(Q38195817)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

review article

1 reference

title

The GABA synapse as a target for antiepileptic drugs: a historical overview focused on GABA transporters (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Melissa L Barker-Haliski

series ordinal

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

author name string

Karsten K Madsen

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

H Steve White

series ordinal

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

language of work or name

1 reference

14 March 2014

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

published in

Neurochemical Research

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

volume

39

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

issue

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

page(s)

1980-1987

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24627365%20AND%20SRC:MED&resulttype=core&format=json

Immunohistochemical localization of glutamate decarboxylase in rat cerebellum

10 March 2020

cites work

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Fine structural localization of glutamine synthetase in astrocytes of rat brain

21 January 2018

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Pyruvate carboxylase activity in primary cultures of astrocytes and neurons

21 January 2018

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Glutamate and GABA synthesis, release, transport and metabolism as targets for seizure control

21 January 2018

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Astrocytic Control of Biosynthesis and Turnover of the Neurotransmitters Glutamate and GABA.

21 January 2018

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Identification and characterization of the vesicular GABA transporter

21 January 2018

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The vesicular neurotransmitter transporters: current perspectives and future prospects

21 January 2018

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https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Postnatal development of the vesicular GABA transporter in rat cerebral cortex.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Effects of valproate, vigabatrin and aminooxyacetic acid on release of endogenous and exogenous GABA from cultured neurons

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Occlusion and metabolism of gamma-aminobutyric acid by brain tissue.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

The uptake of [3H]GABA by slices of rat cerebral cortex

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Cloning and expression of a betaine/GABA transporter from human brain

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

The GABA transporter and its inhibitors

21 January 2018

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Pharmacological and functional characterization of astrocytic GABA transport: a short review

21 January 2018

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Are vesicular neurotransmitter transporters potential treatment targets for temporal lobe epilepsy?

21 January 2018

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Gamma-aminobutyric acid binding to receptor sites in the rat central nervous system.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Properties of γ-aminobutyric acid (GABA) receptor binding in rat brain synaptic membrane fractions

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Structure, pharmacology, and function of GABAA receptor subtypes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

A new class of GABA agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Inhibition of GABA uptake in rat brain slices by nipecotic acid, various isoxazoles and related compounds

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Competitive inhibition of GABA uptake in rat brain slices by some GABA analogues of restricted conformation

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Muscimol uptake, release and binding in rat brain slices

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Betel nut constituents as inhibitors of γ-aminobutyric acid uptake

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Effects of GABA analogues of restricted conformation on GABA transport in astrocytes and brain cortex slices and on GABA receptor binding

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Autoradiographic identification of cerebral and cerebellar cortical neurons accumulating labeled gamma-aminobutyric acid ( 3 H-GABA).

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Studies of the uptake of3H-GABA and [3H]glycine in slices and homogenates of rat brain and spinal cord by electron microscopic autoradiography

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Spinal cord tissue cultures--a model for autoradiographic studies on uptake of putative neurotransmitters such as glycine and GABA.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Selective uptake of [3H]β-alanine by glia: Association with the glial uptake system for GABA

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

The autoradiographic localization of the gaba-releasing nerve terminals in cerebellar glomeruli

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Differential labeling of glial cells and GABA-inhibitory interneurons and nerve terminals following the microinjection of (beta-3H)alanine, (3H)DABA and (3H)GABA into single folia of the cerebellum

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Glial cell function: uptake of transmitter substances

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Uptake of GABA by neuronal and nonneuronal cells in dispersed cell cultures of postnatal rat cerebellum

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Uptake and metabolism of GABA in astrocytes cultured from dissociated mouse brain hemispheres

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Structure-activity relationships of selective GABA uptake inhibitors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

GABAergic mechanisms in the pathogenesis and treatment of epilepsy

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Molecular pathways controlling inhibitory receptor expression

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Influence of inhibitors of the high affinity GABA uptake on seizure thresholds in mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Anticonvulsant activity of GABA uptake inhibitors and their prodrugs following central or systemic administration

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Anticonvulsant activity of the glial-selective GABA uptake inhibitor, THPO.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Transport and Metabolism of 7-Aminobutyric Acid in Neurons and Glia: Implications for Epilepsy

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

The selective blockade by diaminobutyric acid of neuronal uptake of [3H]GABA in rat brain in vivo

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Barbiturate reversal of amino acid antagonism produced by convulsant agents

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Correlation between anticonvulsant activity and inhibitory action on glial gamma-aminobutyric acid uptake of the highly selective mouse gamma-aminobutyric acid transporter 1 inhibitor 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole and its N-

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Orally active and potent inhibitors of gamma-aminobutyric acid uptake

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Kinetic characterization of inhibition of gamma-aminobutyric acid uptake into cultured neurons and astrocytes by 4,4-diphenyl-3-butenyl derivatives of nipecotic acid and guvacine

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain gamma-aminobutyric acid uptake carrier

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

A review of the preclinical pharmacology of tiagabine: a potent and selective anticonvulsant GABA uptake inhibitor

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

1-(3-(9H-carbazol-9-yl)-1-propyl)-4-(2-methoxyphenyl)-4-piperidinol, a novel subtype selective inhibitor of the mouse type II GABA-transporter

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Selective inhibitors of GABA uptake: synthesis and molecular pharmacology of 4-N-methylamino-4,5,6,7-tetrahydrobenzo[d]isoxazol-3-ol analogues

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

First demonstration of a functional role for central nervous system betaine/{gamma}-aminobutyric acid transporter (mGAT2) based on synergistic anticonvulsant action among inhibitors of mGAT1 and mGAT2.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Deletion of the betaine-GABA transporter (BGT1; slc6a12) gene does not affect seizure thresholds of adult mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Neuronal and non-neuronal GABA transporters as targets for antiepileptic drugs

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Synaptic and extrasynaptic GABA transporters as targets for anti-epileptic drugs.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

GABAA receptor alpha 4 subunits mediate extrasynaptic inhibition in thalamus and dentate gyrus and the action of gaboxadol

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Gaboxadol--a new awakening in sleep

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

GABA-level increasing and anticonvulsant effects of three different GABA uptake inhibitors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Differential effects of nipecotic acid and 4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol on extracellular gamma-aminobutyrate levels in rat thalamus.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Selective GABA transporter inhibitors tiagabine and EF1502 exhibit mechanistic differences in their ability to modulate the ataxia and anticonvulsant action of the extrasynaptic GABA(A) receptor agonist gaboxadol.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Effects of gamma-aminobutyric acid (GABA) agonists and GABA uptake inhibitors on pharmacosensitive and pharmacoresistant epileptiform activity in vitro

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

The effects of stiripentol on GABA(A) receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Stiripentol, a putative antiepileptic drug, enhances the duration of opening of GABA-A receptor channels

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

The anti-convulsant stiripentol acts directly on the GABA(A) receptor as a positive allosteric modulator

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Interactions between modulators of the GABA(A) receptor: Stiripentol and benzodiazepines

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Stiripentol in Dravet syndrome: results of a retrospective U.S. study.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Concentrations of stiripentol in children and adults with epilepsy: the influence of dose, age, and comedication

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Anticonvulsant activity of intracerebroventricularly administered glial GABA uptake inhibitors and other GABAmimetics in chemical seizure models

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS11064-014-1263-9

Heterocyclic GABA analogues as selective inhibitors of astroglial GABA uptake

21 January 2018

1 reference

12 December 2020

The excitation and depression of spinal neurones by structurally related amino acids

1 reference

12 December 2020

Convulsant and anticonvulsant actions in DBA/2 mice of compounds blocking the reuptake of GABA

1 reference

12 December 2020

Epilepsy and γ-Aminobutyric Acid-Mediated Inhibition

1 reference

12 December 2020

Novel inhibitors of gamma-aminobutyric acid (GABA) uptake: anticonvulsant actions in rats and mice

1 reference

12 December 2020

Antinociceptive and anticonvulsive effect of THIP, a pure GABA agonist

1 reference

12 December 2020

In vivo changes in the GABA content of nerve endings (synaptosomes) induced by inhibitors of GABA uptake

1 reference

12 December 2020

Anticonvulsant activity of the gamma-aminobutyric acid uptake inhibitor N-4,4-diphenyl-3-butenyl-4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol

1 reference

12 December 2020

Structure and biological activity of a series of conformationally restricted analogues of GABA

1 reference

12 December 2020

gamma-Aminobutyric acid in brain: its formation from glutamic acid.

1 reference

12 December 2020

Transport and Metabolism of Glutamate and Gaba in Neurons and Glial Cells

1 reference

12 December 2020

Cloning of the human homologue of the GABA transporter GAT-3 and identification of a novel inhibitor with selectivity for this site

1 reference

12 December 2020