(Q34560149)

3 August 2017

Zolantidine (SK&F 95282) is a potent selective brain-penetrating histamine H2-receptor antagonist (English)

1 reference

3 August 2017

Calcutt CR

1

1 reference

3 August 2017

Ganellin CR

2

1 reference

3 August 2017

Griffiths R

3

1 reference

3 August 2017

Leigh BK

4

1 reference

3 August 2017

Maguire JP

5

1 reference

3 August 2017

Mitchell RC

6

1 reference

3 August 2017

Mylek ME

7

1 reference

3 August 2017

Parsons ME

8

1 reference

3 August 2017

Smith IR

9

1 reference

3 August 2017

Young RC

10

1 reference

3 August 2017

language of work or name

English

0 references

publication date

1 January 1988

1 reference

British Journal of Pharmacology

3 August 2017

1 reference

3 August 2017

93

1 reference

3 August 2017

1

1 reference

3 August 2017

69-78

1 reference

Some quantitative uses of drug antagonists

3 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Inhibition of histamine synthesis in brain by alpha-fluoromethylhistidine, a new irreversible inhibitor: in vitro and in vivo studies

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Correlation between histamine-induced neuronal excitability and activation of adenylate cyclase in the guinea pig hippocampus

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Characteristics of GABAB receptor binding sites on rat whole brain synaptic membranes

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Characterization of histamine receptors in cat cerebral arteries in vitro and in situ.

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Response of the histamine h2-receptor in brain to antidepressant drugs

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Histamine as a Neurotransmitter in Mammalian Brain: Neurochemical Evidence

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Pharmacological specificity of brain histamine H2-receptors differs in intact cells and cell-free preparations.

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Turnover of histamine in rat brain and its decrease under barbiturate anesthesia.

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

A highly sensitive adenylate cyclase assay

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Definition and antagonism of histamine H 2 -receptors

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Pharmacological studies with SK&F 93944 (temelastine), a novel histamine H1-receptor antagonist with negligible ability to penetrate the central nervous system

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Biochemical indentification of the mammalian muscarinic cholinergic receptor

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

The binding of [3H]mepyramine to histamine H1 receptors in guinea-pig brain

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Use of ADTN to define specific 3H-spirerone binding to receptors in brain

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Brain histamine receptors as targets for antidepressant drugs

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Regional distribution of mast cells containing histamine, dopamine, or 5-hydroxytryptamine in the mammalian brain

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Histamine H1 receptors identified in mammalian brain membranes with [3H]mepyramine

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Multiple receptors for dopamine

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Pharmacological properties of histamine-sensitive adenylate cyclase from mammalian brain

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

The dilating effect of histamine on pial arteries of cats and its mediation by H2 receptors

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Pharmacological characterization of histamine receptors mediating the stimulation of cyclic AMP accumulation in slices from guinea-pig hippocampus

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Antagonism of histamine-activated adenylate cyclase in brain by D-lysergic acid diethylamide

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Tricyclic antidepressant drugs block histamine H2 receptor in brain

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

The interaction of histamine and guanylnucleotides with cardiac adenylate cyclase and its relationship to cardiac contractility

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Histamine-sensitive adenylate cyclase in mammalian brain

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

3Hrauwolscine and 3Hyohimbine binding to rat cerebral and human platelet membranes: Possible heterogeneity of α2-adrenoceptors

7 July 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Histamine-induced inositol phospholipid breakdown mirrors H1-receptor density in brain.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Sidechain-modified histamine analogues as substrates for histamine N-methyltransferase.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Histamine turnover in rat brain.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Specific binding of 3H-tiotidine to histamine H2 receptors in guinea pig cerebral cortex.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Mast cells in rat thalamus: nuclear localization, sex difference and left-right asymmetry.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Binding characteristics of 3H-prazosin to rat brain α-adrenergic receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Cerebral Histamine: Indications for Neuronal and Vascular Regulation

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Effect of alpha-fluoromethylhistidine on the histamine content of the brain of W/Wv mice devoid of mast cells: turnover of brain histamine.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Histamine turnover in the brain of different mammalian species: implications for neuronal histamine half-life

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Histamine H2-binding studies in the guinea-pig brain.

21 January 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Isolated brain microvessels: preparation, morphology, histamine and catecholamine contents.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1853786

Histamine and noradrenaline decrease calcium-activated potassium conductance in hippocampal pyramidal cells

27 October 2018

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1988.TB11406.X

Studies on a capillary-rich fraction isolated from brain: histaminic components and characterization of the histamine receptors linked to adenylate cyclase

21 January 2018

1 reference

12 December 2020

3H-Glycogen hydrolysis elicited by histamine in mouse brain slices: selective involvement of H1 receptors

1 reference

12 December 2020

Regulation of serotonin2 (5-HT2) receptors labeled with [3H]spiroperidol by chronic treatment with the antidepressant amitriptyline

1 reference

12 December 2020

l-Histidine Decarboxylase in the Human Brain: Properties and Localization

1 reference

12 December 2020

Comparison of the pharmacological characteristics of 5 HT1 and 5 HT2 binding sites with those of serotonin autoreceptors which modulate serotonin release

1 reference

12 December 2020

Histamine turnover in regions of rat brain

1 reference

12 December 2020

Normal levels of histamine and tele-methylhistamine in mast cell-deficient mouse brain

1 reference

12 December 2020

Distribution of the histaminergic neuron system in the central nervous system of rats; a fluorescent immunohistochemical analysis with histidine decarboxylase as a marker

1 reference

12 December 2020

10.1111/J.1476-5381.1988.TB11406.X

Identifiers

DOI

1 reference

3 August 2017

1 reference

3 August 2017

1 reference