(Q39370698)

English

Discovery of a novel alpha-7 nicotinic acetylcholine receptor agonist series and characterization of the potent, selective, and orally efficacious agonist 5-(4-acetyl[1,4]diazepan-1-yl)pentanoic acid [5-(4-methoxyphenyl)-1H-pyrazol-3-yl] amide (SEN1

scientific article

Statements

Discovery of a novel alpha-7 nicotinic acetylcholine receptor agonist series and characterization of the potent, selective, and orally efficacious agonist 5-(4-acetyl[1,4]diazepan-1-yl)pentanoic acid [5-(4-methoxyphenyl)-1H-pyrazol-3-yl] amide (SEN1 (English)
Riccardo Zanaletti
Laura Bettinetti
Cristiana Castaldo
Giuseppe Cocconcelli
Giovanni Gaviraghi
Arianna Nencini
Elisa Turlizzi
Michela Valacchi

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