(Q39168354)

English

Synthesis and evaluation of 3-amino/guanidine substituted phenyl oxazoles as a novel class of LSD1 inhibitors with anti-proliferative properties

scientific article published on 10 April 2013

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scholarly article

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Europe PubMed Central

PubMed publication ID

9 September 2017

Synthesis and evaluation of 3-amino/guanidine substituted phenyl oxazoles as a novel class of LSD1 inhibitors with anti-proliferative properties (English)

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

author name string

Balakrishna Dulla

1

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Krishna Tulasi Kirla

2

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Vandana Rathore

3

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Girdhar Singh Deora

4

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Sridhar Kavela

5

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Subbareddy Maddika

6

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Kiranam Chatti

7

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Oliver Reiser

8

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Javed Iqbal

9

1 reference

Europe PubMed Central

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9 September 2017

Manojit Pal

10

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9 September 2017

publication date

10 April 2013

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9 September 2017

Organic and Biomolecular Chemistry

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9 September 2017

11

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9 September 2017

19

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Europe PubMed Central

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9 September 2017

3103-3107

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

Role of histone modifications in defining chromatin structure and function

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Histone deacetylase inhibitor suberoylanilide hydroxamic acid induces apoptosis through both mitochondrial and Fas (Cd95) signaling in head and neck squamous carcinoma cells.

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Lysine-specific demethylase 1 (LSD1) Is required for the transcriptional repression of the telomerase reverse transcriptase (hTERT) gene

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

p53 is regulated by the lysine demethylase LSD1

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Cooperative demethylation by JMJD2C and LSD1 promotes androgen receptor-dependent gene expression

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Androgen receptor coactivators lysine-specific histone demethylase 1 and four and a half LIM domain protein 2 predict risk of prostate cancer recurrence

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Role of the lysine-specific demethylase 1 in the proinflammatory phenotype of vascular smooth muscle cells of diabetic mice

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Histone demethylation mediated by the nuclear amine oxidase homolog LSD1

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

LSD1 and the chemistry of histone demethylation

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Expanding chemical biology of 2-oxoglutarate oxygenases

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Mechanistic analysis of a suicide inactivator of histone demethylase LSD1

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Inhibition of lysine-specific demethylase 1 by polyamine analogues results in reexpression of aberrantly silenced genes

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Structural basis of LSD1-CoREST selectivity in histone H3 recognition

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Lysine demethylases inhibitors

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Oligoamine analogues in combination with 2-difluoromethylornithine synergistically induce re-expression of aberrantly silenced tumour-suppressor genes

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Facile synthesis of substituted trans-2-arylcyclopropylamine inhibitors of the human histone demethylase LSD1 and monoamine oxidases A and B.

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

A mechanism-based inactivator for histone demethylase LSD1.

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Comparative analysis of small molecules and histone substrate analogues as LSD1 lysine demethylase inhibitors

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Amide-substituted farnesylcysteine analogs as inhibitors of human isoprenylcysteine carboxyl methyltransferase

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Solid-Phase Synthesis of 7-Acylamino-1,4-benzodiazepine-2,5-diones

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Application of the Dakin-West reaction for the synthesis of oxazole-containing dual PPARalpha/gamma agonists

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Fluorescent pirenzepine derivatives as potential bitopic ligands of the human M1 muscarinic receptor

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Phase-transfer-catalyzed alkylation of guanidines by alkyl halides under biphasic conditions: a convenient protocol for the synthesis of highly functionalized guanidines.

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Zebrafish: a predictive model for assessing drug-induced toxicity

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Evolutionary history of histone demethylase families: distinct evolutionary patterns suggest functional divergence

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Brain-penetrant LSD1 inhibitors can block memory consolidation.

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Construction and functionalization of fused pyridine ring leading to novel compounds as potential antitubercular agents

1 reference

https://api.crossref.org/works/10.1039%2FC3OB40217G

21 January 2018

Identifiers

10.1039/C3OB40217G

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

9 September 2017

ResearchGate publication ID

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