(Q36105351)

English

Potent inhibition of human sulfotransferase 1A1 by 17α-ethinylestradiol: role of 3'-phosphoadenosine 5'-phosphosulfate binding and structural rearrangements in regulating inhibition and activity

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

Potent inhibition of human sulfotransferase 1A1 by 17α-ethinylestradiol: role of 3'-phosphoadenosine 5'-phosphosulfate binding and structural rearrangements in regulating inhibition and activity (English)

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

author name string

Katie Jo Rohn

1

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

Ian T Cook

2

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

Thomas S Leyh

3

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

Susan A Kadlubar

4

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

Charles N Falany

5

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

language of work or name

1 reference

based on heuristic

inferred from title

publication date

16 May 2012

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

Drug Metabolism and Disposition

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

40

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

8

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

1588-1595

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

24-hydroxycholesterol sulfation by human cytosolic sulfotransferases: formation of monosulfates and disulfates, molecular modeling, sulfatase sensitivity, and inhibition of liver x receptor activation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Comparative protein structure modeling using MODELLER

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Structural and chemical profiling of the human cytosolic sulfotransferases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Pharmacokinetic drug interactions involving 17alpha-ethinylestradiol: a new look at an old drug

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Human cytosolic sulfotransferase SULT1A1.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Establishment of detailed reference values for luteinizing hormone, follicle stimulating hormone, estradiol, and progesterone during different phases of the menstrual cycle on the Abbott ARCHITECT analyzer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

The structure of human SULT1A1 crystallized with estradiol. An insight into active site plasticity and substrate inhibition with multi-ring substrates

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Structure of a human carcinogen-converting enzyme, SULT1A1. Structural and kinetic implications of substrate inhibition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Expression and characterization of the human 3 beta-hydroxysteroid sulfotransferases (SULT2B1a and SULT2B1b)

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Estrogen metabolism by conjugation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Sulfotransferases: genetics and role in toxicology

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

A single amino acid, glu146, governs the substrate specificity of a human dopamine sulfotransferase, SULT1A3

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Sulfuryl transfer: the catalytic mechanism of human estrogen sulfotransferase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Sulfation and sulfotransferases 5: the importance of 3'-phosphoadenosine 5'-phosphosulfate (PAPS) in the regulation of sulfation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Prediction of protein side-chain rotamers from a backbone-dependent rotamer library: a new homology modeling tool

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Enzymology of human cytosolic sulfotransferases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Expression of cytosolic sulfotransferases in normal mammary epithelial cells and breast cancer cell lines

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Human dehydroepiandrosterone sulfotransferase. Purification, molecular cloning, and characterization.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Comparative protein modelling by satisfaction of spatial restraints

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Steroid sulfation by expressed human cytosolic sulfotransferases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Bacterial expression and characterization of a cDNA for human liver estrogen sulfotransferase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 October 2017

Structural rearrangement of SULT2A1: effects on dehydroepiandrosterone and raloxifene sulfation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

2 July 2018

On the perception of molecules from 3D atomic coordinates

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

23 September 2018

Sulfation of environmental estrogens by cytosolic human sulfotransferases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

23 September 2018

Regioselective monosulfation and disulfation of the phytoestrogens daidzein and genistein by human liver sulfotransferases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

23 September 2018

Sulfotransferase 1E1 is a low km isoform mediating the 3-O-sulfation of ethinyl estradiol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

23 September 2018

The involvement of CYP3A4 and CYP2C9 in the metabolism of 17 alpha-ethinylestradiol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

23 September 2018

Regulation of MCF-7 breast cancer cell growth by beta-estradiol sulfation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3400793

23 September 2018

Formation of ethinylestradiol in postmenopausal women during continuous treatment with a combination of estradiol, estriol and norethisterone acetate

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evaluation of ligand overlap by atomic parameters

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The effects of rifampin and rifabutin on the pharmacokinetics and pharmacodynamics of a combination oral contraceptive

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Purification and characterization of human liver phenol-sulfating phenol sulfotransferase

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The effect of fluconazole on circulating ethinyl estradiol levels in women taking oral contraceptives

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Oral Contraceptives Induce Lamotrigine Metabolism: Evidence from a Double-blind, Placebo-controlled Trial

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multiple flexible alignment with SEAL: a study of molecules acting on the colchicine binding site

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Regulation of estrogen activity by sulfation in human Ishikawa endometrial adenocarcinoma cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/22593037

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1124/DMD.112.045583

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

12 August 2017

ResearchGate publication ID

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