(Q37359930)

English

(1R, 3S)-(-)-trans-PAT: a novel full-efficacy serotonin 5-HT2C receptor agonist with 5-HT2A and 5-HT2B receptor inverse agonist/antagonist activity

scientific article published on 03 May 2009

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scholarly article

1 reference

Europe PubMed Central

19 August 2017

(1R, 3S)-(-)-trans-PAT: a novel full-efficacy serotonin 5-HT2C receptor agonist with 5-HT2A and 5-HT2B receptor inverse agonist/antagonist activity (English)

1 reference

Europe PubMed Central

19 August 2017

0 references

author name string

Raymond G Booth

1

1 reference

Europe PubMed Central

19 August 2017

Lijuan Fang

2

1 reference

Europe PubMed Central

19 August 2017

Yingsu Huang

3

1 reference

Europe PubMed Central

19 August 2017

Andrzej Wilczynski

4

1 reference

Europe PubMed Central

19 August 2017

Sashikala Sivendran

5

1 reference

Europe PubMed Central

19 August 2017

language of work or name

0 references

publication date

3 May 2009

1 reference

Europe PubMed Central

19 August 2017

European Journal of Pharmacology

1 reference

Europe PubMed Central

19 August 2017

615

1 reference

Europe PubMed Central

19 August 2017

1-3

1 reference

Europe PubMed Central

19 August 2017

1-9

1 reference

Europe PubMed Central

19 August 2017

Prospects for serotonin 5-HT2R pharmacotherapy in psychostimulant abuse

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Effect of (-)-trans-PAT, a novel 5-HT2C receptor agonist, on intake of palatable food in mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Lorcaserin, a novel selective human 5-hydroxytryptamine2C agonist: in vitro and in vivo pharmacological characterization

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Identification of a key amino acid of the human 5-HT(2B) serotonin receptor important for sarpogrelate binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Serotonin 5-HT(2C) receptors regulate anxiety-like behavior

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Antidepressant-like effects of the novel, selective, 5-HT2C receptor agonist WAY-163909 in rodents

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

CP-809,101, a selective 5-HT2C agonist, shows activity in animal models of antipsychotic activity

1 reference

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6 September 2017

Potential role of new therapies in modifying cardiovascular risk in overweight patients with metabolic risk factors

1 reference

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6 September 2017

Antiobesity-like effects of the 5-HT2C receptor agonist WAY-161503.

1 reference

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6 September 2017

Molecular determinants for the interaction of the valvulopathic anorexigen norfenfluramine with the 5-HT2B receptor

1 reference

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6 September 2017

Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

1 reference

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6 September 2017

H1-histamine receptor affinity predicts short-term weight gain for typical and atypical antipsychotic drugs.

1 reference

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6 September 2017

Differential effects of the 5-HT(2A) receptor antagonist M100907 and the 5-HT(2C) receptor antagonist SB242084 on cocaine-induced locomotor activity, cocaine self-administration and cocaine-induced reinstatement of responding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Function of the serotonin 5-hydroxytryptamine 2B receptor in pulmonary hypertension

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Functional role of internal water molecules in rhodopsin revealed by X-ray crystallography.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Multiplicity of mechanisms of serotonin receptor signal transduction

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Evidence that hypophagia induced by d-fenfluramine and d-norfenfluramine in the rat is mediated by 5-HT2C receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Structural mimicry in G protein-coupled receptors: implications of the high-resolution structure of rhodopsin for structure-function analysis of rhodopsin-like receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Possible role of valvular serotonin 5-HT(2B) receptors in the cardiopathy associated with fenfluramine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Functional characterization of agonists at recombinant human 5-HT2A, 5-HT2B and 5-HT2C receptors in CHO-K1 cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Eating disorder and epilepsy in mice lacking 5-HT2c serotonin receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Cloning of the human serotonin 5-HT2 and 5-HT1C receptor subtypes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

6 September 2017

Identification of amino acid residues important for sarpogrelate binding to the human 5-hydroxytryptamine2A serotonin receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

14 September 2017

Reversal of phenylpropanolamine anorexia in rats by the alpha-1 receptor antagonist benoxathian

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

28 September 2017

Role of PKA and PKC in histamine H1 receptor-mediated activation of catecholamine neurotransmitter synthesis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

26 June 2018

Site-directed mutagenesis of the serotonin 5-Hydroxytryptamine2c receptor: identification of amino acids responsible for sarpogrelate binding.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

26 June 2018

A paradoxical locomotor response in serotonin 5-HT(2C) receptor mutant mice.

1 reference

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26 June 2018

Molecular dynamics simulations of a fluid bilayer of dipalmitoylphosphatidylcholine at full hydration, constant pressure, and constant temperature

1 reference

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26 June 2018

Site-directed mutagenesis of the serotonin 5-hydroxytrypamine2 receptor: identification of amino acids necessary for ligand binding and receptor activation

1 reference

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26 June 2018

Synthesis and pharmacological evaluation of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for a novel receptor with sigma-like neuromodulatory activity

1 reference

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26 June 2018

NIH symposium series: ingestive mechanisms in obesity, substance abuse and mental disorders.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

2 September 2018

Ligand-directed functional heterogeneity of histamine H1 receptors: novel dual-function ligands selectively activate and block H1-mediated phospholipase C and adenylyl cyclase signaling

1 reference

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2 September 2018

Domain swapping in the human histamine H1 receptor

1 reference

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2 September 2018

Aminorex, fenfluramine, and chlorphentermine are serotonin transporter substrates. Implications for primary pulmonary hypertension.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2749987

2 September 2018

5-HT(2C) receptor antagonists enhance the behavioural response to dopamine D(1) receptor agonists in the 6-hydroxydopamine-lesioned rat

1 reference

https://pubmed.ncbi.nlm.nih.gov/19397907

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

5-HT2C receptor binding is increased in the substantia nigra pars reticulata in Parkinson's disease

1 reference

https://pubmed.ncbi.nlm.nih.gov/19397907

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Molecular dynamics simulation of HIV-1 protease in a crystalline environment and in solution

1 reference

https://pubmed.ncbi.nlm.nih.gov/19397907

12 December 2020

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The selective norepinephrine reuptake inhibitor, LY368975, reduces food consumption in animal models of feeding

1 reference

https://pubmed.ncbi.nlm.nih.gov/19397907

12 December 2020

based on heuristic

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In vivo model of drug-induced valvular heart disease in rats: pergolide-induced valvular heart disease demonstrated with echocardiography and correlation with pathology

1 reference

https://pubmed.ncbi.nlm.nih.gov/19397907

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.EJPHAR.2009.04.035

1 reference

Europe PubMed Central

19 August 2017

1 reference

Europe PubMed Central

19 August 2017

1 reference

Europe PubMed Central

19 August 2017

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