(Q34410429)

2 August 2017

1 reference

title

Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications (English)

1 reference

2 August 2017

0 references

Ruben S Vardanyan

1

1 reference

PubMed ID

24635521

2 August 2017

Victor J Hruby

series ordinal

2

1 reference

PubMed ID

24635521

2 August 2017

language of work or name

English

0 references

publication date

1 March 2014

1 reference

Future Medicinal Chemistry

2 August 2017

1 reference

2 August 2017

6

1 reference

2 August 2017

385-412

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2 August 2017

4

1 reference

Synthesis and biological evaluation of new opioid agonist and neurokinin-1 antagonist bivalent ligands

2 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Stop the pain: fentanyl is a viable alternative to morphine

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl for breakthrough pain: a systematic review

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl nasal spray for the treatment of cancer pain

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Design strategies for bivalent ligands targeting GPCRs

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Opioid bifunctional ligands from morphine and the opioid pharmacophore Dmt-Tic

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Development of potent μ and δ opioid agonists with high lipophilicity

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

"Carba"-analogues of fentanyl are opioid receptor agonists

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

The development of new analgesics over the past 50 years: a lack of real breakthrough drugs

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Formulations of fentanyl for the management of pain

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Transdermal fentanyl: pharmacology and toxicology

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl analogs: structure-activity-relationship study

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthesis and investigations of double-pharmacophore ligands for treatment of chronic and neuropathic pain

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Dissociation of the opioid receptor mechanisms that control mechanical and heat pain

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Simultaneous targeting of multiple opioid receptors: a strategy to improve side-effect profile

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Development of mu/delta opioid ligands: enkephalin analogues containing 4-anilidopiperidine moiety

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Bi- or multifunctional opioid peptide drugs

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Design of multivalent ligand targeting G-protein-coupled receptors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

A tribute to Dr. Paul A. J. Janssen: entrepreneur extraordinaire, innovative scientist, and significant contributor to anesthesiology

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl buccal tablet: rapid relief from breakthrough pain

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Development of novel enkephalin analogues that have enhanced opioid activities at both mu and delta opioid receptors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Receptor heterodimerization leads to a switch in signaling: beta-arrestin2-mediated ERK activation by mu-delta opioid receptor heterodimers

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Understanding the structural requirements of 4-anilidopiperidine analogues for biological activities at mu and delta opioid receptors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

New paradigms and tools in drug design for pain and addiction

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthesis and evaluation of 3-aminopropionyl substituted fentanyl analogues for opioid activity

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Remifentanil : a review of its analgesic and sedative use in the intensive care unit

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Designed multiple ligands. An emerging drug discovery paradigm

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Remifentanil: a review of its use during the induction and maintenance of general anaesthesia

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl for acute pain management

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

A personal perspective on Dr. Paul Janssen

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Remifentanil update: clinical science and utility

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

A role for heterodimerization of mu and delta opiate receptors in enhancing morphine analgesia

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

The inhibitory effect of fentanyl and other morphine-like analgesics on the warm water induced tail withdrawl reflex in rats

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl and its analogue N-(1-phenylpyrazol-3-yl)-N-[1-(2-phenylethyl)-4-piperidyl]propanamide: 1H- and 13C-NMR spectroscopy, X-ray crystallography, and theoretical calculations

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Guanidinium and aminoimidazolinium derivatives of N-(4-piperidyl)propanamides as potential ligands for mu opioid and I2-imidazoline receptors: synthesis and pharmacological screening.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Molecular docking reveals a novel binding site model for fentanyl at the mu-opioid receptor.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

An overview of remifentanil

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Interaction models of 3-methylfentanyl derivatives with mu opioid receptors.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Transdermal fentanyl. A review of its pharmacological properties and therapeutic efficacy in pain control

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Remifentanil: a novel, short-acting, mu-opioid

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Antinociceptive profile of biphalin, a dimeric enkephalin analog

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Enantiomers of diastereomeric cis-N-[1-(2-hydroxy-2-phenylethyl)- 3-methyl-4-piperidyl]-N-phenylpropanamides: synthesis, X-ray analysis, and biological activities

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Stereoisomers of N-[1-hydroxy-(2-phenylethyl)-3-methyl-4-piperidyl]- N-phenylpropanamide: synthesis, stereochemistry, analgesic activity, and opioid receptor binding characteristics

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl: a review for clinical and analytical toxicologists.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

4-Anilidopiperidine analgesics. 3. 1-Substituted 4-(propananilido)perhydroazepines as ring-expanded analogues

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Biotransformation of fentanyl. II. Acute drug interactions in rats and men (author's transl)

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Functional opiate receptors in the guinea-pig ileum: their differentiation by means of selective tolerance development

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Opiate receptor interaction of compounds derived from or structurally related to fentanyl

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Studies on synthesis and relationship between analgesic activity and receptor affinity for 3-methyl fentanyl derivatives

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthesis and stereochemistry of 7-phenyl-2-propionanilidobenzo[a]quinolizidine derivatives. Structural probes of fentanyl analgesics

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Clinical pharmacokinetics of fentanyl and its newer derivatives.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

The binding spectrum of narcotic analgesic drugs with different agonist and antagonist properties

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthetic analgesics. Synthesis and pharmacology of the diastereoisomers of N-(3-methyl-1-(2-phenylethyl)-4-piperidyl)-N-phenylpropanamide and N-(3-methyl-1-(1-methyl-2-phenylethyl)-4-piperidyl)-N-phenylpropanamide

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Analgesically active basic anilides: stereospecificity and structure of the basic group

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

On conformation analysis, molecular graphics, fentanyl and its derivatives

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Probes for narcotic receptor mediated phenomena. 12. cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for delta opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivity

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Structure-activity studies of fentanyl.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Conformation-activity relationships of opiate analgesics

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Relative analgesic potency of epidural fentanyl, alfentanil, and morphine in treatment of postoperative pain

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthetic 1,4-disubstituted-1,4-dihydro-5H-tetrazol-5-one derivatives of fentanyl: alfentanil (R 39209), a potent, extremely short-acting narcotic analgesic.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Studies of the pharmacology and pathology of intrathecally administered 4-anilinopiperidine analogues and morphine in the rat and cat.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthesis and pharmacological evaluation of 4,4-disubstituted piperidines.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

4-Phenyl- and 4-heteroaryl-4-anilidopiperidines. A novel class of analgesic and anesthetic agents

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

New 4-(heteroanilido)piperidines, structurally related to the pure opioid agonist fentanyl, with agonist and/or antagonist properties

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Modulation of mu-mediated antinociception by delta agonists in the mouse: selective potentiation of morphine and normorphine by [D-Pen2,D-Pen5]enkephalin

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Design, synthesis, and pharmacological evaluation of ultrashort- to long-acting opioid analgetics

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Evolution of the 4-anilidopiperidine class of opioid analgesics

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

New 1-(heterocyclylalkyl)-4-(propionanilido)-4-piperidinyl methyl ester and methylene methyl ether analgesics

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Development of a conformational search strategy for flexible ligands: a study of the potent mu-selective opioid analgesic fentanyl

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

(+)-Cis-3-methylfentanyl and its analogs bind pseudoirreversibly to the mu opioid binding site: Evidence for pseudoallosteric modulation

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

The history and development of the fentanyl series

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Fentanyl: clinical use as postoperative analgesic--epidural/intrathecal route

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Pharmacological profiles of fentanyl analogs at mu, delta and kappa opiate receptors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Modulation of mu-mediated antinociception in the mouse involves opioid delta-2 receptors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Molecular determinants of mu receptor recognition for the fentanyl class of compounds

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthesis of some conformationally restricted analogues of fentanyl.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

4-Anilidopiperidine analgesics. 2. A study of the conformational aspects of the analgesic activity of the 4-anilidopiperidines utilizing isomeric N-substituted 3-(propananilido)nortropane analogs

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Sufentanil, a very potent and extremely safe intravenous morphine-like compound in mice, rats and dogs

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

N-4-Substituted 1-(2-arylethyl)-4-piperidinyl-N-phenylpropanamides, a novel series of extremely potent analgesics with unusually high safety margin

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthetic analgesics: N-(1-[2-arylethyl]-4-substituted 4-piperidinyl) N-arylalkanamides

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Stimulating the development of mechanism-based, individualized pain therapies

6 July 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

A review of the use of fentanyl analgesia in the management of acute pain in adults

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

A STUDY OF SOME OF THE PHARMACOLOGIC ACTIONS OF FENTANYL CITRATE.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Relative analgesic potency of fentanyl and sufentanil during intermediate-term infusions in patients after long-term opioid treatment for chronic pain

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Synthesis and evaluation of 1- and 2-substituted fentanyl analogues for opioid activity

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Interactions of some 4-anilinopiperidines and 4-phenylpiperidines with the mu, delta- and kappa-binding sites

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Clinical actions of fentanyl and buprenorphine. The significance of receptor binding.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

The synthesis and preliminary pharmacological evaluation of 4-methyl fentanyl

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Alfentanil (R 39 209) ? a particularly short-acting intravenous narcotic analgesic in rats

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

A facile method for preparation of [(2)h(3)]-sufentanil and its metabolites

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Syntheses, biological evaluation, and molecular modeling of 18F-labeled 4-anilidopiperidines as mu-opioid receptor imaging agents

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

21 January 2018

Remifentanil. An update

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Long-acting fentanyl analogues: synthesis and pharmacology of N-(1-phenylpyrazolyl)-N-(1-phenylalkyl-4-piperidyl)propanamides.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Synthesis and opioid activity of new fentanyl analogs.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Analgesic activity and pharmacological characterization of N-[1-phenylpyrazol-3-yl]-N-[1-(2-phenethyl)-4-piperidyl] propenamide, a new opioid agonist acting peripherally

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Fentanyl derivatives bearing aliphatic alkaneguanidinium moieties: a new series of hybrid molecules with significant binding affinity for mu-opioid receptors and I2-imidazoline binding sites.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Antinociceptive activity of the novel fentanyl analogue iso-carfentanil in rats.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Cardiovascular activity of some substituted 2-aminobenzoquinolizines.

21 January 2018

1 reference

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Irreversible Ligands with High Selectivity Toward δ and μ Opiate Receptors

21 January 2018

1 reference

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Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for .mu. or .delta. opiate receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Analgesic activity and selectivity of isothiocyanate derivatives of fentanyl analogs for opioid receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Synthesis and pharmacological studies of new hybrid derivatives of fentanyl active at the mu-opioid receptor and I2-imidazoline binding sites

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Synthesis and Crystallographic Study of N'-(1-benzylpiperidin-4-yl)acetohydrazide

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

The opioid mu agonist/delta antagonist DIPP-NH(2)[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Steric interactions and the activity of fentanyl analogs at the mu-opioid receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

A new consistent model explaining structure (conformation)-activity relationships of opiates with mu-selectivity.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

[Biotransformation of fentanyl. III. Effect of chronic drug exposure on the distribution, metabolism and excretion in the rat]

27 October 2018

1 reference

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Synthesis, and structural, conformational and pharmacological studies of new fentanyl derivatives of the norgranatane system

27 October 2018

1 reference

https://api.crossref.org/works/10.4155%2FFMC.13.215

Clinical pharmacology of fentanyl buccal tablet for the treatment of breakthrough pain

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4137794

Synthesis of 1-(piperidinyl-4)-indolinones-(2) and-3,4-dihydrocarbostyriles (author's transl)

9 December 2018

1 reference

12 December 2020

1 reference

12 December 2020

1 reference

12 December 2020

Structure-activity relations in analgesics based on 4-anilinopiperidine

1 reference

12 December 2020

Compounds Affecting the Central Nervous System. II. Substituted 1,2,3,4-Tetrahydropyrido[4,3-b]indoles

1 reference

12 December 2020

Modulation of mu-mediated antinociception by delta agonists: characterization with antagonists

1 reference

12 December 2020

SYNTHETIC ANALGESICS. IV. SYNTHESIS OF ENANTIOMERS OF BASIC ANILIDES CONTAINING THE PHENALKYL MOIETY

1 reference

12 December 2020

1 reference

12 December 2020

Synthesis and analgetic activity of some 1-substituted 3-pyrrolidinylanilides and dihydrobenzoxazinones

1 reference

12 December 2020

Evaluation of 2-azabicyclo[2.2..2]octane analogs of 4-anilidopiperidine analgesics

1 reference

12 December 2020

4-Anilidopiperidine Analgesics I: Synthesis and Analgesic Activity of Certain Ring-Methylated 1-Substituted 4-Propananilidopiperidines

1 reference

12 December 2020

Identifiers

DOI

10.4155/FMC.13.215

1 reference

2 August 2017

1 reference

2 August 2017

1 reference

PubMed ID

24635521