(Q37568526)

21 August 2017

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title

Ligands, their receptors and ... plasma membranes (English)

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21 August 2017

G Vauquelin

1

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PubMed ID

19647036

21 August 2017

A Packeu

series ordinal

2

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21 August 2017

30 July 2009

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Molecular and Cellular Endocrinology

21 August 2017

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21 August 2017

311

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21 August 2017

1-2

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21 August 2017

1-10

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Kinetic versus allosteric mechanisms to explain insurmountable antagonism and delayed ligand dissociation

21 August 2017

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12 December 2020

Efforts to understand the molecular basis of hypertension through drug:membrane interactions

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12 December 2020

Molecular mechanisms of beta(2)-adrenergic receptor function, response, and regulation

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12 December 2020

How lipophilic cannabinergic ligands reach their receptor sites

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12 December 2020

The agonist effect of dihydropyridines on Ca channels

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12 December 2020

Mapping of ligand binding sites of the cholecystokinin-B/gastrin receptor with lipo-gastrin peptides and molecular modeling.

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12 December 2020

New dimensions in two dimensions

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12 December 2020

Rates of membrane-associated reactions: reduction of dimensionality revisited

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12 December 2020

Carrier proteins determine local pharmacokinetics and arterial distribution of paclitaxel

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12 December 2020

Effect of nonspecific forces and finite receptor number on rate constants of ligand--cell bound-receptor interactions

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12 December 2020

Antagonist-radioligand binding to D2L-receptors in intact cells

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12 December 2020

Evidence for a C-terminal structural motif in gastrin and its bioactive fragments in membrane mimetic media

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12 December 2020

Allosteric modulation of the cannabinoid CB1 receptor

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12 December 2020

Drug-target residence time and its implications for lead optimization

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12 December 2020

Allosteric interactions required for high-affinity binding of dihydropyridine antagonists to Ca(V)1.1 Channels are modulated by calcium in the pore

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12 December 2020

Endothelin ET(B) receptors show different binding profiles in intact cells and cell membrane preparations

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12 December 2020

Conformation and orientation of regulatory peptides on lipid membranes. Key to the molecular mechanism of receptor selection.

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12 December 2020

The pharmacology of salmeterol

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12 December 2020

Residence time of receptor-ligand complexes and its effect on biological function

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12 December 2020

The conformational properties of the highly selective cannabinoid receptor ligand CP-55,940

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12 December 2020

Risperidone irreversibly binds to and inactivates the h5-HT7 serotonin receptor

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12 December 2020

L-type calcium channels: asymmetrical intramembrane binding domain revealed by variable length, permanently charged 1,4-dihydropyridines

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12 December 2020

Peptide hormone-membrane interactions: the aggregational and conformational state of lipo-gastrin derivatives and their receptor binding affinity.

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12 December 2020

The conformation, location, and dynamic properties of the endocannabinoid ligand anandamide in a membrane bilayer

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12 December 2020

Reduction-of-dimensionality kinetics at reaction-limited cell surface receptors

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12 December 2020

Reevaluating equilibrium and kinetic binding parameters for lipophilic drugs based on a structural model for drug interaction with biological membranes

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12 December 2020

Possible molecular basis for the pharmacokinetics and pharmacodynamics of three membrane-active drugs: propranolol, nimodipine and amiodarone

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12 December 2020

Two types of Alzheimer's beta-amyloid (1-40) peptide membrane interactions: aggregation preventing transmembrane anchoring versus accelerated surface fibril formation.

1 reference

12 December 2020

A molecular model involving the membrane bilayer in the binding of lipid soluble drugs to their receptors in heart and brain

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12 December 2020

New evidence for a membrane-bound pathway in hormone receptor binding

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12 December 2020

Kinetics of binding of membrane-active drugs to receptor sites. Diffusion-limited rates for a membrane bilayer approach of 1,4-dihydropyridine calcium channel antagonists to their active site.

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12 December 2020

Role of Receptor Protein and Membrane Lipids in Xanomeline Wash-Resistant Binding to Muscarinic M1Receptors

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12 December 2020

Why are long-acting beta-adrenoceptor agonists long-acting?

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12 December 2020

Lipid membrane-induced optimization for ligand-receptor docking: recent tools and insights for the "membrane catalysis" model.

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12 December 2020

Diffusion of dihydropyridine calcium channel antagonists in cardiac sarcolemmal lipid multibilayers

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12 December 2020

Physics of chemoreception

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12 December 2020

Distinct binding properties of the AT(1) receptor antagonist [(3)H]candesartan to intact cells and membrane preparations

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12 December 2020

On the unique binding and activating properties of xanomeline at the M1 muscarinic acetylcholine receptor

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12 December 2020

On the mechanism of hormone recognition and binding by the CCK-B/gastrin receptor

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12 December 2020

Structure and dynamics of micelle-bound neuropeptide Y: comparison with unligated NPY and implications for receptor selection

1 reference

12 December 2020

Exosites: their current status, and their relevance to the duration of action of long-acting beta 2-adrenoceptor agonists

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12 December 2020

Stable activation and desensitization of beta 2-adrenergic receptor stimulation of adenylyl cyclase by salmeterol: evidence for quasi-irreversible binding to an exosite.

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12 December 2020

A thermodynamic approach to problems of drug antagonism I. The "Charnière theory".

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12 December 2020

Losartan's molecular basis of interaction with membranes and AT1 receptor.

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12 December 2020

Salmeterol, a novel, long-acting β2-adrenoceptor agonist: characterization of pharmacological activity in vitro and in vivo

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12 December 2020

Cannabinoid CB1 receptor recognition of endocannabinoids via the lipid bilayer: molecular dynamics simulations of CB1 transmembrane helix 6 and anandamide in a phospholipid bilayer

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12 December 2020

Membrane lipid phase as catalyst for peptide-receptor interactions

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12 December 2020

Conformational changes of adrenocorticotropin peptides upon interaction with lipid membranes revealed by infrared attenuated total reflection spectroscopy

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12 December 2020

The effect of cell size and receptor density on ligand-receptor reaction rate constants

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12 December 2020

Extent of salmeterol-mediated reassertion of relaxation in guinea-pig trachea pretreated with aliphatic side chain structural analogues

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12 December 2020

Mutation studies of Ser7.39 and Ser2.60 in the human CB1 cannabinoid receptor: evidence for a serine-induced bend in CB1 transmembrane helix 7.

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12 December 2020

Integrity of extracellular loop 1 of the human cannabinoid receptor 1 is critical for high-affinity binding of the ligand CP 55,940 but not SR 141716A

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12 December 2020

Allosteric modulation by persistent binding of xanomeline of the interaction of competitive ligands with the M1 muscarinic acetylcholine receptor

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12 December 2020

Partition coefficients of dopamine antagonists in brain membranes and liposomes

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12 December 2020

Conformational studies of corticotropin1–32 and constitutive peptides by circular dichroism

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12 December 2020

Kinetic analysis of drug-receptor interactions of long-acting beta2 sympathomimetics in isolated receptor membranes: evidence against prolonged effects of salmeterol and formoterol on receptor-coupled adenylyl cyclase.

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12 December 2020

Equilibrium and kinetic studies of the interactions of salmeterol with membrane bilayers

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12 December 2020

Molecular mechanisms for the persistent bronchodilatory effect of the beta 2-adrenoceptor agonist salmeterol

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12 December 2020

Amphiphilic Secondary Structure: Design of Peptide Hormones

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12 December 2020

Extracellular space diffusion and extrasynaptic transmission.

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12 December 2020

100 years lock-and-key concept: are peptide keys shaped and guided to their receptors by the target cell membrane?

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12 December 2020

Interaction between dihydropyridines and phospholipid bilayers: a molecular dynamics simulation

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12 December 2020

Formoterol: pharmacology, molecular basis of agonism, and mechanism of long duration of a highly potent and selective beta 2-adrenoceptor agonist bronchodilator

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12 December 2020

Dihydropyridine derivatives prolong the open state of Ca channels in cultured cardiac cells

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12 December 2020

Formoterol on airway smooth muscle and human lung mast cells: a comparison with salbutamol and salmeterol

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12 December 2020

Lipids, lipid rafts and caveolae: their importance for GPCR signaling and their centrality to the endocannabinoid system

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12 December 2020

Reaction rate enhancement by surface diffusion of adsorbates

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12 December 2020

Diffusion delays and unstirred layer effects at monolayer cultures of Chinese hamster ovary cells: radioligand binding, confocal microscopy, and mathematical simulations.

1 reference

12 December 2020

QSAR and the rational design of long-acting dual D2-receptor/beta 2-adrenoceptor agonists

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12 December 2020

Interaction of alpha-melanocyte stimulating hormone with binary phospholipid membranes: structural changes and relevance of phase behavior

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12 December 2020

Effects of the geometry of the immunological synapse on the delivery of effector molecules.

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12 December 2020

Contribution of dead-space microdomains to tortuosity of brain extracellular space

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12 December 2020

Interactions of angiotensin II non-peptide AT(1) antagonist losartan with phospholipid membranes studied by combined use of differential scanning calorimetry and electron spin resonance spectroscopy

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12 December 2020

Sustained activation of a G protein-coupled receptor via "anchored" agonist binding. Molecular localization of the salmeterol exosite within the 2-adrenergic receptor

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12 December 2020

Molecular dynamics simulations of the endocannabinoid N-arachidonoylethanolamine (anandamide) in a phospholipid bilayer: probing structure and dynamics

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12 December 2020

10.1016/J.MCE.2009.07.022

Identifiers

DOI

1 reference

21 August 2017

1 reference

PubMed ID

19647036