(Q34340266)

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The behavioral profile of the potent and selective mGlu5 receptor antagonist 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine (MTEP) in rodent models of anxiety

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Europe PubMed Central

1 August 2017

The behavioral profile of the potent and selective mGlu5 receptor antagonist 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine (MTEP) in rodent models of anxiety (English)

1 reference

Europe PubMed Central

1 August 2017

author name string

Chris S Busse

1

1 reference

Europe PubMed Central

1 August 2017

Jesse Brodkin

2

1 reference

Europe PubMed Central

1 August 2017

David Tattersall

3

1 reference

Europe PubMed Central

1 August 2017

Jeffery J Anderson

4

1 reference

Europe PubMed Central

1 August 2017

Noelle Warren

5

1 reference

Europe PubMed Central

1 August 2017

Lida Tehrani

6

1 reference

Europe PubMed Central

1 August 2017

Linda J Bristow

7

1 reference

Europe PubMed Central

1 August 2017

Mark A Varney

8

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Europe PubMed Central

1 August 2017

Nicholas D P Cosford

9

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1 August 2017

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1 November 2004

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1 August 2017

Neuropsychopharmacology

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1 August 2017

29

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1 August 2017

11

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Europe PubMed Central

1 August 2017

1971-1979

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Europe PubMed Central

1 August 2017

https://scigraph.springernature.com/pub.10.1038/sj.npp.1300540

0 references

In vivo receptor occupancy of mGlu5 receptor antagonists using the novel radioligand [3H]3-methoxy-5-(pyridin-2-ylethynyl)pyridine).

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

[3H]Methoxymethyl-3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine binding to metabotropic glutamate receptor subtype 5 in rodent brain: in vitro and in vivo characterization

1 reference

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21 January 2018

The psychobiology of anxiolytic drug. Part 2: Pharmacological treatments of anxiety

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

The metabotropic glutamate receptor (mGluR1 alpha) is concentrated at perisynaptic membrane of neuronal subpopulations as detected by immunogold reaction.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Reduced stress-induced hyperthermia in mGluR5 knockout mice

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Anxiolytic-like activity of the mGluR5 antagonist MPEP: a comparison with diazepam and buspirone

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Alnespirone and buspirone have anxiolytic-like effects in a conflict procedure in rats by stimulating 5-HT(1A) receptors.

1 reference

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21 January 2018

Pharmacology and functions of metabotropic glutamate receptors

1 reference

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21 January 2018

[3H]-methoxymethyl-MTEP and [3H]-methoxy-PEPy: potent and selective radioligands for the metabotropic glutamate subtype 5 (mGlu5) receptor

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]-pyridine: a potent and highly selective metabotropic glutamate subtype 5 receptor antagonist with anxiolytic activity

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Diazepam and flurazepam: Effects on conditioned fear as measured with the potentiated startle paradigm

1 reference

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21 January 2018

Fear-potentiated startle: a neural and pharmacological analysis

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Economic costs of anxiety disorders.

1 reference

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21 January 2018

2-Methyl-6-(phenylethynyl)-pyridine (MPEP), a potent, selective and systemically active mGlu5 receptor antagonist

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Anticonflict effect of alpidem as compared with the benzodiazepine alprazolam in rats.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Activation of a metabotropic glutamate receptor and protein kinase C reduce the extent of inactivation of the K+ channel Kv1.1/Kvbeta1.1 via dephosphorylation of Kv1.1.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

An overview of generalized anxiety disorder: disease state--appropriate therapy

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Recent developments in the psychopharmacology of anxiety disorders

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Drug interactions with ethanol. Effects on body temperature and motor impairment.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Positive allosteric modulation of the human metabotropic glutamate receptor 4 (hmGluR4) by SIB-1893 and MPEP

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

The metabotropic glutamate receptors, mGluR2 and mGluR3, show unique postsynaptic, presynaptic and glial localizations

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Multiple MPEP administrations evoke anxiolytic- and antidepressant-like effects in rats

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

The metabotropic glutamate receptor antagonist 2-methyl-6-(phenylethynyl)-pyridine (MPEP) blocks fear conditioning in rats

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Use of benzodiazepines in anxiety disorders

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Immunohistochemical localization of a metabotropic glutamate receptor, mGluR5, in the rat brain

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Pharmacological and endocrinological characterisation of stress-induced hyperthermia in singly housed mice using classical and candidate anxiolytics (LY314582, MPEP and NKP608).

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Presynaptic calcium current modulation by a metabotropic glutamate receptor.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Potential anxiolytic- and antidepressant-like effects of MPEP, a potent, selective and systemically active mGlu5 receptor antagonist

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

L-Arginine abolishes the anxiolytic-like effect of diazepam in the elevated plus-maze test in rats.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

The pharmacological properties of Y-23684, a benzodiazepine receptor partial agonist

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

21 January 2018

Chronic but not acute treatment with a metabotropic glutamate 5 receptor antagonist reverses the akinetic deficits in a rat model of parkinsonism.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

7 January 2021

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Efficacy, safety, and tolerability of venlafaxine extended release and buspirone in outpatients with generalized anxiety disorder

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

7 January 2021

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Heterologous expression of metabotropic glutamate receptors in adult rat sympathetic neurons: subtype-specific coupling to ion channels

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

7 January 2021

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Rat group I metabotropic glutamate receptors inhibit neuronal Ca2+ channels via multiple signal transduction pathways in HEK 293 cells.

1 reference

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7 January 2021

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Long-term buspirone therapy for chronic anxiety: a multicenter international study to determine safety.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

7 January 2021

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Distribution of metabotropic glutamate receptor mGluR5 immunoreactivity in rat brain

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1300540

7 January 2021

based on heuristic

inferred from DOI database lookup

Differential presynaptic localization of metabotropic glutamate receptor subtypes in the rat hippocampus

1 reference

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7 January 2021

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Metabotropic glutamate receptor enhancement of spontaneous IPSCs in neocortical interneurons.

1 reference

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10.1038/SJ.NPP.1300540

1 reference

Europe PubMed Central

1 August 2017

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https://api.fatcat.wiki/v0/release/nshhd4utvfairkg55au6nvl4xe

24 November 2022

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1 reference

Europe PubMed Central

1 August 2017

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