(Q34717142)

4 August 2017

title

Antiinflammatory glucocorticoid receptor ligand with reduced side effects exhibits an altered protein-protein interaction profile (English)

1 reference

protein-protein interaction

4 August 2017

main subject

1 reference

Jeffrey N Miner

1

1 reference

4 August 2017

Bob Ardecky

2

1 reference

4 August 2017

Khalid Benbatoul

3

1 reference

4 August 2017

Kimberly Griffiths

4

1 reference

4 August 2017

Christopher J Larson

5

1 reference

4 August 2017

Dale E Mais

6

1 reference

4 August 2017

Keith Marschke

7

1 reference

4 August 2017

Jon Rosen

8

1 reference

4 August 2017

Eric Vajda

9

1 reference

4 August 2017

Lin Zhi

10

1 reference

4 August 2017

Andres Negro-Vilar

11

1 reference

4 August 2017

language of work or name

English

0 references

publication date

21 November 2007

1 reference

Proceedings of the National Academy of Sciences of the United States of America

4 August 2017

published in

1 reference

4 August 2017

volume

104

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4 August 2017

issue

49

1 reference

4 August 2017

page(s)

19244-19249

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Nuclear compartmentalization of N-CoR and its interactions with steroid receptors

4 August 2017

cites work

1 reference

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Dissociated nonsteroidal glucocorticoid receptor modulators; discovery of the agonist trigger in a tetrahydronaphthalene-benzoxazine series

7 July 2018

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Conformational changes of the glucocorticoid receptor ligand binding domain induced by ligand and cofactor binding, and the location of cofactor binding sites determined by hydrogen/deuterium exchange mass spectrometry

7 July 2018

1 reference

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Novel arylpyrazole compounds selectively modulate glucocorticoid receptor regulatory activity

7 July 2018

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New and improved glucocorticoid receptor ligands

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

A fully dissociated compound of plant origin for inflammatory gene repression

7 July 2018

1 reference

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The nitrosterols--a step forward from the steroid anti-inflammatory drugs?

7 July 2018

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Dissociated glucocorticoid receptor ligands: compounds with an improved therapeutic index.

7 July 2018

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Repression of interleukin-5 transcription by the glucocorticoid receptor targets GATA3 signaling and involves histone deacetylase recruitment

7 July 2018

1 reference

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The search for safer glucocorticoid receptor ligands

7 July 2018

1 reference

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Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

7 July 2018

1 reference

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Corepressor binding to progesterone and glucocorticoid receptors involves the activation function-1 domain and is inhibited by molybdate

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Novel N-arylpyrazolo[3,2-c]-based ligands for the glucocorticoid receptor: receptor binding and in vivo activity

7 July 2018

1 reference

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Selective LXXLL peptides antagonize transcriptional activation by the retinoid-related orphan receptor RORgamma

7 July 2018

1 reference

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Dissociation of transactivation from transrepression by a selective glucocorticoid receptor agonist leads to separation of therapeutic effects from side effects

7 July 2018

1 reference

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Pharmacological regulation of hepatic glucose production.

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

A novel antiinflammatory maintains glucocorticoid efficacy with reduced side effects

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Alternate surfaces of transcriptional coregulator GRIP1 function in different glucocorticoid receptor activation and repression contexts

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

trans-Activation and repression properties of the novel nonsteroid glucocorticoid receptor ligand 2,5-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5-(1-methylcyclohexen-3-y1)-1H-[1]benzopyrano[3,4-f]quinoline (A276575) and its four stereoisomers

7 July 2018

1 reference

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Potent antiarthritic properties of a glucocorticoid derivative, NCX-1015, in an experimental model of arthritis

7 July 2018

1 reference

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Synthesis and characterization of non-steroidal ligands for the glucocorticoid receptor: selective quinoline derivatives with prednisolone-equivalent functional activity

7 July 2018

1 reference

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Cross-talk between glucocorticoid receptor and AP-1.

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

The TRAP/SMCC/Mediator complex and thyroid hormone receptor function

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Nuclear receptors: coactivators, corepressors and chromatin remodeling in the control of transcription

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Dissection of the LXXLL nuclear receptor-coactivator interaction motif using combinatorial peptide libraries: discovery of peptide antagonists of estrogen receptors alpha and beta

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Collagen-induced arthritis in mice: an animal model to study the pathogenesis of rheumatoid arthritis

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Structure and specificity of nuclear receptor-coactivator interactions

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

DNA binding of the glucocorticoid receptor is not essential for survival

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Synthetic glucocorticoids that dissociate transactivation and AP-1 transrepression exhibit antiinflammatory activity in vivo

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Differential interactions of Id proteins with basic-helix-loop-helix transcription factors

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Formation, mineralization, and resorption of bone in vitamin D—deficient rats

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Androgen treatment prevents loss of cancellous bone in the orchidectomized rat

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2148275

Advances in male contraception

7 July 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0705517104

5-Benzylidene 1,2-dihydrochromeno[3,4-f]quinolines, a novel class of nonsteroidal human progesterone receptor agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0705517104

Evaluation of ligand-dependent changes in AR structure using peptide probes

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0705517104

Steroid receptor coactivator (SRC)-1 and SRC-3 differentially modulate tissue-specific activation functions of the progesterone receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0705517104

Novel ketal ligands for the glucocorticoid receptor: in vitro and in vivo activity

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0705517104

Differential effects of gonadal function on bone histomorphometry in male and female rats

21 January 2018

1 reference

12 December 2020

Effect of RU 486 on the atrophogenic and antiinflammatory effects of glucocorticoids in skin

1 reference

12 December 2020

Intermolecular NH2-/carboxyl-terminal interactions in androgen receptor dimerization revealed by mutations that cause androgen insensitivity

1 reference

12 December 2020

Rodent models of arthritis: relevance for human disease

1 reference

12 December 2020

Design of potent and selective 2-aminobenzimidazole-based p38alpha MAP kinase inhibitors with excellent in vivo efficacy

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.0705517104

1 reference

4 August 2017

0 references

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4 August 2017

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