(Q36052584)

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Antagonist, partial agonist and antiproliferative actions of B-9870 (CU201) as a function of the expression and density of the bradykinin B1 and B2 receptors

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

Antagonist, partial agonist and antiproliferative actions of B-9870 (CU201) as a function of the expression and density of the bradykinin B1 and B2 receptors (English)

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

François Marceau

5

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

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G Morissette

1

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23 December 2019

S Houle

2

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

L Gera

3

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

J M Stewart

4

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23 December 2019

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18 December 2006

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23 December 2019

British Journal of Pharmacology

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

150

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

3

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23 December 2019

369-379

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

Arginine-rich cell penetrating peptides: from endosomal uptake to nuclear delivery

1 reference

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2 October 2017

The C3a receptor antagonist SB 290157 has agonist activity

1 reference

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2 October 2017

Combination cancer chemotherapy with one compound: pluripotent bradykinin antagonists

1 reference

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2 October 2017

International union of pharmacology. XLV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences

1 reference

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2 October 2017

Loss of function of vascular smooth muscle cells by nitric oxide-dependent and -independent interactions with tumorigenic cells

1 reference

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2 October 2017

A novel nonpeptide antagonist of the kinin B1 receptor: effects at the rabbit receptor

1 reference

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2 October 2017

Tissue kallikrein actions at the rabbit natural or recombinant kinin B2 receptors.

1 reference

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2 October 2017

Arginine containing peptides as delivery vectors.

1 reference

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2 October 2017

Kinin receptors: functional aspects.

1 reference

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2 October 2017

Bradykinin-related compounds as new drugs for cancer and inflammation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Bradykinin antagonist dimer, CU201, inhibits the growth of human lung cancer cell lines by a "biased agonist" mechanism

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Bombesin and substance P analogues differentially regulate G-protein coupling to the bombesin receptor. Direct evidence for biased agonism

1 reference

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2 October 2017

In various tumour cell lines the peptide bradykinin B(2) receptor antagonist, Hoe 140 (Icatibant), may act as mitogenic agonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Antagonist-induced intracellular sequestration of rabbit bradykinin B(2) receptor.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Pharmacological profile of LF 16-0687, a new potent non-peptide bradykinin B2 receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Spontaneous human B2 bradykinin receptor activity determines the action of partial agonists as agonists or inverse agonists. Effect of basal desensitization

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Bradykinin-induced internalization of the human B2 receptor requires phosphorylation of three serine and two threonine residues at its carboxyl tail.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Ligand-induced phosphorylation/dephosphorylation of the endogenous bradykinin B2 receptor from human fibroblasts

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

A new class of potent bradykinin antagonist dimers

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Cloning and pharmacological characterization of the rabbit bradykinin B2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Agonistic and antagonistic properties of the bradykinin B2 receptor antagonist, Hoe 140, in isolated blood vessels from different species

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

A synthetic inhibitor of the mitogen-activated protein kinase cascade

1 reference

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2 October 2017

Methods used for the study of opioid receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

2 October 2017

Potent, long-acting bradykinin antagonists for a wide range of applications

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

11 July 2018

Cloning and functional characterization of the ornithokinin receptor. Recognition of the major kinin receptor antagonist, HOE140, as a full agonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

11 July 2018

A new generation of bradykinin antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

11 July 2018

Receptor-mediated internalization of bradykinin. DDT1 MF-2 smooth muscle cells process internalized bradykinin via multiple degradative pathways

1 reference

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11 July 2018

Prostaglandin E2 inhibits the phospholipase D pathway stimulated by formyl-methionyl-leucyl-phenylalanine in human neutrophils. Involvement of EP2 receptors and phosphatidylinositol 3-kinase gamma.

1 reference

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23 September 2018

Discovery of a potent, non-peptide bradykinin B1 receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

23 September 2018

Bradykinin antagonist dimer, CU201, inhibits the growth of human lung cancer cell lines in vitro and in vivo and produces synergistic growth inhibition in combination with other antitumor agents

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2013894

23 September 2018

Agonist-induced translocation of the kinin B(1) receptor to caveolae-related rafts.

1 reference

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23 September 2018

Bradykinin B(2) receptor endocytosis, recycling, and down-regulation assessed using green fluorescent protein conjugates

1 reference

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23 September 2018

Bradykinin receptor subtype 1 expression and function in prostate cancer

1 reference

https://pubmed.ncbi.nlm.nih.gov/17179948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Bradykinin Sequesters B2 Bradykinin Receptors and the Receptor-coupled Gα Subunits Gαq and Gαiin Caveolae in DDT1 MF-2 Smooth Muscle Cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/17179948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Agonist-induced redistribution of bradykinin B2 receptor in caveolae

1 reference

https://pubmed.ncbi.nlm.nih.gov/17179948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1038/SJ.BJP.0706982

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17179948%20AND%20SRC:MED&resulttype=core&format=json

23 December 2019

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