(Q34260033)

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Pharmacological properties of S1RA, a new sigma-1 receptor antagonist that inhibits neuropathic pain and activity-induced spinal sensitization

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scholarly article

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Europe PubMed Central

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1 August 2017

Pharmacological properties of S1RA, a new sigma-1 receptor antagonist that inhibits neuropathic pain and activity-induced spinal sensitization (English)

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Europe PubMed Central

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1 August 2017

neuropathic pain

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author name string

L Romero

1

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1 August 2017

D Zamanillo

2

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1 August 2017

X Nadal

3

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1 August 2017

R Sánchez-Arroyos

4

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1 August 2017

I Rivera-Arconada

5

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1 August 2017

A Dordal

6

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1 August 2017

A Montero

7

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1 August 2017

A Muro

8

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1 August 2017

A Bura

9

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1 August 2017

C Segalés

10

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1 August 2017

M Laloya

11

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1 August 2017

E Hernández

12

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1 August 2017

E Portillo-Salido

13

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1 August 2017

M Escriche

14

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1 August 2017

X Codony

15

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1 August 2017

G Encina

16

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1 August 2017

J Burgueño

17

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1 August 2017

M Merlos

18

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1 August 2017

J M Baeyens

19

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1 August 2017

J Giraldo

20

1 reference

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1 August 2017

J A López-García

21

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1 August 2017

R Maldonado

22

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1 August 2017

C R Plata-Salamán

23

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1 August 2017

J M Vela

24

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1 August 2017

language of work or name

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publication date

1 August 2012

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1 August 2017

British Journal of Pharmacology

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1 August 2017

166

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1 August 2017

8

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PubMed publication ID

1 August 2017

2289-2306

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Europe PubMed Central

PubMed publication ID

1 August 2017

Sigma-1 Receptor Antagonist BD1047 Reduces Allodynia and Spinal ERK Phosphorylation Following Chronic Compression of Dorsal Root Ganglion in Rats

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

The sigma-1 receptor chaperone as an inter-organelle signaling modulator

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Guidelines for reporting experiments involving animals: the ARRIVE guidelines

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Sigma-1 receptor-induced increase in murine spinal NR1 phosphorylation is mediated by the PKCalpha and epsilon, but not the PKCzeta, isoforms.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Sigma 1 receptor modulation of G-protein-coupled receptor signaling: potentiation of opioid transduction independent from receptor binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Sigma-1 receptor chaperones and diseases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Central sensitization: a generator of pain hypersensitivity by central neural plasticity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

The pharmacology of sigma-1 receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Pharmacology and therapeutic potential of sigma(1) receptor ligands

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Antagonism by haloperidol and its metabolites of mechanical hypersensitivity induced by intraplantar capsaicin in mice: role of sigma-1 receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Intrathecal injection of the sigma(1) receptor antagonist BD1047 blocks both mechanical allodynia and increases in spinal NR1 expression during the induction phase of rodent neuropathic pain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Activation of the spinal sigma-1 receptor enhances NMDA-induced pain via PKC- and PKA-dependent phosphorylation of the NR1 subunit in mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Irreversible blockade of sigma-1 receptors by haloperidol and its metabolites in guinea pig brain and SH-SY5Y human neuroblastoma cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

The sigma-1 receptor modulates NMDA receptor synaptic transmission and plasticity via SK channels in rat hippocampus.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Intrathecal treatment with sigma1 receptor antagonists reduces formalin-induced phosphorylation of NMDA receptor subunit 1 and the second phase of formalin test in mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Understanding the molecular mechanism of sigma-1 receptors: towards a hypothesis that sigma-1 receptors are intracellular amplifiers for signal transduction

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Immunocytochemical localization of the sigma(1) receptor in the adult rat central nervous system

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Wind-up of spinal cord neurones and pain sensation: much ado about something?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Operational models of pharmacological agonism.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

N-methyl-D-aspartate-induced neuronal activation is selectively modulated by sigma receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

The induction and maintenance of central sensitization is dependent on N -methyl-d-aspartic acid receptor activation; implications for the treatment of post-injury pain hypersensitivity states

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Characterization of the binding of [3H](+)-pentazocine to sigma recognition sites in guinea pig brain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

6 July 2018

Antinociceptive effects of haloperidol and its metabolites in the formalin test in mice

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Neurosteroid dehydroepiandrosterone sulphate inhibits persistent sodium currents in rat medial prefrontal cortex via activation of sigma-1 receptors

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Phenytoin differentially modulates the affinity of agonist and antagonist ligands for sigma 1 receptors of guinea pig brain

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Sigma-1 receptors are essential for capsaicin-induced mechanical hypersensitivity: studies with selective sigma-1 ligands and sigma-1 knockout mice.

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

sigma-1 receptor modulation of acid-sensing ion channel a (ASIC1a) and ASIC1a-induced Ca2+ influx in rat cortical neurons

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Ionotropic and metabotropic receptors, protein kinase A, protein kinase C, and Src contribute to C-fiber-induced ERK activation and cAMP response element-binding protein phosphorylation in dorsal horn neurons, leading to central sensitization.

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Sigma1 receptor modulation of opioid analgesia in the mouse

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Spinal NMDA receptor phosphorylation correlates with the presence of neuropathic signs following peripheral nerve injury in the rat.

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.01942.X

21 January 2018

Sigma receptors inhibit high-voltage-activated calcium channels in rat sympathetic and parasympathetic neurons

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

28 October 2018

Potentiation of neuronal NMDA response induced by dehydroepiandrosterone and its suppression by progesterone: effects mediated via sigma receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

28 October 2018

Selective antagonism of opioid analgesia by a sigma system

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

28 October 2018

Modulation by sigma ligands of intracellular free Ca++ mobilization by N-methyl-D-aspartate in primary culture of rat frontal cortical neurons

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3448894

28 October 2018

Formalin-induced pain is reduced in sigma(1) receptor knockout mice

1 reference

https://pubmed.ncbi.nlm.nih.gov/22404321

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Sigma-1 receptors regulate activity-induced spinal sensitization and neuropathic pain after peripheral nerve injury

1 reference

https://pubmed.ncbi.nlm.nih.gov/22404321

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Central sensitization needs sigma receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/22404321

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence for a role of the NMDA receptor in the frequency dependent potentiation of deep rat dorsal horn nociceptive neurones following C fibre stimulation

1 reference

https://pubmed.ncbi.nlm.nih.gov/22404321

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Ca(2+) signaling via sigma(1)-receptors: novel regulatory mechanism affecting intracellular Ca(2+) concentration

1 reference

https://pubmed.ncbi.nlm.nih.gov/22404321

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.2012.01942.X

1 reference

Europe PubMed Central

PubMed publication ID

1 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

1 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

1 August 2017

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