(Q35190730)

7 August 2017

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title

Mechanistic considerations in high-throughput screening (English)

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7 August 2017

Robert A Copeland

1

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7 August 2017

language of work or name

English

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publication date

1 September 2003

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7 August 2017

published in

Analytical Biochemistry

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7 August 2017

volume

320

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7 August 2017

issue

1

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7 August 2017

page(s)

1-12

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A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

7 August 2017

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7 January 2021

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Dose any enzyme follow the Michaelis-Menten equation?

7 January 2021

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7 January 2021

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Enoyl-ACP reductase (FabI) of Haemophilus influenzae: steady-state kinetic mechanism and inhibition by triclosan and hexachlorophene

7 January 2021

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7 January 2021

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Mutagenesis and mechanism-based inhibition of Streptococcus pyogenes Glu-tRNAGln amidotransferase implicate a serine-based glutaminase site

7 January 2021

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Comparative studies of active site-ligand interactions among various recombinant constructs of human beta-amyloid precursor protein cleaving enzyme

7 January 2021

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Designing screens: how to make your hits a hit.

7 January 2021

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7 January 2021

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Specificity of natural and artificial substrates for human Cdc25A.

7 January 2021

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7 January 2021

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An exact mathematical expression for describing competitive binding of two different ligands to a protein molecule.

7 January 2021

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Nematode anticoagulant protein c2 reveals a site on factor Xa that is important for macromolecular substrate binding to human prothrombinase

7 January 2021

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Is the isolated ligand binding domain a good model of the domain in the native receptor?

7 January 2021

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10.1016/S0003-2697(03)00346-4

7 January 2021

Identifiers

DOI

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7 August 2017

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