(Q36011743)

11 August 2017

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title

Endothelin receptor antagonists. (English)

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11 August 2017

Joel B Nelson

1

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11 August 2017

15 January 2005

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11 August 2017

World Journal of Urology

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11 August 2017

23

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11 August 2017

1

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11 August 2017

19-27

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https://scigraph.springernature.com/pub.10.1007/s00345-004-0478-9

11 August 2017

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cites work

Local injection of endothelin-1 produces pain-like behavior and excitation of nociceptors in rats

1 reference

12 December 2020

Role of transactivation of the EGF receptor in signalling by G-protein-coupled receptors

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12 December 2020

New bone formation in an osteoblastic tumor model is increased by endothelin-1 overexpression and decreased by endothelin A receptor blockade

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12 December 2020

Production of endothelin in human cancer cell lines

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12 December 2020

Neutral endopeptidase 24.11 loss in metastatic human prostate cancer contributes to androgen-independent progression

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12 December 2020

Gene expression and autoradiographic localization of endothelin-1 and its receptors A and B in the different zones of the normal human prostate

1 reference

12 December 2020

The endothelin receptor B (EDNRB) promoter displays heterogeneous, site specific methylation patterns in normal and tumor cells

1 reference

12 December 2020

Endothelin-1 is an autocrine/paracrine growth factor for human cancer cell lines

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12 December 2020

A survey of gene-specific methylation in human prostate cancer among black and white men.

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12 December 2020

Localization of endothelin receptors in the human prostate

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12 December 2020

Atrasentan, an endothelin-receptor antagonist for refractory adenocarcinomas: safety and pharmacokinetics

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12 December 2020

Endothelin-1 participation in overt and inflammatory pain

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12 December 2020

Endothelin-1-induced nociception

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12 December 2020

Endothelin B receptor gene hypermethylation in prostate adenocarcinoma

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12 December 2020

Promoter hypermethylation of the EDNRB gene in nasopharyngeal carcinoma.

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12 December 2020

Molecular and physiologic evidence for 5'CpG island methylation of the endothelin B receptor gene in lung cancer

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12 December 2020

Endothelin-1 activates phospholipase C and mobilizes Ca2+ from extra- and intracellular pools in osteoblastic cells

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12 December 2020

Cell proliferation, DNA repair, and p53 function are not required for programmed death of prostatic glandular cells induced by androgen ablation

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12 December 2020

Upregulation of endothelin 1 and its precursor by IL-1beta, TNF-alpha, and TGF-beta in the PC3 human prostate cancer cell line

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12 December 2020

Suppression of prostate cancer induced bone remodeling by the endothelin receptor A antagonist atrasentan

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12 December 2020

Endothelin-1 gene expression and regulation of endothelin mRNA and protein biosynthesis in avascular human amnion. Potential source of amniotic fluid endothelin

1 reference

12 December 2020

Endothelin-1 in the human prostate: tissue levels, source of production and isometric tension studies

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12 December 2020

Expression of endothelin receptor a associated with prostate cancer progression

1 reference

12 December 2020

Identification of endothelin-1 in the pathophysiology of metastatic adenocarcinoma of the prostate

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12 December 2020

Pharmacokinetics and pharmacodynamic effects of ABT-627, an oral ETA selective endothelin antagonist, in humans

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12 December 2020

Endothelin-1 (ET-1) selectively enhances the activation gating of slowly inactivating tetrodotoxin-resistant sodium currents in rat sensory neurons: a mechanism for the pain-inducing actions of ET-1.

1 reference

12 December 2020

Regional haemodynamic effects of endothelin-1 in rat and man: unexpected adverse reaction

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12 December 2020

Articular nociception induced by endothelin-1, carrageenan and LPS in naive and previously inflamed knee-joints in the rat: inhibition by endothelin receptor antagonists

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12 December 2020

Conversion of big endothelin-1 to 21-residue endothelin-1 is essential for expression of full vasoconstrictor activity: structure-activity relationships of big endothelin-1

1 reference

12 December 2020

Functional interactions between tumor and peripheral nerve: morphology, algogen identification, and behavioral characterization of a new murine model of cancer pain

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12 December 2020

A novel potent vasoconstrictor peptide produced by vascular endothelial cells

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12 December 2020

Mitogenic activity of endothelin on human cultured prostatic smooth muscle cells.

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12 December 2020

Presence of immunoreactive endothelin in human plasma

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12 December 2020

The endothelin axis: emerging role in cancer

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12 December 2020

Endothelins: circulating plasma levels and presence in other biologic fluids

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12 December 2020

Endothelin family in human plasma and cerebrospinal fluid

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12 December 2020

Production of endothelin-1 and big-endothelin-1 by tumor cells with epithelial-like morphology

1 reference

12 December 2020

Effect of endothelin-A receptor blockade with atrasentan on tumor progression in men with hormone-refractory prostate cancer: a randomized, phase II, placebo-controlled trial

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12 December 2020

Methylation of the 5' CpG island of the endothelin B receptor gene is common in human prostate cancer.

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12 December 2020

Endothelin stimulates DNA synthesis in Swiss 3T3 cells. Synergy with polypeptide growth factors

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12 December 2020

Endothelin-1 production by prostate cancer cell lines is up-regulated by factors involved in cancer progression and down-regulated by androgens

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12 December 2020

Single-dose pharmacokinetics of atrasentan, an endothelin-A receptor antagonist

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12 December 2020

Pharmacological characterization of A-127722: an orally active and highly potent ETA-selective receptor antagonist.

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12 December 2020

Massive amounts of immunoreactive endothelin in human seminal fluid

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12 December 2020

Endothelin-1-induced ET(A) receptor-mediated nociception, hyperalgesia and oedema in the mouse hind-paw: modulation by simultaneous ET(B) receptor activation

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12 December 2020

Endothelin-1 production and decreased endothelin B receptor expression in advanced prostate cancer

1 reference

12 December 2020

Behavioral signs of acute pain produced by application of endothelin-1 to rat sciatic nerve.

1 reference

12 December 2020

Phase I dose-escalation study of the safety and pharmacokinetics of atrasentan: an endothelin receptor antagonist for refractory prostate cancer.

1 reference

12 December 2020

Hypermethylation of CpG islands in primary and metastatic human prostate cancer.

1 reference

12 December 2020

Presence of immunoreactive endothelin in human milk

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12 December 2020

1 reference

12 December 2020

The human endothelin family: three structurally and pharmacologically distinct isopeptides predicted by three separate genes

1 reference

12 December 2020

Characterization of endothelin-induced nociception in mice: evidence for a mechanistically distinct analgesic model

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12 December 2020

Endothelin and the tumorigenic component of bone cancer pain.

1 reference

12 December 2020

A causal role for endothelin-1 in the pathogenesis of osteoblastic bone metastases

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12 December 2020

Perioperative plasma endothelin-1 and Big endothelin-1 concentrations in elderly patients undergoing major surgical procedures

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12 December 2020

10.1007/S00345-004-0478-9

Identifiers

DOI

1 reference

11 August 2017

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PubMed ID

15654644