(Q34208810)

English

Identification of (3R)-7-hydroxy-N-((1S)-1-[[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a novel potent and selective opioid kappa receptor antagonist.

scientific article

Statements

Identification of (3R)-7-hydroxy-N-((1S)-1-[[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a novel potent and selective opioid kappa receptor antagonist. (English)
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James B Thomas
Robert N Atkinson
N Ariane Vinson
Jennifer L Catanzaro
Carin L Perretta
S Wayne Mascarella
Richard B Rothman
Christina M Dersch
Buddy E Cantrell
Dennis M Zimmerman
F Ivy Carroll
3127-3137

Identifiers

 
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