(Q34498106)

English

Straightforward protocol for the efficient synthesis of varied N(1)-acylated (aza)indole 2-/3-alkanoic acids and esters: optimization and scale-up

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

Straightforward protocol for the efficient synthesis of varied N(1)-acylated (aza)indole 2-/3-alkanoic acids and esters: optimization and scale-up (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

author name string

Andy J Liedtke

1

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

Kwangho Kim

2

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

Donald F Stec

3

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

Gary A Sulikowski

4

1 reference

Europe PubMed Central

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2 August 2017

Lawrence J Marnett

5

1 reference

Europe PubMed Central

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2 August 2017

publication date

1 December 2012

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Europe PubMed Central

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2 August 2017

1 reference

Europe PubMed Central

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2 August 2017

68

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Europe PubMed Central

PubMed publication ID

2 August 2017

48

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

10049-10058

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

Development of potent and selective inhibitors of aldo-keto reductase 1C3 (type 5 17β-hydroxysteroid dehydrogenase) based on N-phenyl-aminobenzoates and their structure-activity relationships

1 reference

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CRTH2 and D-type prostanoid receptor antagonists as novel therapeutic agents for inflammatory diseases

1 reference

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Anti-inflammatory drugs in the 21st century

1 reference

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Structural and functional basis of cyclooxygenase inhibition

1 reference

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Total synthesis of (-)- and ent-(+)-vindoline

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Indolyl esters and amides related to indomethacin are selective COX-2 inhibitors

1 reference

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Development of a prostaglandin D2 receptor antagonist: discovery of a new chemical lead

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Structural determinants of arylacetic acid nonsteroidal anti-inflammatory drugs necessary for binding and activation of the prostaglandin D2 receptor CRTH2.

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7-Azaindole-3-acetic acid derivatives: potent and selective CRTh2 receptor antagonists.

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A microwave-assisted facile regioselective Fischer indole synthesis and antitubercular evaluation of novel 2-aryl-3,4-dihydro-2H-thieno[3,2-b]indoles.

1 reference

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27 October 2018

Single-flask synthesis of N-acylated indoles by catalytic dehydrogenative coupling with primary alcohols

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3509943

27 October 2018

Synthesis of C3-substituted 4-azaindoles: an easy access to 4-azamelatonin and protected 4-azatryptophan

1 reference

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Structure-based design, synthesis, and biological evaluation of indomethacin derivatives as cyclooxygenase-2 inhibiting nitric oxide donors

1 reference

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Aminopiperidine indazoles as orally efficacious melanin concentrating hormone receptor-1 antagonists

1 reference

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27 October 2018

Molecular basis of the time-dependent inhibition of cyclooxygenases by indomethacin

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3509943

27 October 2018

Discovery of new chemical leads for prostaglandin D2 receptor antagonists

1 reference

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27 October 2018

NSAID-induced gastric damage in rats: Requirement for inhibition of both cyclooxygenase 1 and 2

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Synthesis of indomethacin analogues for evaluation as modulators of MRP activity

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A general synthesis of substituted indoles from cyclic enol ethers and enol lactones

1 reference

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A mild and selective method for the hydrolysis of esters with trimethyltin hydroxide

1 reference

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A new entry to the synthesis of 2,3-disubstituted indoles

1 reference

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Desmethyl derivatives of indomethacin and sulindac as probes for cyclooxygenase-dependent biology

1 reference

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An indomethacin analogue, N-(4-chlorobenzoyl)-melatonin, is a selective inhibitor of aldo-keto reductase 1C3 (type 2 3alpha-HSD, type 5 17beta-HSD, and prostaglandin F synthase), a potential target for the treatment of hormone dependent and hormone

1 reference

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Atropisomerism observed in indometacin derivatives

1 reference

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NSAIDs: Old Drugs Reveal New Anticancer Targets.

1 reference

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1-acyl-indoles. II. A new syntheses of 1-(p-chlorobenzoyl)-5-methyoxy-3-indolyacetic acid and its polymorphism

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.TET.2012.08.044

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

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