(Q37204922)

18 August 2017

1 reference

title

Allosteric antagonists of the muscarinic acetylcholine receptor (English)

1 reference

18 August 2017

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

author name string

N. H. Lee

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1859442

11 December 2022

E. E. el-Fakahany

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1859442

11 December 2022

language of work or name

English

0 references

publication date

1 July 1991

1 reference

18 August 2017

5 July 1991

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=1859442

full work available at URL

11 December 2022

https://api.elsevier.com/content/article/PII:0006295291907038?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

https://api.elsevier.com/content/article/PII:0006295291907038?httpAccept=text/plain

11 December 2022

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

published in

Biochemical Pharmacology

1 reference

18 August 2017

42

1 reference

18 August 2017

199-205

1 reference

18 August 2017

2

1 reference

Identification of a family of muscarinic acetylcholine receptor genes

18 August 2017

2

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

A family of receptors coupled to guanine nucleotide regulatory proteins

11 December 2022

3

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Molecular biology of adrenergic and muscarinic cholinergic receptors. A perspective

11 December 2022

4

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Cloning, sequencing and expression of complementary DNA encoding the muscarinic acetylcholine receptor

11 December 2022

5

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Muscarinic receptor differentiation

11 December 2022

7

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

ON THE NATURE OF ALLOSTERIC TRANSITIONS: A PLAUSIBLE MODEL

11 December 2022

10

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Comparison of Experimental Binding Data and Theoretical Models in Proteins Containing Subunits*

11 December 2022

11

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Pirenzepine distinguishes between different subclasses of muscarinic receptors

11 December 2022

15

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Modification of the binding properties of muscarinic receptors by gallamine

11 December 2022

16

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Some quantitative uses of drug antagonists

11 December 2022

18

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The Uptake of Atropine and Related Drugs by Intestinal Smooth Muscle of the Guinea-Pig in Relation to Acetylcholine Receptors

11 December 2022

19

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The inhibitory effect of gallamine on muscarinic receptors

11 December 2022

21

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Heterogeneity of binding sites on cardiac muscarinic receptors induced by the neuromuscular blocking agents gallamine and pancuronium

11 December 2022

22

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Stabilization of antagonist binding to cardiac muscarinic acetylcholine receptors by gallamine and other neuromuscular blocking drugs

11 December 2022

24

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Effects of d-tubocurarine on rat cardiac muscarinic receptors: a comparison with gallamine

11 December 2022

25

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The interaction of pancuronium with cardiac and ileal muscarinic receptors

11 December 2022

26

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The interaction of nicotinic receptor antagonists at muscarinic receptors.

11 December 2022

27

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Binding and functional characterization of the cardioselective muscarinic antagonist methoctramine

11 December 2022

28

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Allosteric interactions of three muscarine antagonists at bovine tracheal smooth muscle and cardiac M2 receptors

11 December 2022

29

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The allosteric binding profile of himbacine: a comparison with other cardioselective muscarinic antagonists

11 December 2022

30

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Characterization of the antimuscarinic effect of heptane-1,7-bis-(dimethyl-3'-phthalimidopropyl ammonium bromide).

11 December 2022

31

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The interaction of hexamethonium with muscarinic receptor subtypes in vitro

11 December 2022

32

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Inhibitory effects of quinidine on rat heart muscarinic receptors.

11 December 2022

33

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Interactions of quinidine and lidocaine with rat brain and heart muscarinic receptors.

11 December 2022

34

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Bretylium tosylate binds preferentially to muscarinic receptors labelled with [3H]oxotremorine M (SH or 'high affinity' receptors) in rat heart and brain cortex

11 December 2022

35

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Interaction of DPI 201-106 with cardiac muscarinic receptors

11 December 2022

36

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Potassium channel blockers differentially affect carbachol and (-)-N6-phenylisopropyladenosine on guinea-pig atria

11 December 2022

37

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Effects of verapamil on the binding properties of rat heart muscarinic receptors: evidence for an allosteric site

11 December 2022

38

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Verapamil interaction with the muscarinic receptor: stereoselectivity at two sites

11 December 2022

39

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Gallamine exerts biphasic allosteric effects at muscarinic receptors

11 December 2022

40

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Characterization of guinea-pig cardiac muscarinic receptors by radioligand dissociation kinetics

11 December 2022

41

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The effect of McN-A-343 on muscarinic receptors in the cerebral cortex and heart

11 December 2022

42

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Myocardial muscarinic acetylcholine receptor: choline and tris unmask heterogeneity of antagonist binding sites.

11 December 2022

43

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Obligatory role of a Tris/choline allosteric site in guanine nucleotide regulation of [3H]-L-QNB binding to muscarinic acetylcholine receptors

11 December 2022

44

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Comparative binding studies with cholinergic ligands and histrionicotoxin at muscarinic receptors of neural cell lines

11 December 2022

45

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Allosteric effect of gallamine on muscarinic cholinergic receptor binding: influence of guanine nucleotides and conformational state

11 December 2022

46

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

In vitro effects of gallamine on dissociation kinetics of (3H)N-methylscopolamine and (3H)pirenzepine from rat brain muscarinic receptors.

11 December 2022

47

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Mixed competitive and allosteric antagonism by gallamine of muscarinic receptor-mediated second messenger responses in N1E-115 neuroblastoma cells.

11 December 2022

48

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Possible allosteric interaction of 4-aminopyridine with rat brain muscarinic acetylcholine receptors.

11 December 2022

49

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Effects of verapamil on the binding characteristics of muscarinic receptor subtypes.

11 December 2022

50

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Secoverine is a non-selective muscarinic antagonist on rat heart and brain receptors.

11 December 2022

51

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Allosteric interactions between muscarinic agonist binding sites and effector sites demonstrated by the use of bisquaternary pyridinium oximes.

11 December 2022

53

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The differential loss of [3H]pirenzepine vs [3H] (-) quinuclidinylbenzilate binding to soluble rat brain muscarinic receptors indicates that pirenzepine binds to an allosteric state of the muscarinic receptor

11 December 2022

54

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Multiple in vitro interactions with and differential in vivo regulation of muscarinic receptor subtypes by tetrahydroaminoacridine

11 December 2022

56

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Different mechanisms of antagonism by methoctramine of two neuronal muscarinic receptor-mediated second messenger responses

11 December 2022

57

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Antimuscarinic action of methoctramine, a new cardioselective M-2 muscarinic receptor antagonist, alone and in combination with atropine and gallamine

11 December 2022

58

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The interaction of methoctramine and himbacine at atrial, smooth muscle and endothelial muscarinic receptors in vitro

11 December 2022

59

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Competitive and non-competitive antagonism exhibited by 'selective' antagonists at atrial and ileal muscarinic receptor subtypes

11 December 2022

60

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Pharmacologic discrimination between receptor heterogeneity and allosteric interaction: resultant analysis of gallamine and pirenzepine antagonism of muscarinic responses in rat trachea

11 December 2022

62

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Differential allosteric effects of 8-(N,N-diethylamino)octyl-3,4,5-trimethoxybenzoate-HCl (TMB-8) on muscarinic receptor subtypes

11 December 2022

64

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The pharmacology of Flaxedil, with observations on certain analogs

11 December 2022

65

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The sympathomimetic effect of gallamine on the heart

11 December 2022

66

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Regional distribution of muscarinic receptors preferring gallamine in the rat brain.

11 December 2022

68

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The interaction of hemicholinium-3 (HC-3) with cholinomimetics and atropine

11 December 2022

69

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Muscarinic receptor heterogeneity in rat central nervous system. II. Brain receptors labeled by [3H]oxotremorine-M correspond to heterogeneous M2 receptors with very high affinity for agonists

11 December 2022

70

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Competitive interaction of gallamine with multiple muscarinic receptors.

11 December 2022

71

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Characterization of the interactions of gallamine with muscarinic receptors from brain.

11 December 2022

72

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Effects of gallamine triethiodide on membrane currents in amphibian and mammalian peripheral nerve

11 December 2022

76

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

GTP-binding proteins couple cardiac muscarinic receptors to a K channel.

11 December 2022

79

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Uncoupling of cardiac muscarinic and beta-adrenergic receptors from ion channels by a guanine nucleotide analogue

11 December 2022

80

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Polymethylene tetraamines as muscarinic receptor probes

11 December 2022

83

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Reduction of muscarinic acetylcholine receptor number and affinity by an endogenous substance.

11 December 2022

84

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Endogenous inhibitor of ligand binding to the muscarinic acetylcholine receptor

11 December 2022

85

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

Identifiers

1 reference

18 August 2017

1 reference