(Q35906971)

11 August 2017

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title

Beta-lactamase inhibitors: evolving compounds for evolving resistance targets (English)

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11 August 2017

author name string

Nafsika H Georgopapadakou

series ordinal

1

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11 August 2017

language of work or name

English

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publication date

1 October 2004

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Expert Opinion on Investigational Drugs

11 August 2017

published in

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11 August 2017

volume

13

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11 August 2017

issue

10

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11 August 2017

page(s)

1307-1318

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Recent Developments in the Field of β-Lactam Antibiotics

11 August 2017

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21 January 2018

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Site-saturation mutagenesis and three-dimensional modelling of ROB-1 define a substrate binding role of Ser130 in class A beta-lactamases

21 January 2018

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21 January 2018

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21 January 2018

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Critical involvement of a carbamylated lysine in catalytic function of class D -lactamases

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Predicting the emergence of antibiotic resistance by directed evolution and structural analysis

21 January 2018

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Evolution of the serine beta-lactamases: past, present and future.

21 January 2018

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21 January 2018

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b-Lactamase inhibitors

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Variety of beta-lactamases produced by amoxicillin-clavulanate-resistant Escherichia coli isolated in the northeastern United States

21 January 2018

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Tazobactam inactivation of SHV-1 and the inhibitor-resistant Ser130 -->Gly SHV-1 beta-lactamase: insights into the mechanism of inhibition

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Structures of ceftazidime and its transition-state analogue in complex with AmpC beta-lactamase: implications for resistance mutations and inhibitor design

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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In vitro and in vivo activities of AM-112, a novel oxapenem.

21 January 2018

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Pharmacokinetic studies and renal dehydropeptidase stability of the new beta-lactamase inhibitor BRL 42715 in animals

21 January 2018

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Inhibition of Class A and Class C β-Lactamases by Penems: Crystallographic Structures of a Novel 1,4-Thiazepine Intermediate,

21 January 2018

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The complexed structure and antimicrobial activity of a non-β-lactam inhibitor of AmpC β-lactamase

21 January 2018

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Mechanism of inhibition of the class C beta-lactamase of Enterobacter cloacae P99 by phosphonate monoesters

21 January 2018

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Crystallographic structure of a phosphonate derivative of the Enterobacter cloacae P99 cephalosporinase: mechanistic interpretation of a beta-lactamase transition-state analog

21 January 2018

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21 January 2018

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21 January 2018

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Role of OmpD2 and chromosomal β-lactamase in carbapenem resistance in clinical isolates of Pseudomonas aeruginosa

21 January 2018

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Alterations of susceptibility of Pseudomonas aeruginosa by overproduction of multidrug efflux systems, MexAB-OprM, MexCD-OprJ, and MexXY/OprM to carbapenems: substrate specificities of the efflux systems

21 January 2018

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Extrusion of penem antibiotics by multicomponent efflux systems MexAB-OprM, MexCD-OprJ, and MexXY-OprM of Pseudomonas aeruginosa

21 January 2018

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Substrate specificities of MexAB-OprM, MexCD-OprJ, and MexXY-oprM efflux pumps in Pseudomonas aeruginosa

21 January 2018

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Multiple antibiotic resistance in Stenotrophomonas maltophilia: involvement of a multidrug efflux system

21 January 2018

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10.1517/13543784.13.10.1307

21 January 2018

Identifiers

DOI

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11 August 2017

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