(Q34217246)

31 July 2017

title

Novel chalcone-based fluorescent human histamine h(3) receptor ligands as pharmacological tools (English)

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31 July 2017

Miriam Tomasch

1

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31 July 2017

J Stephan Schwed

series ordinal

2

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31 July 2017

Lilia Weizel

series ordinal

3

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31 July 2017

Holger Stark

series ordinal

4

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31 July 2017

publication date

26 March 2012

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Frontiers in Systems Neuroscience

31 July 2017

published in

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31 July 2017

volume

6

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31 July 2017

page(s)

14

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Histamine receptor subtypes: a century of rational drug design

31 July 2017

cites work

1 reference

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Kojic acid derivatives as histamine H(3) receptor ligands

5 July 2018

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Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties

5 July 2018

1 reference

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Use of the H3 receptor antagonist radioligand [3H]-A-349821 to reveal in vivo receptor occupancy of cognition enhancing H3 receptor antagonists

5 July 2018

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Histamine H3 receptor antagonists go to clinics

5 July 2018

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Fluorescent GPCR ligands as new tools in pharmacology.

5 July 2018

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The alkaloid conessine and analogues as potent histamine H3 receptor antagonists

5 July 2018

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Ether derivatives of 3-piperidinopropan-1-ol as non-imidazole histamine H3 receptor antagonists

5 July 2018

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Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives

5 July 2018

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Role of the histamine system in nefopam-induced antinociception in mice

5 July 2018

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Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

5 July 2018

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Characterization of histamine H3 receptors in mouse brain using the H3 antagonist [125I]iodophenpropit.

5 July 2018

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DAPI: a DNA-specific fluorescent probe

5 July 2018

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Three histamine receptors (H1, H2 and H3) visualized in the brain of human and non-human primates.

5 July 2018

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

5 July 2018

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Detection of low level histamine H3 receptor occupancy by autoradiography

5 July 2018

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Piperidine variations in search for non-imidazole histamine H(3) receptor ligands.

28 October 2018

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Fluorescent benzofuran histamine H(3) receptor antagonists with sub-nanomolar potency.

28 October 2018

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Fluorescent non-imidazole histamine H3 receptor ligands with nanomolar affinities

28 October 2018

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Search for histamine H3 receptor antagonists with combined inhibitory potency at Ntau-methyltransferase: ether derivatives.

28 October 2018

1 reference

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Comparison of effect of selected synthetic chalcone analogues on mitochondrial outer membrane determined by fluorescence spectroscopy.

28 October 2018

1 reference

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Application of ionic liquid halide nucleophilicity for the cleavage of ethers: a green protocol for the regeneration of phenols from ethers

28 October 2018

1 reference

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Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists

28 October 2018

1 reference

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[125I]iodoproxyfan and related compounds: a reversible radioligand and novel classes of antagonists with high affinity and selectivity for the histamine H3 receptor.

28 October 2018

1 reference

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Highly potent fluorescence-tagged nonimidazole histamine H3 receptor ligands

28 October 2018

1 reference

12 December 2020

[125I]iodoproxyfan, a new antagonist to label and visualize cerebral histamine H3 receptors

1 reference

12 December 2020

Histamine H1, H3 and H4 receptors are involved in pruritus

1 reference

12 December 2020

Receptor-specific functional efficacies of alkyl imidazoles as dual histamine H3/H4 receptor ligands

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12 December 2020

Identifiers

DOI

10.3389/FNSYS.2012.00014

1 reference

31 July 2017

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31 July 2017

1 reference