(Q33796345)

29 July 2017

A high-throughput fluorescence polarization assay for inhibitors of gyrase B (English)

1 reference

29 July 2017

Bryan T Glaser

1

1 reference

29 July 2017

Jeremiah P Malerich

2

1 reference

29 July 2017

Sarah J Duellman

3

1 reference

29 July 2017

Julie Fong

4

1 reference

29 July 2017

Christopher Hutson

5

1 reference

29 July 2017

Richard M Fine

6

1 reference

29 July 2017

Boris Keblansky

7

1 reference

29 July 2017

Mary J Tang

8

1 reference

29 July 2017

Peter B Madrid

9

1 reference

29 July 2017

18 January 2011

1 reference

Journal of Biomolecular Screening

29 July 2017

1 reference

29 July 2017

16

1 reference

29 July 2017

2

1 reference

29 July 2017

230-238

1 reference

Chromosomal aberration and micronucleus studies of two topoisomerase (II) targeting anthracyclines

29 July 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

A high-throughput assay for DNA topoisomerases and other enzymes, based on DNA triplex formation.

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Effect of the anti-neoplastic drug doxorubicin on XPD-mutated DNA repair-deficient human cells

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Discovery and development of ATPase inhibitors of DNA gyrase as antibacterial agents

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Thirty years of Escherichia coli DNA gyrase: from in vivo function to single-molecule mechanism.

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Recent advances in understanding structure–function relationships in the type II topoisomerase mechanism

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

The complete genome sequence of Francisella tularensis, the causative agent of tularemia

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

A general framework for development and data analysis of competitive high-throughput screens for small-molecule inhibitors of protein-protein interactions by fluorescence polarization

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Active-site residues of Escherichia coli DNA gyrase required in coupling ATP hydrolysis to DNA supercoiling and amino acid substitutions leading to novobiocin resistance

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

An open conformation of the Thermus thermophilus gyrase B ATP-binding domain

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Fluorescence polarization and anisotropy in high throughput screening: perspectives and primer

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Novel inhibitors of DNA gyrase: 3D structure based biased needle screening, hit validation by biophysical methods, and 3D guided optimization. A promising alternative to random screening

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

The entropic penalty of ordered water accounts for weaker binding of the antibiotic novobiocin to a resistant mutant of DNA gyrase: a thermodynamic and crystallographic study

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Recent developments in DNA topoisomerase II structure and mechanism

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Variation of the supercoils in closed circular DNA by binding of antibiotics and drugs: Evidence for molecular models involving intercalation

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

The mode of action of 4-quinolones and possible mechanisms of resistance

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Mechanisms of action of and resistance to ciprofloxacin

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Energy coupling in DNA gyrase and the mechanism of action of novobiocin

4 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Development and use of a high-throughput bacterial DNA gyrase assay to identify mammalian topoisomerase II inhibitors with whole-cell anticancer activity

4 July 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057110392038

A high-throughput, homogeneous, bioluminescent assay for Pseudomonas aeruginosa gyrase inhibitors and other DNA-damaging agents

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057110392038

A scintillation proximity assay amenable for screening and characterization of DNA gyrase B subunit inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057110392038

Novel dual-targeting benzimidazole urea inhibitors of DNA gyrase and topoisomerase IV possessing potent antibacterial activity: intelligent design and evolution through the judicious use of structure-guided design and structure-activity relationship

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057110392038

Anthracycline-dependent heat-induced transition from positive to negative supercoiled DNA.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057110392038

Tryptic fragments of the Escherichia coli DNA gyrase A protein.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3176662

Characterization of the binding site for cyclothialidine on the B subunit of DNA gyrase

30 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21245469

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

DNA topoisomerase II-mediated interaction of doxorubicin and daunorubicin congeners with DNA

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21245469

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Interaction specificity of the anthracyclines with deoxyribonucleic acid

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21245469

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1177/1087057110392038

1 reference

29 July 2017

1 reference

29 July 2017

1 reference