(Q33867215)

29 July 2017

title

Synthesis and characterization of fluorescent 4-hydroxytamoxifen conjugates with unique antiestrogenic properties (English)

1 reference

29 July 2017

Emily L Rickert

1

1 reference

29 July 2017

Sean Oriana

2

1 reference

29 July 2017

Cori Hartman-Frey

3

1 reference

29 July 2017

Xinghua Long

4

1 reference

29 July 2017

Timothy T Webb

5

1 reference

29 July 2017

Kenneth P Nephew

6

1 reference

29 July 2017

Ross V Weatherman

7

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29 July 2017

publication date

1 May 2010

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29 July 2017

published in

Bioconjugate Chemistry

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29 July 2017

volume

21

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29 July 2017

issue

5

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29 July 2017

page(s)

903-910

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describes a project that uses

29 July 2017

ImageJ

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC2874112/fullTextXML

inferred from PubMed Central ID database lookup

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5 July 2018

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Estrogen receptor-alpha hinge-region lysines 302 and 303 regulate receptor degradation by the proteasome

5 July 2018

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Synthesis and characterization of bioactive tamoxifen-conjugated polymers

5 July 2018

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Synthetic estrogen derivatives demonstrate the functionality of intracellular GPR30.

5 July 2018

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SERMs: meeting the promise of multifunctional medicines

5 July 2018

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Diverse gene expression and DNA methylation profiles correlate with differential adaptation of breast cancer cells to the antiestrogens tamoxifen and fulvestrant

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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A transmembrane intracellular estrogen receptor mediates rapid cell signaling

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Intracellular dynamics of steroid hormone receptor

5 July 2018

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Differential effects of estradiol and estradiol-BSA conjugates

5 July 2018

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The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

5 July 2018

1 reference

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Identification of a new class of steroid hormone receptors

5 July 2018

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Estradiol membrane binding sites on human breast cancer cell lines. Use of a fluorescent estradiol conjugate to demonstrate plasma membrane binding systems

5 July 2018

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Donor-acceptor tetrahydrochrysenes, inherently fluorescent, high-affinity ligands for the estrogen receptor: binding and fluorescence characteristics and fluorometric assay of receptor

5 July 2018

1 reference

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Specific binding sites for oestrogen at the outer surfaces of isolated endometrial cells

5 July 2018

1 reference

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Fulvestrant (ICI 182,780)-dependent interacting proteins mediate immobilization and degradation of estrogen receptor-alpha

5 July 2018

1 reference

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Estrogen dendrimer conjugates that preferentially activate extranuclear, nongenomic versus genomic pathways of estrogen action

29 October 2018

1 reference

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Activity of a tamoxifen-raloxifene hybrid ligand for estrogen receptors at an AP-1 site

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2874112

Differential SERM activation of the estrogen receptors (ERalpha and ERbeta) at AP-1 sites

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2874112

Tamoxifen perturbs lipid bilayer order and permeability: comparison of DSC, fluorescence anisotropy, laurdan generalized polarization and carboxyfluorescein leakage studies

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2874112

Cytochemical demonstration of estrogen binding sites in breast cancer by estradiol covalently linked to horseradish peroxidase

29 October 2018

1 reference

12 December 2020

Analogues of tamoxifen: the role of the basic side-chain. Applications of a whole-cell oestrogen-receptor binding assay to N-oxides and quaternary salts

1 reference

12 December 2020

Studies using fluorescent tetrahydrochrysene estrogens for in situ visualization of the estrogen receptor in living cells

1 reference

12 December 2020

Antiestrogen basicity--activity relationships: a comparison of the estrogen receptor binding and antiuterotrophic potencies of several analogues of (Z)-1,2-diphenyl-1-[4-[2-(dimethylamino)ethoxy]phenyl]-1-butene (tamoxifen, Nolvadex) having altered

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12 December 2020

Chemoprevention of breast cancer with selective oestrogen-receptor modulators

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12 December 2020

Facile geometric isomerization of phenolic non-steroidal estrogens and antiestrogens: limitations to the interpretation of experiments characterizing the activity of individual isomers

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12 December 2020

Estrogen and antiestrogen action: studies in reproductive target tissues and tumors

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12 December 2020

Fluoresceinated estrone binding by human and mouse breast cancer cells

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12 December 2020

Receptor binding of NBD-labeled fluorescent estrogens and progestins in whole cells and cell-free preparations

1 reference

12 December 2020

Tamoxifen-based probes for the study of estrogen receptor-mediated transcription

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12 December 2020

Identifiers

DOI

10.1021/BC900461H

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29 July 2017

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29 July 2017

1 reference