highly sensitive to clonidine

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Complementary antihypertensive action of rilmenidine on the pressure-natriuresis relationship and sodium preference in spontaneously hypertensive rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Inhibition of centrally induced ventricular arrhythmias by rilmenidine and idazoxan in rabbits

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antihypertensive drugs and baroreflex sensitivity. Effects of rilmenidine

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Involvement of alpha 2-adrenoceptors in the cardiovascular effects of moxonidine

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Suppressing sympathetic activation in congestive heart failure. A new therapeutic strategy.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Acceptability of rilmenidine and long-term surveillance of plasma concentrations in hypertensive patients with renal insufficiency.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

I1-imidazoline receptors. Definition, characterization, distribution, and transmembrane signaling

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of a partial cDNA clone detected by imidazoline receptor-selective antisera

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Sympathoinhibitory action of rilmenidine in conscious sinoaortically denervated rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Moxonidine inhibits Na+/H+ exchange in proximal tubule cells and cortical collecting duct

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Rilmenidine selectivity for imidazoline receptors in human brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Clonidine withdrawal in hypertension. Changes in blood-pressure and plasma and urinary noradrenaline

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mediation of the hypotensive action of systemic clonidine in the rat by alpha 2-adrenoceptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cardiovascular and central nervous system effects of rilmenidine (S 3341) in rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Isolation and partial purification of a clonidine-displacing endogenous brain substance

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Comparative effects of rilmenidine and atenolol on tests of autonomic function and mental and dynamic exercise in patients with essential hypertension.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Catecholamines and their blockade in congestive heart failure

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological properties of (N-dicyclopropylmethyl) amino-2-oxazoline (S 3341), an alpha-2 adrenoceptor agonist.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Moxonidine and hydrochlorothiazide in combination: a synergistic antihypertensive effect

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effect of imidazolines on Na+ transport and intracellular pH in renal proximal tubule cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Localization of the imidazoline binding domain on monoamine oxidase B

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Crossover comparison of moxonidine and clonidine in mild to moderate hypertension

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Correlation between the inhibitory effect on catecholaminergic ventrolateral medullary neurons and the hypotension evoked by clonidine: a voltammetric approach

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multicenter, double-blind study comparing rilmenidine 1 mg and hydrochlorothiazide 25 mg in 244 patients

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification, localization and functional analysis of imidazoline and alpha adrenergic receptors in canine prostate.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A multicenter double-blind comparative study of rilmenidine and clonidine in 333 hypertensive patients

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effort blood pressure control in the course of antihypertensive treatment

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[Long-term experiences with moxonidine, a new antihypertensive agent]

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Selectivity of rilmenidine for the nucleus reticularis lateralis, a ventrolateral medullary structure containing imidazoline-preferring receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Relative importance of central imidazoline receptors for the antihypertensive effects of moxonidine and rilmenidine

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antiarrhythmic action of rilmenidine on adrenaline-induced arrhythmia via central imidazoline receptors in halothane-anaesthetized dogs

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The I1-imidazoline-binding site is a functional receptor mediating vasodepression via the ventral medulla.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Moxonidine, a centrally acting antihypertensive agent, is a selective ligand for I1-imidazoline sites.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Imidazoline receptors and their endogenous ligands

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A comparison of the haemodynamic and behavioural effects of moxonidine and clonidine in normotensive subjects

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Activation of phosphatidylcholine-selective phospholipase C by I1-imidazoline receptors in PC12 cells and rostral ventrolateral medulla.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Dose and concentration-effect relations for rilmenidine

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Agmatine: an endogenous clonidine-displacing substance in the brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[Moxonidine vs. captopril in minor to intermediate hypertension. Double-blind study of effectiveness and tolerance]

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Site and receptors involved in the sympathoinhibitory actions of rilmenidine

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Rilmenidine in patients with left ventricular hypertrophy: beyond the reduction of left ventricular mass

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Placebo-controlled comparison of the efficacy and tolerability of once-daily moxonidine and enalapril in mild-to-moderate essential hypertension

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of imidazoline receptors in the cardiovascular actions of moxonidine, rilmenidine and clonidine in conscious rabbits.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Rilmenidine-induced hypotension in conscious rabbits involves imidazoline-preferring receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The I1-imidazoline receptor: from binding site to therapeutic target in cardiovascular disease

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regression of left ventricular hypertrophy

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Participation of imidazoline receptors and alpha(2-)-adrenoceptors in the central hypotensive effects of imidazoline-like drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Is the hypotensive effect of clonidine and related drugs due to imidazoline binding sites?

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Chronic Sympathetic Suppression in the Treatment of Chronic Congestive Heart Failure

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Twenty-four-hour blood pressure profiles in patients with mild-to-moderate hypertension: moxonidine versus captopril.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Central and peripheral effects of S 3341 [(N-dicyclopropylmethyl)-amino-2-oxazoline] in animal models

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effect of moxonidine on urinary electrolyte excretion and renal haemodynamics in man.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification of human I1 receptors and their relationship to alpha 2-adrenoceptors.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Sympathetic inhibition with clonidine improves autonomic balance in congestive heart failure

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Imidazoline receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effect of moxonidine on arrhythmias induced by coronary artery occlusion and reperfusion

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Rilmenidine and vigilance. Review of clinical studies

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Preventive effect of rilmenidine on the occurrence of neurogenic ventricular arrhythmias in rabbits

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Efficacy and acceptability of rilmenidine for mild to moderate systemic hypertension

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence for the existence of imidazoline-specific binding sites in synaptosomal plasma membranes of the bovine brainstem.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Renal effects of rilmenidine in anesthetized rats: importance of renal nerves.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Autonomic nervous system and sudden cardiac death

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Central cardiovascular effects of alpha adrenergic drugs: differences between catecholamines and imidazolines

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regression of left ventricular hypertrophy in hypertensive patients after 1 year of treatment with rilmenidine: a double-blind, randomized, controlled (versus nifedipine) study

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Comparison of ligand binding affinities at human I1-imidazoline binding sites and the high affinity state of alpha-2 adrenoceptor subtypes

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Central hypotensive effects of the alpha2a-adrenergic receptor subtype.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

I2-imidazoline binding sites: relationship with different monoamine oxidase domains and identification of histidine residues mediating ligand binding regulation by H+1

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of imidazole receptors in the vasodepressor response to clonidine analogs in the rostral ventrolateral medulla.

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The effects of rilmenidine on tests of autonomic function in humans

1 reference

https://pubmed.ncbi.nlm.nih.gov/10595861

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.2165/00003495-199958050-00003

1 reference

Europe PubMed Central

29 July 2017

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0 references

release_xlu2vpvl6vgy5n73ipgkhjpbei

1 reference

https://api.fatcat.wiki/v0/release/xlu2vpvl6vgy5n73ipgkhjpbei

24 November 2022

based on heuristic

mapped directly with Wikidata item

1 reference

Europe PubMed Central

29 July 2017

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