(Q34174011)

31 July 2017

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title

Regulation of 5-HT1A receptor function in brain following agonist or antidepressant administration (English)

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31 July 2017

Julie G Hensler

1

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PubMed ID

12559389

31 July 2017

language of work or name

English

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publication date

1 February 2003

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31 July 2017

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31 July 2017

72

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31 July 2017

15

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31 July 2017

1665-1682

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Electrophysiology of the central serotonin system: receptor subtypes and transducer mechanisms.

31 July 2017

1 reference

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The 5-HT1A receptor: signaling, desensitization, and gene transcription

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A G protein couples serotonin and GABAB receptors to the same channels in hippocampus.

7 January 2021

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Novel anxiolytics discriminate between postsynaptic serotonin receptors mediating different physiological responses on single neurons of the rat hippocampus.

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How does pindolol improve antidepressant action?

7 January 2021

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Acceleration of the effect of selected antidepressant drugs in major depression by 5-HT1A antagonists.

7 January 2021

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Reconstitution of receptors and GTP-binding regulatory proteins (G proteins) in Sf9 cells. A direct evaluation of selectivity in receptor.G protein coupling

7 January 2021

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A single dose of 8-OH-DPAT reduces raphe binding of [3H]8-OH-DPAT and increases the effect of raphe stimulation on 5-HT metabolism

7 January 2021

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Effects of sustained administration of the serotonin and norepinephrine reuptake inhibitor venlafaxine: I. in vivo electrophysiological studies in the rat

7 January 2021

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Attenuation of 5-HT1A and 5-HT2 but not 5-HT1C receptor mediated behaviour in rats following chronic treatment with 5-HT receptor agonists, antagonists or antidepressants

7 January 2021

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Effect of chronic tricylic antidepressant treatment on the serotoninergic autoreceptor: a microiontophoretic study in the rat

7 January 2021

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Electrophysiological investigations on the effect of repeated zimelidine administration on serotonergic neurotransmission in the rat

7 January 2021

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Serotoninergic but not noradrenergic neurons in rat central nervous system adapt to long-term treatment with monoamine oxidase inhibitors.

7 January 2021

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Modification of 5-HT neuron properties by sustained administration of the 5-HT1A agonist gepirone: electrophysiological studies in the rat brain.

7 January 2021

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Current advances and trends in the treatment of depression

7 January 2021

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Piperazine derivatives including the putative anxiolytic drugs, buspirone and ipsapirone, are agonists at 5-HT1A receptors negatively coupled with adenylate cyclase in hippocampal neurons

7 January 2021

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Regulatory mechanisms that modulate signalling by G-protein-coupled receptors

7 January 2021

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Postsynaptic 5-HT1A receptors mediate 5-hydroxytryptamine release in the amygdala through a feedback to the caudal linear raphe.

7 January 2021

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Acute and chronic effects of citalopram on postsynaptic 5-hydroxytryptamine(1A) receptor-mediated feedback: a microdialysis study in the amygdala

7 January 2021

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The inhibitory effect of 8-OH-DPAT on the firing activity of dorsal raphe serotoninergic neurons in rats is attenuated by lesion of the frontal cortex.

7 January 2021

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Control of dorsal raphe serotonergic neurons by the medial prefrontal cortex: Involvement of serotonin-1A, GABA(A), and glutamate receptors.

7 January 2021

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Effects of a selective 5-HT reuptake blocker, citalopram, on the sensitivity of 5-HT autoreceptors: electrophysiological studies in the rat brain

7 January 2021

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Differential effects of protein kinase C activation on 5-HT1A receptor coupling to Ca2+ and K+ currents in rat serotonergic neurones.

7 January 2021

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Serotonin decreases population spike amplitude in hippocampal cells through a pertussis toxin substrate

7 January 2021

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Electrophysiological evidence for a large receptor reserve for inhibition of dorsal raphe neuronal firing by 5-HT1A agonists.

7 January 2021

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Tricyclic antidepressants: long-term treatment increases responsivity of rat forebrain neurons to serotonin.

7 January 2021

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Electrophysiologically-identified serotonin receptors in the rat CNS. Effect of antidepressant treatment

7 January 2021

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5-HT1A receptor agonists: recent developments and controversial issues

7 January 2021

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Effect of acute and repeated versus sustained administration of the 5-HT1A receptor agonist ipsapirone: electrophysiological studies in the rat hippocampus and dorsal raphe.

7 January 2021

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Altered regulation of the 5-HT system in the brain of MAO-A knock-out mice

7 January 2021

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Altered expression and functions of serotonin 5-HT1Aand 5-HT1Breceptors in knock-out mice lacking the 5-HT transporter

7 January 2021

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Homeostatic regulation of serotonergic function by the serotonin transporter as revealed by nonviral gene transfer.

7 January 2021

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Alteration of 5-HT1A receptor binding sites following chronic treatment with ipsapirone measured by quantitative autoradiography.

7 January 2021

1 reference

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Comparative study of pre- and postsynaptic 5-HT1A receptor modulation of anxiety in two ethological animal tests.

7 January 2021

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Pharmacology of Antidepressants

7 January 2021

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Inhibition of 5-HT cell firing in the DRN by non-selective 5-HT reuptake inhibitors: studies on the role of 5-HT1A autoreceptors and noradrenergic mechanisms.

7 January 2021

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Tandospirone and its metabolite, 1-(2-pyrimidinyl)-piperazine--I. Effects of acute and long-term administration of tandospirone on serotonin neurotransmission.

7 January 2021

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The pharmacology of the hypothermic response in mice to 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT). A model of presynaptic 5-HT1 function.

7 January 2021

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Attenuation by electroconvulsive shock and antidepressant drugs of the 5-HT1A receptor-mediated hypothermia and serotonin syndrome produced by 8-OH-DPAT in the rat.

7 January 2021

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Identification of presynaptic serotonin autoreceptors using a new ligand: 3H-PAT

7 January 2021

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Effects of chronically administered venlafaxine on 5-HT receptor activity in rat hippocampus and hypothalamus

7 January 2021

1 reference

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Role of the medial prefrontal cortex in 5-HT1A receptor-induced inhibition of 5-HT neuronal activity in the rat.

7 January 2021

1 reference

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Differential regulation of 5-HT1A receptor-G protein interactions in brain following chronic antidepressant administration

7 January 2021

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Regulation of 5-HT(1A) receptor-stimulated [35S]-GtpgammaS binding as measured by quantitative autoradiography following chronic agonist administration

7 January 2021

1 reference

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Desensitization of 5-HT(1A) autoreceptors by a low chronic fluoxetine dose effect of the concurrent administration of WAY-100635.

7 January 2021

1 reference

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Pharmacokinetics of venlafaxine and O-desmethylvenlafaxine in laboratory animals

7 January 2021

1 reference

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Pertussis toxin blocks 5-HT1A and GABAB receptor-mediated inhibition of serotonergic neurons.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

[3H]8-OH-DPAT labels a 5-HT site coupled to inhibition of phosphoinositide hydrolysis in the dorsal raphe.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Long lasting attenuation of 8-OH-DPAT-induced corticosterone secretion after a single injection of a 5-HT1A receptor agonist

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Single administration of 5-HT1A agonists decreases 5-HT1A presynaptic, but not postsynaptic receptor-mediated responses: relationship to antidepressant-like action

7 January 2021

1 reference

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5-HT1A receptor activation and antidepressant-like effects: F 13714 has high efficacy and marked antidepressant potential

7 January 2021

1 reference

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5-Hydroxytryptamine1A receptor-mediated effects of buspirone, gepirone and ipsapirone

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Chronic administration of the 5-HT1A receptor agonist 8-OH-DPAT differentially desensitizes 5-HT1A autoreceptors of the dorsal and median raphe nuclei.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Different effects on the responses of functional pre- and postsynaptic 5-HT1A receptors by repeated treatment of rats with the 5-HT1A receptor agonist 8-OH-DPAT

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Differential adaptation of brain 5-HT1A and 5-HT1B receptors and 5-HT transporter in rats treated chronically with fluoxetine

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Regulation of G proteins by chronic antidepressant drug treatment in rat brain: tricyclics but not clorgyline increase Goα subunits

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

5-HT1A receptor function in depression: effect of chronic amitriptyline treatment

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Autoradiographic evidence for differential G-protein coupling of 5-HT1A receptors in rat brain: lack of effect of repeated injections of fluoxetine.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Reduction in the density and expression, but not G-protein coupling, of serotonin receptors (5-HT1A) in 5-HT transporter knock-out mice: gender and brain region differences.

7 January 2021

1 reference

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Molecular mechanisms of membrane receptor desensitization.

7 January 2021

1 reference

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Prevention of the serotonin syndrome in rats by repeated administration of monoamine oxidase inhibitors but not tricyclic antidepressants.

7 January 2021

1 reference

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Pharmacological effects of venlafaxine, a new antidepressant, given repeatedly, on the alpha 1-adrenergic, dopamine and serotonin systems.

7 January 2021

1 reference

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Functional consequences of 5-HT transporter gene disruption on 5-HT(1a) receptor-mediated regulation of dorsal raphe and hippocampal cell activity.

7 January 2021

1 reference

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5-HT1A-receptors mediate stimulation of adenylate cyclase in rat hippocampus.

7 January 2021

1 reference

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Region-dependent effects of flibanserin and buspirone on adenylyl cyclase activity in the human brain

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0024-3205%2802%2902482-7

Isapirone is a partial agonist at 5-hydroxytryptamine 1A (5-HT1A) receptors in the rat hippocampus: electrophysiological evidence.

7 January 2021

1 reference

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Effects of repeated doses of azapirones on rat brain 5-HT1A receptors and plasma corticosterone levels

7 January 2021

1 reference

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Chloroamphetamine did not prevent the effects of chronic antidepressants on 5-hydroxytryptamine inhibition of forskolin-stimulated adenylate cyclase in rat hippocampus.

7 January 2021

1 reference

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Chronic electroconvulsive shock and desimipramine reduce the degree of inhibition by 5-HT and carbachol of forskolin-stimulated adenylate cyclase in rat hippocampal membranes.

7 January 2021

1 reference

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Effects of postmortem delay on serotonin and (+)8-OH-DPAT-mediated inhibition of adenylyl cyclase activity in rat and human brain tissues.

7 January 2021

1 reference

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Chronic fluoxetine treatment selectively uncouples raphe 5-HT(1A) receptors as measured by [(35)S]-GTP gamma S autoradiography

7 January 2021

1 reference

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Serotonin receptor activation reduces calcium current in an acutely dissociated adult central neuron

7 January 2021

1 reference

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Whole-cell recordings of inwardly rectifying K+ currents activated by 5-HT1A receptors on dorsal raphe neurones of the adult rat

7 January 2021

1 reference

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Repeated treatment with 8-OH-DPAT induces tolerance to its ability to produce the 5-HT1A behavioural syndrome, but not to its ability to attenuate haloperidol-induced catalepsy

7 January 2021

1 reference

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Serotonin receptor 1A knockout: an animal model of anxiety-related disorder

7 January 2021

1 reference

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Cell-specific physical and functional coupling of human 5-HT1A receptors to inhibitory G protein alpha-subunits and lack of coupling to Gs alpha

7 January 2021

1 reference

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Somatodendritic localization of 5-HT1A and preterminal axonal localization of 5-HT1B serotonin receptors in adult rat brain

7 January 2021

1 reference

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Agonist-induced internalization of serotonin-1a receptors in the dorsal raphe nucleus (autoreceptors) but not hippocampus (heteroreceptors).

7 January 2021

1 reference

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Modification of serotonin neuron properties in mice lacking 5-HT1A receptors

7 January 2021

1 reference

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Effect of paroxetine and nefazodone on 5-HT 1A receptor sensitivity

7 January 2021

1 reference

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Evidence that G(z)-proteins couple to hypothalamic 5-HT(1A) receptors in vivo.

7 January 2021

1 reference

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Repeated treatment with antidepressants differentially alters 5-HT1A agonist-stimulated [35S]GTP gamma S binding in rat brain regions

7 January 2021

1 reference

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Region-specific changes in 5-HT(1A) receptor-activated G-proteins in rat brain following chronic buspirone

7 January 2021

1 reference

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Chronic MAO A and MAO B inhibition decreases the 5-HT1A receptor-mediated inhibition of forskolin-stimulated adenylate cyclase

7 January 2021

1 reference

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Direct Immunohistochemical Evidence of the Existence of 5-HT1A Autoreceptors on Serotoninergic Neurons in the Midbrain Raphe Nuclei

7 January 2021

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Neuroendocrine pharmacology of serotonergic (5-HT) neurons

7 January 2021

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Quantitative autoradiography of multiple 5-HT1 receptor subtypes in the brain of control or 5,7-dihydroxytryptamine-treated rats

7 January 2021

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Autoradiographic quantification of serotonin1A receptors in rat brain following antidepressant drug treatment

7 January 2021

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Effect of chronic treatments with tandospirone and imipramine on serotonin-mediated behavioral responses and monoamine receptors.

7 January 2021

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The effect of 8-OH-DPAT on temperature in the rat and its modification by chronic antidepressant treatments

7 January 2021

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The effect of chronic administration of antidepressants and electroconvulsive shock on the 5-HT1A receptor mediated hypothermic response induced by 8-OH-DPAT in the rat

7 January 2021

1 reference

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10.1016/S0024-3205(02)02482-7

7 January 2021

Identifiers

DOI

1 reference

31 July 2017

1 reference

PubMed ID

12559389