(Q34125185)

31 July 2017

1 reference

title

H1-antihistamines: inverse agonism, anti-inflammatory actions and cardiac effects (English)

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31 July 2017

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R Leurs

1

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31 July 2017

M K Church

series ordinal

2

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31 July 2017

M Taglialatela

series ordinal

3

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31 July 2017

language of work or name

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1 April 2002

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Clinical & Experimental Allergy

31 July 2017

published in

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31 July 2017

volume

32

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31 July 2017

issue

4

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31 July 2017

page(s)

489-498

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Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

31 July 2017

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High constitutive activity of native H3 receptors regulates histamine neurons in brain.

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21 January 2018

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21 January 2018

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Postnatal expression of H1-receptor mRNA in the rat brain: correlation to L-histidine decarboxylase expression and local upregulation in limbic seizures

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Inhibition of histamine release from human lung in vitro by antihistamines and related drugs

21 January 2018

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In vitro effects of H1-antihistamines on histamine and PGD2 release from mast cells of human lung, tonsil, and skin

21 January 2018

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Divalent cation dependence of the inhibition by phenothiazines of mediator release from mast cells

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Effects of the anti-allergics astemizole and norastemizole on Fc epsilon RI receptor-mediated signal transduction processes

21 January 2018

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Structure-activity relationships of astemizole derivatives for inhibition of store operated Ca2+ channels and exocytosis

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Action of azelastine on intracellular Ca2+ in cultured airway smooth muscle

21 January 2018

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Inhibitory effect of oral cetirizine on in vivo antigen-induced histamine and PAF-acether release and eosinophil recruitment in human skin

21 January 2018

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21 January 2018

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Nedocromil sodium and levocabastine reduce the symptoms of conjunctival allergen challenge by different mechanisms

21 January 2018

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Effects of capsaicin, bradykinin and prostaglandin E2 in the human skin

21 January 2018

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Effects of H1 antagonists on the cutaneous vascular response to histamine and bradykinin: a study using scanning laser Doppler imaging

21 January 2018

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Human skin mast cells: in vitro and in vivo studies

21 January 2018

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Mechanisms of mediator release from human skin mast cells upon stimulation by the bradykinin analog, [dArg0-Hyp3-dPhe7]bradykinin

21 January 2018

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21 January 2018

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Platelet-activating factor induces histamine release from human skin mast cells in vivo, which is reduced by local nerve blockade

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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AT1-receptor heterodimers show enhanced G-protein activation and altered receptor sequestration

21 January 2018

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Cardiotoxic effect with convulsions in terfenadine overdose

21 January 2018

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Risk of torsades de pointes with non-cardiac drugs. Doctors need to be aware that many drugs can cause qt prolongation

21 January 2018

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Positional cloning of a novel potassium channel gene: KVLQT1 mutations cause cardiac arrhythmias

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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MiRP1 forms IKr potassium channels with HERG and is associated with cardiac arrhythmia

21 January 2018

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A distinct potassium channel polypeptide encoded by the Drosophila eag locus

21 January 2018

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A mechanistic link between an inherited and an acquired cardiac arrhythmia: HERG encodes the IKr potassium channel

21 January 2018

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HERG, a primary human ventricular target of the nonsedating antihistamine terfenadine

21 January 2018

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21 January 2018

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21 January 2018

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QT lengthening and life-threatening arrhythmias associated with fexofenadine

21 January 2018

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Torsade de pointes with an antihistamine metabolite: potassium channel blockade with desmethylastemizole

21 January 2018

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New insights into the second generation antihistamines

21 January 2018

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Inhibition of HERG1 K(+) channels by the novel second-generation antihistamine mizolastine

21 January 2018

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Cardiotoxic potential and CNS effects of first-generation antihistamines.

21 January 2018

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Risk of developing life-threatening ventricular arrhythmia associated with tefenadine in comparison with over-the-counter antihistamines, ibuprofen and clemastine

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.0954-7894.2002.01314.X

A structural basis for drug-induced long QT syndrome

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.0954-7894.2002.01314.X

HERG K+ channels: friend and foe.

21 January 2018

1 reference

https://api.crossref.org/works/10.1046%2FJ.0954-7894.2002.01314.X

10.1046/J.0954-7894.2002.01314.X

21 January 2018

Identifiers

DOI

1 reference

31 July 2017

1 reference